Two distinct α1-adrenoceptor subtypes in the human prostate: Assessment by radioligand binding assay using 31H-prazosin

General Pharmacology

Volumn 27, Issue 8, 1996, Pages 1377-1381

  Maruyama, Keiko ^a   Fukutomi, Junya ^a   Chiba, Takako ^a   Yamaguchi, Machiko ^a   Takeda, Masayuki ^b   Hattori, Kaoru ^a   Nagatomo, Takafumi ^a  

^a NIIGATA UNIVERSITY OF PHARMACY AND APPLIED LIFE SCIENCES   (Japan)

^b NIIGATA UNIVERSITY   (Japan)

Author keywords

1 adrenoceptor subtype; 3H prazosin; human prostate; radioligand binding assay

Indexed keywords

2 [[2 (2,6 DIMETHOXYPHENOXY)ETHYL]AMINOMETHYL] 1,4 BENZODIOXAN; 5 METHYLURAPIDIL; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA 1C ADRENERGIC RECEPTOR; ALPHA 1H ADRENERGIC RECEPTOR; ALPHA 1L ADRENERGIC RECEPTOR; ALPHA ETHYL 3,4,5 TRIMETHOXY ALPHA [3 [[2 (2 METHOXYPHENOXY)ETHYL]AMINO]PROPYL]BENZENEACETONITRILE FUMARATE; CHLOROETHYLCLONIDINE; NIFEDIPINE; NIGULDIPINE; PHENOXYBENZAMINE; PHENTOLAMINE; PRAZOSIN; RADIOLIGAND; RECEPTOR SUBTYPE; TAMSULOSIN; TERAZOSIN; UNCLASSIFIED DRUG; 5-METHYLURAPIDIL; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; DIOXANE DERIVATIVE; DRUG DERIVATIVE; PIPERAZINE DERIVATIVE; SULFONAMIDE; TERAZOSINE; TRITIUM;

ARTICLE; BINDING AFFINITY; BINDING COMPETITION; CELL MEMBRANE; CONTROLLED STUDY; HUMAN; HUMAN TISSUE; LIGAND BINDING; MALE; MOLECULAR CLONING; PRIORITY JOURNAL; PROSTATE; RECEPTOR BINDING; CHEMISTRY; CLASSIFICATION; DRUG ANTAGONISM; DRUG EFFECT; IN VITRO STUDY; KINETICS; METABOLISM; PROTEIN BINDING; RADIOASSAY;

ADRENERGIC ALPHA-ANTAGONISTS; BINDING, COMPETITIVE; DIOXANES; HUMANS; KINETICS; MALE; NIFEDIPINE; PHENTOLAMINE; PIPERAZINES; PRAZOSIN; PROSTATE; PROTEIN BINDING; RADIOLIGAND ASSAY; RECEPTORS, ADRENERGIC, ALPHA-1; SULFONAMIDES; TRITIUM;

EID: 0030299076     PISSN: 03063623     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0306-3623(96)00071-7     Document Type: Article

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