Hybrid peptides having mixed substance P (NK1), neurokinin A (NK2) and bradykinin (BK2) antagonist properties

Immunopharmacology

Volumn 33, Issue 1-3, 1996, Pages 194-197

  Srivastava, Ved P ^a   Goodfellow, Val S ^a   Zuzack, John S ^a   Jones, Steve ^a   Francis, Mary ^a   Beckey, Virginia E ^a   Whalley, Eric T ^a  

^a Departments of New Leads Chemistry and Pharmacology   (United States)

Author keywords

asthma; bradykinin antagonist; heterodimer; neurokinin A; substance P

Indexed keywords

BRADYKININ; BRADYKININ B2 RECEPTOR ANTAGONIST; HYBRID PROTEIN; NEUROKININ 1 RECEPTOR ANTAGONIST; NEUROKININ 2 RECEPTOR ANTAGONIST; NEUROKININ A; PEPTIDE DERIVATIVE; RADIOLIGAND; SUBSTANCE P;

ANIMAL TISSUE; CONFERENCE PAPER; CONTROLLED STUDY; DRUG SYNTHESIS; GUINEA PIG; HUMAN; ILEUM; MOLECULAR CLONING; NONHUMAN; PEPTIDE SYNTHESIS; PRIORITY JOURNAL; RECEPTOR BINDING; STRUCTURE ACTIVITY RELATION;

EID: 0030175551     PISSN: 01623109     EISSN: None     Source Type: Journal    
DOI: 10.1016/0162-3109(96)00038-0     Document Type: Conference Paper

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