(E)-1-(Heterocyclyl or cyclohexyl)-2-[1,3,7-trisubstituted (xanthin-8-yl)] ethenes as A2a adenosine receptor antagonists

European Journal of Medicinal Chemistry

Volumn 31, Issue 1, 1996, Pages 59-63

  Del Giudice, M R ^a   Borioni, A ^a   Mustazza, C ^a   Gatta, F ^a   Dionisotti, S ^b   Zocchi, C ^b   Ongini, E ^b  

^a ISTITUTO SUPERIORE DI SANITÀ   (Italy)

^b Schering Plough   (Italy)

Author keywords

8 styrylxanthine analogue; Adenosine A2a receptor antagonist

Indexed keywords

7 METHYL 1,3 DIPROPYL 8 [2 (3 THIENYL)VINYL]XANTHINE; ADENOSINE A1 RECEPTOR; ADENOSINE A2 RECEPTOR; ADENOSINE RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG; XANTHINE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; CONTROLLED STUDY; CORPUS STRIATUM; DRUG RECEPTOR BINDING; DRUG STABILITY; DRUG STRUCTURE; DRUG SYNTHESIS; LIGHT; MALE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; RAT; STEREOCHEMISTRY; STRUCTURE ACTIVITY RELATION;

EID: 0030069866     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0223-5234(96)80007-9     Document Type: Article

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