메뉴 건너뛰기




Volumn 139, Issue 2, 1996, Pages 243-251

Use of the vial equilibration technique for determination of metabolic rate constants for dichloromethane

Author keywords

[No Author keywords available]

Indexed keywords

CYTOCHROME P450 ISOENZYME; DICHLOROMETHANE;

EID: 0030220583     PISSN: 0041008X     EISSN: None     Source Type: Journal    
DOI: 10.1006/taap.1996.0163     Document Type: Article
Times cited : (12)

References (36)
  • 1
    • 0018090905 scopus 로고
    • Inhibition and enhancement of microsomal drug metabolism by diethyl maleate
    • Anders, M. W. (1978). Inhibition and enhancement of microsomal drug metabolism by diethyl maleate. Biochem. Pharmacol. 27, 1098-1101.
    • (1978) Biochem. Pharmacol. , vol.27 , pp. 1098-1101
    • Anders, M.W.1
  • 2
    • 0017551374 scopus 로고
    • Metabolism of halogenated methanes and macromolecular binding
    • Anders, M. W., Kubic, V. L., and Ahmed, A. E. (1977). Metabolism of halogenated methanes and macromolecular binding. J. Environ. Pathol. Toxicol. 1, 117-124.
    • (1977) J. Environ. Pathol. Toxicol. , vol.1 , pp. 117-124
    • Anders, M.W.1    Kubic, V.L.2    Ahmed, A.E.3
  • 3
    • 0023158895 scopus 로고
    • Physiologically based pharmacokinetics and the risk assessment process for methylene chloride
    • Andersen, M. E., Clewell, H. J., III, Gargas, M. L., Smith, F. A., and Reitz, R. H. (1987). Physiologically based pharmacokinetics and the risk assessment process for methylene chloride. Toxicol. Appl. Pharmacol. 87, 185-205.
    • (1987) Toxicol. Appl. Pharmacol. , vol.87 , pp. 185-205
    • Andersen, M.E.1    Clewell H.J. III2    Gargas, M.L.3    Smith, F.A.4    Reitz, R.H.5
  • 4
    • 0025981543 scopus 로고
    • Physiologically based pharmacokinetic modeling with dichloromethane, its metabolite, carbon monoxide, and blood carboxyhemoglobin in rats and humans
    • Andersen, M. E., Clewell, H. J., III., Gargas, M. L., MacNaughton, M. G., Reitz, R. H., Nolan, R. J., and McKenna, M. J. (1991). Physiologically based pharmacokinetic modeling with dichloromethane, its metabolite, carbon monoxide, and blood carboxyhemoglobin in rats and humans. Toxicol. Appl. Pharmacol. 108, 14-27.
    • (1991) Toxicol. Appl. Pharmacol. , vol.108 , pp. 14-27
    • Andersen, M.E.1    Clewell H.J. III2    Gargas, M.L.3    MacNaughton, M.G.4    Reitz, R.H.5    Nolan, R.J.6    McKenna, M.J.7
  • 5
    • 0004330014 scopus 로고
    • TP-92/13, Agency for Toxic Substances and Disease Registry, U.S. Public Health Service, Atlanta, GA
    • ATSDR (1993). Toxicological Profile for Methylene Chloride. TP-92/13, Agency for Toxic Substances and Disease Registry, U.S. Public Health Service, Atlanta, GA.
    • (1993) Toxicological Profile for Methylene Chloride
  • 7
    • 0025239050 scopus 로고
    • Oxidation of pyrazole by reconstituted systems containing cytochrome P-450 IIE1
    • Clejan, L. A., and Cederbaum, A. I. (1990). Oxidation of pyrazole by reconstituted systems containing cytochrome P-450 IIE1. Biochem. Biophys. Acta 1034, 233-237.
    • (1990) Biochem. Biophys. Acta , vol.1034 , pp. 233-237
    • Clejan, L.A.1    Cederbaum, A.I.2
  • 8
    • 0022656857 scopus 로고
    • Metabolism of inhaled dichloromethane in vivo: Differentiation of kinetic constants for two independent pathways
    • Gargas, M. L., Clewell, H. J., III, and Andersen, M. E. (1986). Metabolism of inhaled dichloromethane in vivo: Differentiation of kinetic constants for two independent pathways. Toxicol. Appl. Pharmacol. 82, 211-223.
    • (1986) Toxicol. Appl. Pharmacol. , vol.82 , pp. 211-223
    • Gargas, M.L.1    Clewell H.J. III2    Andersen, M.E.3
  • 9
    • 0024524118 scopus 로고
    • Partition coefficients of low-molecular-weight volatile chemicals in various liquids and tissues
    • Gargas, M. L., Burgess, R. J., Voisard, D. E., Cason, G. H., and Andersen, M. E. (1989). Partition coefficients of low-molecular-weight volatile chemicals in various liquids and tissues. Toxicol. Appl. Pharmacol. 98, 87-99.
    • (1989) Toxicol. Appl. Pharmacol. , vol.98 , pp. 87-99
    • Gargas, M.L.1    Burgess, R.J.2    Voisard, D.E.3    Cason, G.H.4    Andersen, M.E.5
  • 10
    • 0026035519 scopus 로고
    • Role of human cytochrome P-450 IIE1 in the oxidation of many low molecular weight cancer suspects
    • Guengerich, F. P., Kim, D.-H., and Iwasaki, M. (1991). Role of human cytochrome P-450 IIE1 in the oxidation of many low molecular weight cancer suspects. Chem. Res. Toxicol. 4, 168-179.
    • (1991) Chem. Res. Toxicol. , vol.4 , pp. 168-179
    • Guengerich, F.P.1    Kim, D.-H.2    Iwasaki, M.3
  • 11
    • 0001567332 scopus 로고
    • Glutathione S-transferase: The first enzymatic step in mercapturic acid formation
    • Habig, W. H., Pabst, M. J., and Jakoby, W. B. (1974). Glutathione S-transferase: The first enzymatic step in mercapturic acid formation. J. Biol. Chem. 19, 1-20.
    • (1974) J. Biol. Chem. , vol.19 , pp. 1-20
    • Habig, W.H.1    Pabst, M.J.2    Jakoby, W.B.3
  • 12
    • 0025356936 scopus 로고
    • Regional distribution of ethanol-inducible cytochrome P-450 IIE1 in the rat central nervous system
    • Hansson, T., Tindberg, N., Ingelman-Sundberg, M., and Kohler, C. (1990). Regional distribution of ethanol-inducible cytochrome P-450 IIE1 in the rat central nervous system. Neuroscience 34, 451-463.
    • (1990) Neuroscience , vol.34 , pp. 451-463
    • Hansson, T.1    Tindberg, N.2    Ingelman-Sundberg, M.3    Kohler, C.4
  • 13
    • 0026004357 scopus 로고
    • Sensitivity analysis for physiologically based pharmacokinetic models
    • Hetrick, D. M., Jarabek, A. M., and Travis, C. C. (1991). Sensitivity analysis for physiologically based pharmacokinetic models. J. Pharmacokin. Biopharm. 19, 1-20.
    • (1991) J. Pharmacokin. Biopharm. , vol.19 , pp. 1-20
    • Hetrick, D.M.1    Jarabek, A.M.2    Travis, C.C.3
  • 14
    • 0026567713 scopus 로고
    • Oxidative and reductive metabolism by cytochrome P-450 2E1
    • Koop, D. R. (1992). Oxidative and reductive metabolism by cytochrome P-450 2E1. FASEB J. 6, 724-730.
    • (1992) FASEB J. , vol.6 , pp. 724-730
    • Koop, D.R.1
  • 15
    • 0021806780 scopus 로고
    • Immunochemical evidence for induction of the alcohol-oxidizing cytochrome P-450 of rabbit liver microsomes by diverse agents: Ethanol, imidazole, trichloroethylene, acetone, pyrazole, and isoniazid
    • Koop, D. R., Crump, B. L., Nordblom, G. D., and Coon, M. J. (1985). Immunochemical evidence for induction of the alcohol-oxidizing cytochrome P-450 of rabbit liver microsomes by diverse agents: Ethanol, imidazole, trichloroethylene, acetone, pyrazole, and isoniazid. Proc. Natl. Acad. Sci. 82, 4065-4069.
    • (1985) Proc. Natl. Acad. Sci. , vol.82 , pp. 4065-4069
    • Koop, D.R.1    Crump, B.L.2    Nordblom, G.D.3    Coon, M.J.4
  • 16
    • 0018085060 scopus 로고
    • Metabolism of dihalomethane to carbon monoxide. Studies on the mechanism of the reaction
    • Kubic, V. L., and Anders, M. W. (1978). Metabolism of dihalomethane to carbon monoxide. Studies on the mechanism of the reaction. Biochem. Pharmacol. 27, 2349-2355.
    • (1978) Biochem. Pharmacol. , vol.27 , pp. 2349-2355
    • Kubic, V.L.1    Anders, M.W.2
  • 17
    • 33751330608 scopus 로고
    • The determination of enzyme dissociation constants
    • Lineweaver, H., and Burk, D. (1934). The determination of enzyme dissociation constants. J. Am. Chem. Soc. 56, 658-666.
    • (1934) J. Am. Chem. Soc. , vol.56 , pp. 658-666
    • Lineweaver, H.1    Burk, D.2
  • 18
    • 0021261696 scopus 로고
    • Drug metabolism in man and its relationship to that in three rodent species: Monooxygenase, epoxide hydrolyase, and glutathione S-transferase activities in subcellular fractions of lung and liver
    • Lorenz, J., Glatt, H. R., Fleischmann, R., Ferlinz, R., and Oesch, F. (1984). Drug metabolism in man and its relationship to that in three rodent species: Monooxygenase, epoxide hydrolyase, and glutathione S-transferase activities in subcellular fractions of lung and liver. Biochem. Med. 32, 43-56.
    • (1984) Biochem. Med. , vol.32 , pp. 43-56
    • Lorenz, J.1    Glatt, H.R.2    Fleischmann, R.3    Ferlinz, R.4    Oesch, F.5
  • 21
    • 0023943088 scopus 로고
    • Complexation of cytochrome P-450 isozymes in hepatic microsomes from SKF-525A-induced rats
    • Murray, M. (1988). Complexation of cytochrome P-450 isozymes in hepatic microsomes from SKF-525A-induced rats. Arch. Biochem. Biophys. 262, 381-388.
    • (1988) Arch. Biochem. Biophys. , vol.262 , pp. 381-388
    • Murray, M.1
  • 22
    • 0014629497 scopus 로고
    • Kinetic experiments on the binding of metyrapone to liver microsomes
    • Netter, K. J., Kahl, G.-F., and Magnussen, M. P. (1969). Kinetic experiments on the binding of metyrapone to liver microsomes. Naunyn-Schm. Arch. Pharmakol. 265, 205-215.
    • (1969) Naunyn-Schm. Arch. Pharmakol. , vol.265 , pp. 205-215
    • Netter, K.J.1    Kahl, G.-F.2    Magnussen, M.P.3
  • 23
    • 78651165715 scopus 로고
    • The carbon monoxide-binding pigment of liver microsomes
    • Omura, T., and Sato, R. (1964). The carbon monoxide-binding pigment of liver microsomes. J. Biol. Chem. 239, 2370-2378.
    • (1964) J. Biol. Chem. , vol.239 , pp. 2370-2378
    • Omura, T.1    Sato, R.2
  • 24
    • 0017818061 scopus 로고
    • Modeling the uptake, metabolism and excretion of dichloromethane by man
    • Peterson, J. E. (1975). Modeling the uptake, metabolism and excretion of dichloromethane by man. Am. Ind. Hyg. Assoc. J. 39, 41-47.
    • (1975) Am. Ind. Hyg. Assoc. J. , vol.39 , pp. 41-47
    • Peterson, J.E.1
  • 25
    • 0023751819 scopus 로고
    • Incorporation of in vitro enzyme data into the physiologically-based pharmacokinetic (PB-PK) model for methylene chloride: Implications for risk assessment
    • Reitz, R. H., Mendrala, A. L., Park, C. N., Andersen, M. E., and Guengerich, F. P. (1988). Incorporation of in vitro enzyme data into the physiologically-based pharmacokinetic (PB-PK) model for methylene chloride: Implications for risk assessment. Toxicol. Lett. 43, 97-116.
    • (1988) Toxicol. Lett. , vol.43 , pp. 97-116
    • Reitz, R.H.1    Mendrala, A.L.2    Park, C.N.3    Andersen, M.E.4    Guengerich, F.P.5
  • 26
    • 0024515167 scopus 로고
    • In vitro metabolism of methylene chloride in human and animal tissues: Use in physiologically based pharmacokinetic models
    • Reitz, R. H., Mendrala, A. L., and Guengerich, F. P. (1989). In vitro metabolism of methylene chloride in human and animal tissues: Use in physiologically based pharmacokinetic models. Toxicol. Appl. Pharmacol. 97, 230-246.
    • (1989) Toxicol. Appl. Pharmacol. , vol.97 , pp. 230-246
    • Reitz, R.H.1    Mendrala, A.L.2    Guengerich, F.P.3
  • 27
    • 0018350651 scopus 로고
    • A vial-equilibration method to evaluate the drug-metabolizing enzyme activity for volatile hydrocarbons
    • Sato, A., and Nakajima, T. (1979a). A vial-equilibration method to evaluate the drug-metabolizing enzyme activity for volatile hydrocarbons. Toxicol. Appl. Pharmacol. 47, 41-46.
    • (1979) Toxicol. Appl. Pharmacol. , vol.47 , pp. 41-46
    • Sato, A.1    Nakajima, T.2
  • 28
    • 0018760585 scopus 로고
    • A structure-activity relationship of some chlorinated hydrocarbons
    • Sato, A., and Nakajima, T. (1979b). A structure-activity relationship of some chlorinated hydrocarbons. Arch. Environ. Health 34, 69-75.
    • (1979) Arch. Environ. Health , vol.34 , pp. 69-75
    • Sato, A.1    Nakajima, T.2
  • 29
    • 0018693845 scopus 로고
    • A structure-activity relationship of some chlorinated hydrocarbons
    • Sato, A., and Nakajima, T. (1979c). A structure-activity relationship of some chlorinated hydrocarbons. Brit. J. Ind. Med. 36, 231-234.
    • (1979) Brit. J. Ind. Med. , vol.36 , pp. 231-234
    • Sato, A.1    Nakajima, T.2
  • 30
    • 0015394053 scopus 로고
    • Diethylaminoethyl 2,2-diphenylvalerate HCl (SKF 525-A)-in vivo and in vitro effects of metabolism by rat liver microsomes - Formation of an oxygenated complex
    • Schenkman, J. B., Wilson, B. J., and Cinti, D. L. (1972). Diethylaminoethyl 2,2-diphenylvalerate HCl (SKF 525-A)-in vivo and in vitro effects of metabolism by rat liver microsomes - Formation of an oxygenated complex. Biochem. Pharmacol. 21, 2373-2383.
    • (1972) Biochem. Pharmacol. , vol.21 , pp. 2373-2383
    • Schenkman, J.B.1    Wilson, B.J.2    Cinti, D.L.3
  • 31
    • 0022340278 scopus 로고
    • Effect of phorone-induced glutathione depletion on the metabolism and hepatotoxicity of carbon tetrachloride and vinylidene chloride in rats
    • Siegers, C. P., Horn, W., and Younes, M. (1985). Effect of phorone-induced glutathione depletion on the metabolism and hepatotoxicity of carbon tetrachloride and vinylidene chloride in rats. J. Appl. Toxicol. 5, 352-356.
    • (1985) J. Appl. Toxicol. , vol.5 , pp. 352-356
    • Siegers, C.P.1    Horn, W.2    Younes, M.3
  • 34
    • 0018225140 scopus 로고
    • Synergistic effects of phorone on the hepatotoxicity of bromobenzene and paracetamol in mice
    • Van Doom, R., Leijdekkers, CH-. M., and Henderson, P. T. H. (1978). Synergistic effects of phorone on the hepatotoxicity of bromobenzene and paracetamol in mice. Toxicology 11, 225-233.
    • (1978) Toxicology , vol.11 , pp. 225-233
    • Van Doom, R.1    Leijdekkers, C.H.-M.2    Henderson, P.T.H.3
  • 35
    • 0025099248 scopus 로고
    • Oxidation of glycerol to formaldehyde by rat liver microsomes. Effects of cytochrome P-450 inducing agents
    • Winters, D. K., and Cederbaum, A. I. (1990). Oxidation of glycerol to formaldehyde by rat liver microsomes. Effects of cytochrome P-450 inducing agents. Biochem. Pharmacol. 39, 697-705.
    • (1990) Biochem. Pharmacol. , vol.39 , pp. 697-705
    • Winters, D.K.1    Cederbaum, A.I.2
  • 36
    • 0023263168 scopus 로고
    • Nature of N-nitrosodimethylamine demethylase and its inhibitors
    • Yoo, J.-S. H., Cheung, R. J., Pattern, C. J., Wade, D., and Yang, S. S. (1987). Nature of N-nitrosodimethylamine demethylase and its inhibitors. Cancer Res. 47, 3378-3383.
    • (1987) Cancer Res. , vol.47 , pp. 3378-3383
    • Yoo, J.-S.H.1    Cheung, R.J.2    Pattern, C.J.3    Wade, D.4    Yang, S.S.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.