Tyrphostins IV - Highly potent inhibitors of EGF receptor kinase. Structure-activity relationship study of 4-anilidoquinazolines

Bioorganic and Medicinal Chemistry

Volumn 4, Issue 8, 1996, Pages 1203-1207

  Gazit, Aviv ^a   Chen, Jeffrey ^b   Harald, App ^b   McMahon, Gerald ^b   Hirth, Peter ^b   Chen, Irit ^a   Levitzki, Alexander ^a  

^a HEBREW UNIVERSITY OF JERUSALEM   (Israel)

^b SUGEN INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ENZYME INHIBITOR; EPIDERMAL GROWTH FACTOR RECEPTOR; EPIDERMAL GROWTH FACTOR RECEPTOR KINASE; QUINAZOLINE DERIVATIVE; TYRPHOSTIN;

ARTICLE; AUTOPHOSPHORYLATION; CELL MEMBRANE; CONTROLLED STUDY; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; HUMAN CELL; IN VITRO STUDY; STRUCTURE ACTIVITY RELATION;

EID: 0030220783     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/0968-0896(96)00107-1     Document Type: Article

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