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Volumn 59, Issue 5-6, 1996, Pages 449-457

RUI 58668: Further in vitro and in vivo pharmacological data related to its antitumoral activity

Author keywords

[No Author keywords available]

Indexed keywords

11 [4 [[5 [(4,4,5,5,5 PENTAFLUOROPENTYL)SULFONYL]PENTYL]OXY]PHENYL]ESTRADIOL; 4 HYDROXYTAMOXIFEN; ANTIESTROGEN; DOXORUBICIN; ESTRADIOL; FULVESTRANT; TAMOXIFEN; UNCLASSIFIED DRUG; ANTINEOPLASTIC AGENT; DRUG DERIVATIVE;

EID: 0030300130     PISSN: 09600760     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-0760(96)00140-9     Document Type: Article
Times cited : (30)

References (25)
  • 2
    • 0024456451 scopus 로고
    • Cytostatic effect of antiestrogens in lymphoid cells: Relationship to high affinity antiestrogen-binding sites and cholesterol
    • 2. Tang B. L., Teo C. C., Sim K. J., Ng M. L. and Kon O. N.: Cytostatic effect of antiestrogens in lymphoid cells: relationship to high affinity antiestrogen-binding sites and cholesterol. Biochim. Biophys. Acta 1014 (1989) 162-172.
    • (1989) Biochim. Biophys. Acta , vol.1014 , pp. 162-172
    • Tang, B.L.1    Teo, C.C.2    Sim, K.J.3    Ng, M.L.4    Kon, O.N.5
  • 3
    • 0026756472 scopus 로고
    • Tamoxifen as a single agent for advanced melanoma in postmenopausal women. A phase II study of the EORTC malignant melanoma cooperative group
    • 3. Rumke P., Kleeberg U. R., MacKie R. M., Lejeune F. J., Planting A. S., Brocker E. B., Bierhorst J. F. and Lentz M. A.: Tamoxifen as a single agent for advanced melanoma in postmenopausal women. A phase II study of the EORTC malignant melanoma cooperative group. Melanoma Res. 2 (1992) 153-156.
    • (1992) Melanoma Res. , vol.2 , pp. 153-156
    • Rumke, P.1    Kleeberg, U.R.2    MacKie, R.M.3    Lejeune, F.J.4    Planting, A.S.5    Brocker, E.B.6    Bierhorst, J.F.7    Lentz, M.A.8
  • 4
    • 0026672032 scopus 로고
    • The treatment of intracranial malignant gliomas using orally administered tamoxifen therapy: Preliminary results in a series of "failed" patients
    • 4. Vertosick F. t. Jr, Selker R. J., Pollack I. F. and Arena V.: The treatment of intracranial malignant gliomas using orally administered tamoxifen therapy: preliminary results in a series of "failed" patients. Neurosurgery 30 (1992) 897-903.
    • (1992) Neurosurgery , vol.30 , pp. 897-903
    • Vertosick F.T., Jr.1    Selker, R.J.2    Pollack, I.F.3    Arena, V.4
  • 7
    • 0023371203 scopus 로고
    • Tamoxifen therapy in unresectable adenocarcinoma of the pancreas
    • 7. Wong A., Chan A. and Arthur K.: Tamoxifen therapy in unresectable adenocarcinoma of the pancreas. Cancer Treat. Rep. 71 (1987) 749-750.
    • (1987) Cancer Treat. Rep. , vol.71 , pp. 749-750
    • Wong, A.1    Chan, A.2    Arthur, K.3
  • 8
    • 0025689160 scopus 로고
    • The only true antiestrogen is no estrogen
    • 8. Jordan V. C.: The only true antiestrogen is no estrogen. Molec. Cell. Endocr. 74 (1990) C91-C95.
    • (1990) Molec. Cell. Endocr. , vol.74
    • Jordan, V.C.1
  • 10
    • 0023760993 scopus 로고
    • Development of tamoxifen-stimulated growth of MCF-7 tumors in athymic mice after long-term antiestrogen administration
    • 10. Gottardis M. M. and Jordan V. C.: Development of tamoxifen-stimulated growth of MCF-7 tumors in athymic mice after long-term antiestrogen administration. Cancer Res. 48 (1988) 5183-5187.
    • (1988) Cancer Res. , vol.48 , pp. 5183-5187
    • Gottardis, M.M.1    Jordan, V.C.2
  • 12
    • 0026425624 scopus 로고
    • Growth factor messenger RNA expression by human breast fibroblasts from benign and malignant lesions
    • 12. Cullen K. J., Smith H. S., Hill S., Rosen N. and Lippman M. E.: Growth factor messenger RNA expression by human breast fibroblasts from benign and malignant lesions. Cancer Res. 51 (1991) 4978-4985.
    • (1991) Cancer Res. , vol.51 , pp. 4978-4985
    • Cullen, K.J.1    Smith, H.S.2    Hill, S.3    Rosen, N.4    Lippman, M.E.5
  • 13
    • 0022485353 scopus 로고
    • Estrogen-induced factors of breast cancer cells partially replace estrogen to promote tumor growth
    • 13. Dickson B. D., McManaway M. E. and Lippman M. E.: Estrogen-induced factors of breast cancer cells partially replace estrogen to promote tumor growth. Science 232 (1986) 1540-1542.
    • (1986) Science , vol.232 , pp. 1540-1542
    • Dickson, B.D.1    McManaway, M.E.2    Lippman, M.E.3
  • 14
    • 0026395885 scopus 로고
    • A potent specific pure antiestrogen with clinical potential
    • 14. Wakeling A. E., Dukes M. and Bowler J.: A potent specific pure antiestrogen with clinical potential. Cancer Res. 51 (1991) 3867-3873.
    • (1991) Cancer Res. , vol.51 , pp. 3867-3873
    • Wakeling, A.E.1    Dukes, M.2    Bowler, J.3
  • 16
    • 0024539364 scopus 로고
    • Effect of tamoxifen on plasma insulin-like growth factor I in patients with breast cancer
    • 16. Colletti R. B., Roberts J. D., Devlin J. T. and Copeland K. C.: Effect of tamoxifen on plasma insulin-like growth factor I in patients with breast cancer. Cancer Res. 49 (1989) 1882-1884.
    • (1989) Cancer Res. , vol.49 , pp. 1882-1884
    • Colletti, R.B.1    Roberts, J.D.2    Devlin, J.T.3    Copeland, K.C.4
  • 17
    • 0023701360 scopus 로고
    • Novel antioestrogens without partial agonist activity
    • 17. Wakeling A. E. and Bowler J.: Novel antioestrogens without partial agonist activity. J. Steroid. Biochem. 31 (1988) 645-653.
    • (1988) J. Steroid. Biochem. , vol.31 , pp. 645-653
    • Wakeling, A.E.1    Bowler, J.2
  • 18
    • 0025615574 scopus 로고
    • Therapeutic potential of pure antiestrogens in the treatment of breast cancer
    • 18. Wakeling A. E.: Therapeutic potential of pure antiestrogens in the treatment of breast cancer. J. Steroid Biochem. Molec. Biol. 37 (1990) 771-775.
    • (1990) J. Steroid Biochem. Molec. Biol. , vol.37 , pp. 771-775
    • Wakeling, A.E.1
  • 20
    • 4243559560 scopus 로고
    • Investigation of a pure antioestrogen (ICI 182,780) in tamoxifen resistant breast cancer
    • 20. Howell A., Defriend D. J., Blamey R. W., Robertson J. F. and Walton P. J.: Investigation of a pure antioestrogen (ICI 182,780) in tamoxifen resistant breast cancer. Eur. J. Cancer 30A (1994) S24.
    • (1994) Eur. J. Cancer , vol.30 A
    • Howell, A.1    Defriend, D.J.2    Blamey, R.W.3    Robertson, J.F.4    Walton, P.J.5
  • 21
  • 22
    • 0028215513 scopus 로고
    • RU 58668: Profil des activités pharmacologiques d'un nouvel antiestrogène pur susceptible de traiter certains échappements au tamoxifène
    • 22. Van de Velde P., Nique F., Brémaud J., Delettre G., Hameau M. C., Lucas D., Moratille C., Philibert D. and Teutsch G.: RU 58668: Profil des activités pharmacologiques d'un nouvel antiestrogène pur susceptible de traiter certains échappements au tamoxifène. Pathol. Biol. 42 (1994) 30.
    • (1994) Pathol. Biol. , vol.42 , pp. 30
    • Van De Velde, P.1    Nique, F.2    Brémaud, J.3    Delettre, G.4    Hameau, M.C.5    Lucas, D.6    Moratille, C.7    Philibert, D.8    Teutsch, G.9
  • 24
    • 0023784250 scopus 로고
    • Application of bromodeoxyuridine incorporation measurements to the determination of cell distribution within the S-phase of the cell cycle
    • 24. Khochbin S., Chabanas A., Albert P., Albert J. and Laurence J. J.: Application of bromodeoxyuridine incorporation measurements to the determination of cell distribution within the S-phase of the cell cycle. Cytometry 9 (1988) 499-503.
    • (1988) Cytometry , vol.9 , pp. 499-503
    • Khochbin, S.1    Chabanas, A.2    Albert, P.3    Albert, J.4    Laurence, J.J.5
  • 25
    • 0025064215 scopus 로고
    • Growth properties and tumorigenesis of MCF-7 cells transfected with isogenic mutant of ras
    • 25. Sommers C. L., Papageorge A., Wilding G. and Gelmann P.: Growth properties and tumorigenesis of MCF-7 cells transfected with isogenic mutant of ras. Cancer Res. 50 (1990) 67-71.
    • (1990) Cancer Res. , vol.50 , pp. 67-71
    • Sommers, C.L.1    Papageorge, A.2    Wilding, G.3    Gelmann, P.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.