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Volumn 140, Issue 1, 1996, Pages 124-130

Prediction of furan pharmacokinetics from hepatocyte studies: Comparison of bioactivation and hepatic dosimetry in rats, mice, and humans'

Author keywords

[No Author keywords available]

Indexed keywords

CYTOCHROME P450; FURAN;

EID: 0030246901     PISSN: 0041008X     EISSN: None     Source Type: Journal    
DOI: 10.1006/taap.1996.0205     Document Type: Article
Times cited : (75)

References (38)
  • 2
    • 85030272698 scopus 로고
    • Reference Physiological Parameters in Pharmacokinetic Modeling. US EPA/600/6-88/004, Final Report, NTIS, PB88-196019
    • Arms, A. D., and Travis, C. C. (1988). Reference Physiological Parameters in Pharmacokinetic Modeling. US EPA/600/6-88/004, Final Report, NTIS, PB88-196019.
    • (1988)
    • Arms, A.D.1    Travis, C.C.2
  • 3
    • 0025689878 scopus 로고
    • Prediction of intrinsic clearance of loxtidine from kinetic studies in rat, dog and human hepatocytes
    • Bayliss, M. K., Bell, J. A., Jenner, W. N., and Wilson, K. (1990). Prediction of intrinsic clearance of loxtidine from kinetic studies in rat, dog and human hepatocytes. Biochem. Soc. Trans. 18, 1198-1199.
    • (1990) Biochem. Soc. Trans. , vol.18 , pp. 1198-1199
    • Bayliss, M.K.1    Bell, J.A.2    Jenner, W.N.3    Wilson, K.4
  • 4
    • 0017609420 scopus 로고
    • The metabolism of drugs in isolated rat hepatocytes: A comparison with in vivo drug metabolism and drug metabolism in subcellular liver fractions
    • Billings, R. E., McMahon, R. E., Ashmore, J., and Wagle, S. R. (1977). The metabolism of drugs in isolated rat hepatocytes: A comparison with in vivo drug metabolism and drug metabolism in subcellular liver fractions. Drug Metab. Dispos. 5, 518-526.
    • (1977) Drug Metab. Dispos. , vol.5 , pp. 518-526
    • Billings, R.E.1    McMahon, R.E.2    Ashmore, J.3    Wagle, S.R.4
  • 6
    • 0027377274 scopus 로고
    • Furan-induced cytolethality in isolated rat hepatocytes: Correspondence with in vivo dosimetry
    • Carfagna, M. A., Held, S. D., and Kedderis, G. L. (1993). Furan-induced cytolethality in isolated rat hepatocytes: Correspondence with in vivo dosimetry. Toxicol. Appl. Pharmacol. 123, 265-273.
    • (1993) Toxicol. Appl. Pharmacol. , vol.123 , pp. 265-273
    • Carfagna, M.A.1    Held, S.D.2    Kedderis, G.L.3
  • 7
    • 0028785113 scopus 로고
    • Identification of cis-2-butene-1,4-dial as a microsomal metabolite of furan
    • Chen, L.-J., Hecht, S. S., and Peterson, L. A. (1995). Identification of cis-2-butene-1,4-dial as a microsomal metabolite of furan. Chem. Res. Toxicol. 8, 903-906.
    • (1995) Chem. Res. Toxicol. , vol.8 , pp. 903-906
    • Chen, L.-J.1    Hecht, S.S.2    Peterson, L.A.3
  • 9
    • 0015925332 scopus 로고
    • Blood flow limitations in interpreting Michaelis constants for ethanol oxidation in vivo
    • Dedrick, R. L., and Forrester, D. D. (1973). Blood flow limitations in interpreting Michaelis constants for ethanol oxidation in vivo. Biochem. Pharmacol. 22, 1133-1140.
    • (1973) Biochem. Pharmacol. , vol.22 , pp. 1133-1140
    • Dedrick, R.L.1    Forrester, D.D.2
  • 10
    • 0022335175 scopus 로고
    • Species differences in carcinogenicity and peroxisome proliferation due to trichloroethylene: A biochemical human hazard assessment
    • Elcombe, C. R. (1985). Species differences in carcinogenicity and peroxisome proliferation due to trichloroethylene: A biochemical human hazard assessment. Arch. Toxicol. (Suppl. 8), 6-17.
    • (1985) Arch. Toxicol. , Issue.SUPPL. 8 , pp. 6-17
    • Elcombe, C.R.1
  • 11
    • 0022872403 scopus 로고
    • A physiologically based simulation approach for determining metabolic constants from gas uptake data
    • Gargas, M. L., Andersen, M. E., and Clewell, H. J., III (1986a). A physiologically based simulation approach for determining metabolic constants from gas uptake data. Toxicol. Appl. Pharmacol. 86, 341-352.
    • (1986) Toxicol. Appl. Pharmacol. , vol.86 , pp. 341-352
    • Gargas, M.L.1    Andersen, M.E.2    Clewell H.J. III3
  • 12
    • 0022656857 scopus 로고
    • Metabolism of inhaled dihalomethanes in vivo: Differentiation of kinetic constants for two independent pathways
    • Gargas, M. L., Clewell, H. J., III, and Andersen, M. E. (1986b). Metabolism of inhaled dihalomethanes in vivo: Differentiation of kinetic constants for two independent pathways. Toxicol. Appl. Pharmacol. 82, 211-223.
    • (1986) Toxicol. Appl. Pharmacol. , vol.82 , pp. 211-223
    • Gargas, M.L.1    Clewell H.J. III2    Andersen, M.E.3
  • 13
    • 0024524118 scopus 로고
    • Partition coefficients of low-molecular-weight volatile chemicals in various liquids and tissues
    • Gargas, M. L., Burgess, R. J., Voisard, D. E., Cason, G. H., and Andersen, M. E. (1989). Partition coefficients of low-molecular-weight volatile chemicals in various liquids and tissues. Toxicol. Appl. Pharmacol. 98, 87-99.
    • (1989) Toxicol. Appl. Pharmacol. , vol.98 , pp. 87-99
    • Gargas, M.L.1    Burgess, R.J.2    Voisard, D.E.3    Cason, G.H.4    Andersen, M.E.5
  • 14
    • 0022506192 scopus 로고
    • Comparison of amphetamine metabolism using isolated hepatocytes from five species including human
    • Green, C. E., LeValley, S. E., and Tyson, C. A. (1986). Comparison of amphetamine metabolism using isolated hepatocytes from five species including human. J. Pharmacol. Exp. Ther. 237, 931-936.
    • (1986) J. Pharmacol. Exp. Ther. , vol.237 , pp. 931-936
    • Green, C.E.1    LeValley, S.E.2    Tyson, C.A.3
  • 15
    • 0026035519 scopus 로고
    • Role of human cytochrome P450 IIE1 in the oxidation of many low molecular weight cancer suspects
    • Guengerich, F. P., Kim, D.-H., and Iwasaki, M. (1991). Role of human cytochrome P450 IIE1 in the oxidation of many low molecular weight cancer suspects. Chem. Res. Toxicol. 4, 168-179.
    • (1991) Chem. Res. Toxicol. , vol.4 , pp. 168-179
    • Guengerich, F.P.1    Kim, D.-H.2    Iwasaki, M.3
  • 16
    • 0028342648 scopus 로고
    • Utility of in vitro drug metabolism data in predicting in vivo metabolic clearance
    • Houston, J. B. (1994). Utility of in vitro drug metabolism data in predicting in vivo metabolic clearance. Biochem. Pharmacol. 47, 1469-1479.
    • (1994) Biochem. Pharmacol. , vol.47 , pp. 1469-1479
    • Houston, J.B.1
  • 17
    • 74049148466 scopus 로고    scopus 로고
    • Hepatic blood flow limitation of the bioactivation of hazardous chemical air pollutants
    • Kedderis, G. L. (1996). Hepatic blood flow limitation of the bioactivation of hazardous chemical air pollutants. Fundam. Appl. Toxicol. 30, 34-35.
    • (1996) Fundam. Appl. Toxicol. , vol.30 , pp. 34-35
    • Kedderis, G.L.1
  • 18
    • 0023891002 scopus 로고
    • Studies with nitrogen-containing steroids and freshly isolated rat hepatocytes: Role of cytochrome P450 in detoxication
    • Kedderis, G. L., Argenbright, L. S., and Miwa, G. T. (1988). Studies with nitrogen-containing steroids and freshly isolated rat hepatocytes: Role of cytochrome P450 in detoxication. Toxicol. Appl. Pharmacol. 93, 403-412.
    • (1988) Toxicol. Appl. Pharmacol. , vol.93 , pp. 403-412
    • Kedderis, G.L.1    Argenbright, L.S.2    Miwa, G.T.3
  • 20
    • 0028586025 scopus 로고
    • Metabolic disposition of tacrine in primary suspensions of rat hepatocytes and in single-pass perfused liver: In vitro/in vivo comparisons
    • Kukan, M., Bezek, S., Pool, W. F., and Woolf, T. F. (1994). Metabolic disposition of tacrine in primary suspensions of rat hepatocytes and in single-pass perfused liver: In vitro/in vivo comparisons. Xenobiotica 24, 1107-1117.
    • (1994) Xenobiotica , vol.24 , pp. 1107-1117
    • Kukan, M.1    Bezek, S.2    Pool, W.F.3    Woolf, T.F.4
  • 21
    • 0023811891 scopus 로고
    • Inhibition of taurocholate transport by cyclosporin A in cultured rat hepatocytes
    • Kukongviriyapan, V., and Stacey, N. H. (1988). Inhibition of taurocholate transport by cyclosporin A in cultured rat hepatocytes. J. Pharmacol. Exp. Ther. 247, 685-689.
    • (1988) J. Pharmacol. Exp. Ther. , vol.247 , pp. 685-689
    • Kukongviriyapan, V.1    Stacey, N.H.2
  • 23
    • 0020279521 scopus 로고
    • Physiological pharmacokinetics of ethoxybenzamide based on biochemical data obtained in vitro as well as on physiological data
    • Lin, J. H., Sugiyama, Y., Awazu, S., and Hanano, M. (1982). Physiological pharmacokinetics of ethoxybenzamide based on biochemical data obtained in vitro as well as on physiological data. J. Pharmacokin. Biopharm. 10, 649-661.
    • (1982) J. Pharmacokin. Biopharm. , vol.10 , pp. 649-661
    • Lin, J.H.1    Sugiyama, Y.2    Awazu, S.3    Hanano, M.4
  • 25
    • 0021203649 scopus 로고
    • The effects of diethyldithiocarbamate and carbon disulfide on acute nephrotoxicity induced by furan, bromobenzene and cephaloridine in mice
    • Masuda, Y., Nakayama, N., Yamaguchi, A., and Murohashi, M. (1984). The effects of diethyldithiocarbamate and carbon disulfide on acute nephrotoxicity induced by furan, bromobenzene and cephaloridine in mice. Jpn. J. Pharmacol. 34, 221-229.
    • (1984) Jpn. J. Pharmacol. , vol.34 , pp. 221-229
    • Masuda, Y.1    Nakayama, N.2    Yamaguchi, A.3    Murohashi, M.4
  • 26
    • 0023033053 scopus 로고
    • Man versus beast: Pharmacokinetic scaling in mammals
    • Mordenti, J. (1986). Man versus beast: Pharmacokinetic scaling in mammals. J. Pharm. Sci. 75, 1028-1040.
    • (1986) J. Pharm. Sci. , vol.75 , pp. 1028-1040
    • Mordenti, J.1
  • 27
    • 0022458177 scopus 로고
    • Salmonella mutagenicity tests. II. Results from the testing of 270 chemicals
    • Mortelmans, K., Haworth, S., Lawlor, T., Speck, W., Tainer, B., and Zeiger, E. (1986). Salmonella mutagenicity tests. II. Results from the testing of 270 chemicals. Environ. Mutagen. (Suppl. 7), 1-119.
    • (1986) Environ. Mutagen. , Issue.SUPPL. 7 , pp. 1-119
    • Mortelmans, K.1    Haworth, S.2    Lawlor, T.3    Speck, W.4    Tainer, B.5    Zeiger, E.6
  • 28
    • 0003541547 scopus 로고
    • Toxicology and Carcinogenesis Studies of Furan in F-344/N Rats and B6C3F1 Mice
    • U.S. Dept. of Health and Human Services, Public Health Service, National Institutes of Health, Research Triangle Park, NC
    • National Toxicology Program (1993). Toxicology and Carcinogenesis Studies of Furan in F-344/N Rats and B6C3F1 Mice. NTP Technical Report 402, U.S. Dept. of Health and Human Services, Public Health Service, National Institutes of Health, Research Triangle Park, NC.
    • (1993) NTP Technical Report , pp. 402
  • 29
    • 0021104396 scopus 로고
    • Fitting enzyme-kinetic data to V/K
    • Northrop, D. B. (1983). Fitting enzyme-kinetic data to V/K. Anal. Biochem. 132, 457-461.
    • (1983) Anal. Biochem. , vol.132 , pp. 457-461
    • Northrop, D.B.1
  • 31
    • 0024832058 scopus 로고
    • Modulation of cytochrome P450 isozymes in human liver by ethanol and drug intake
    • Perrot, N., Nalpas, B., Yang, C. S., and Beaune, P. H. (1989). Modulation of cytochrome P450 isozymes in human liver by ethanol and drug intake. Eur. J. Clin. Invest. 19, 549-555.
    • (1989) Eur. J. Clin. Invest. , vol.19 , pp. 549-555
    • Perrot, N.1    Nalpas, B.2    Yang, C.S.3    Beaune, P.H.4
  • 32
    • 0027476657 scopus 로고
    • Bioactivation of halogenated hydrocarbons by cytochrome P4502E1
    • Raucy, J. L., Kraner, J. C., and Lasker, J. M. (1993). Bioactivation of halogenated hydrocarbons by cytochrome P4502E1. Crit. Rev. Toxicol. 23, 1-20.
    • (1993) Crit. Rev. Toxicol. , vol.23 , pp. 1-20
    • Raucy, J.L.1    Kraner, J.C.2    Lasker, J.M.3
  • 33
    • 0024510208 scopus 로고
    • Comparative drug metabolism of diazepam in hepatocytes isolated from man, rat, monkey and dog
    • Seddon, T., Michelle, I., and Chenery, R. J. (1989). Comparative drug metabolism of diazepam in hepatocytes isolated from man, rat, monkey and dog. Biochem. Pharmacol. 38, 1657-1665.
    • (1989) Biochem. Pharmacol. , vol.38 , pp. 1657-1665
    • Seddon, T.1    Michelle, I.2    Chenery, R.J.3
  • 34
    • 0017101039 scopus 로고
    • Preparation of isolated rat liver cells
    • Seglen, P. O. (1976). Preparation of isolated rat liver cells. Methods Cell Biol. 13, 29-83.
    • (1976) Methods Cell Biol. , vol.13 , pp. 29-83
    • Seglen, P.O.1
  • 35
    • 0026050247 scopus 로고
    • Determination of in vivo hepatic extraction ratio from in vitro metabolism by rat hepatocytes
    • Singh, K., Tripp, S. L., Dunton, A. W., Douglas, F. L., and Rakhit, A. (1991). Determination of in vivo hepatic extraction ratio from in vitro metabolism by rat hepatocytes. Drug Metab. Dispos. 19, 990-996.
    • (1991) Drug Metab. Dispos. , vol.19 , pp. 990-996
    • Singh, K.1    Tripp, S.L.2    Dunton, A.W.3    Douglas, F.L.4    Rakhit, A.5
  • 37
    • 0000920633 scopus 로고
    • Ventilation-perfusion relationships
    • (R. G. Crystal and J. B. West, Eds.) . Raven Press, New York
    • West, J. B., and Wagner, P. D. (1991). Ventilation-perfusion relationships. In The Lung: Scientific Foundations (R. G. Crystal and J. B. West, Eds.), Vol. 2, pp. 1289-1305. Raven Press, New York.
    • (1991) The Lung: Scientific Foundations , vol.2 , pp. 1289-1305
    • West, J.B.1    Wagner, P.D.2
  • 38
    • 0026603074 scopus 로고
    • Evaluation of genotoxicity, pathological lesions and cell proliferation in livers of rats and mice treated with furan
    • Wilson, D. M., Goldsworthy, T. L., Popp, J. A., and Butterworth, B. E. (1992). Evaluation of genotoxicity, pathological lesions and cell proliferation in livers of rats and mice treated with furan. Environ. Mol. Mutagen. 19, 209-222.
    • (1992) Environ. Mol. Mutagen. , vol.19 , pp. 209-222
    • Wilson, D.M.1    Goldsworthy, T.L.2    Popp, J.A.3    Butterworth, B.E.4


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