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Volumn 43, Issue 2, 1996, Pages 127-136

Comparison of binding mechanisms at cholinergic, serotonergic, glycinergic and GABAergic receptors

Author keywords

ACh; chloride ion channel; GABA; GABA receptor; glycine; glycine receptor; nicotinic ACh receptor; sodium potassium ion channel

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID RECEPTOR; ACETYLCHOLINE; CHOLINERGIC RECEPTOR; GLYCINE; GLYCINE RECEPTOR; NEUROTRANSMITTER; NICOTINIC RECEPTOR; SEROTONIN; SEROTONIN 3 RECEPTOR; SEROTONIN RECEPTOR; TUBOCURARINE CHLORIDE;

EID: 0030064633     PISSN: 03604012     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1097-4547(19960115)43:2<127::AID-JNR1>3.0.CO;2-I     Document Type: Review
Times cited : (24)

References (39)
  • 1
    • 0027787023 scopus 로고
    • A receptor needs two homologous domains of the β-subunit for activation by GABA but not by pentobarbital
    • A receptor needs two homologous domains of the β-subunit for activation by GABA but not by pentobarbital. Nature 366:565-569.
    • (1993) Nature , vol.366 , pp. 565-569
    • Amin, J.1    Weiss, D.S.2
  • 3
    • 0025991904 scopus 로고
    • Molecular modeling of the weak glycine antagonist iso-THAO
    • Aprison MH, Lipkowitz KB (1991): Molecular modeling of the weak glycine antagonist iso-THAO. J Neurosci Res 30:442-446.
    • (1991) J Neurosci Res , vol.30 , pp. 442-446
    • Aprison, M.H.1    Lipkowitz, K.B.2
  • 4
    • 0026601764 scopus 로고
    • Muscimol and N,N-dimethyl-muscimol: From a GABA agonist to a glycine antagonist
    • Aprison MH, Lipkowitz KB (1992): Muscimol and N,N-dimethyl-muscimol: From a GABA agonist to a glycine antagonist. J Neurosci Res 31:166-174.
    • (1992) J Neurosci Res , vol.31 , pp. 166-174
    • Aprison, M.H.1    Lipkowitz, K.B.2
  • 5
    • 0028834218 scopus 로고
    • Identification of a second glycine-like fragment on the strychnine molecule
    • Aprison MH, Galvez-Ruano E, Lipkowitz KB (1995a): Identification of a second glycine-like fragment on the strychnine molecule. J Neurosci Res 40:396-400.
    • (1995) J Neurosci Res , vol.40 , pp. 396-400
    • Aprison, M.H.1    Galvez-Ruano, E.2    Lipkowitz, K.B.3
  • 6
    • 0029007833 scopus 로고
    • On a molecular comparison of strong and weak antagonists at the glycinergic receptor
    • Aprison MH, Galvez-Ruano E, Lipkowitz KB (1995b): On a molecular comparison of strong and weak antagonists at the glycinergic receptor. J Neurosci Res 41:259-269.
    • (1995) J Neurosci Res , vol.41 , pp. 259-269
    • Aprison, M.H.1    Galvez-Ruano, E.2    Lipkowitz, K.B.3
  • 10
    • 0000942975 scopus 로고
    • The crystal and molecular structure of a potent neuromuscular blocking agent: D-Tubocurarine Dichloride Pentahydrate
    • Codding PW, James MNG (1973): The crystal and molecular structure of a potent neuromuscular blocking agent: d-Tubocurarine Dichloride Pentahydrate. Acta Crystallogr B 29:935-942.
    • (1973) Acta Crystallogr B , vol.29 , pp. 935-942
    • Codding, P.W.1    James, M.N.G.2
  • 11
    • 0026344986 scopus 로고
    • Structure of the agonist-binding site of the nicotinic acetylcholine receptor
    • Cohen JB, Sharp SD, Liu WS (1991): Structure of the agonist-binding site of the nicotinic acetylcholine receptor. J Biol Chem 266: 23354-23364.
    • (1991) J Biol Chem , vol.266 , pp. 23354-23364
    • Cohen, J.B.1    Sharp, S.D.2    Liu, W.S.3
  • 15
    • 0029129275 scopus 로고
    • On identifying a second molecular antagonistic mechanism operative at the glycine receptor
    • Galvez-Ruano E, Lipkowitz KB, Aprison MH (1995a): On identifying a second molecular antagonistic mechanism operative at the glycine receptor. J Neurosci Res 41:775-781.
    • (1995) J Neurosci Res , vol.41 , pp. 775-781
    • Galvez-Ruano, E.1    Lipkowitz, K.B.2    Aprison, M.H.3
  • 16
    • 0028886410 scopus 로고
    • Identifying agonistic and antagonistic mechanisms operative at the GABA receptor
    • Galvez-Ruano E, Aprison MH, Robertson DH, Lipkowitz KB (1995b): Identifying agonistic and antagonistic mechanisms operative at the GABA receptor. J Neurosci Res 42:666-673.
    • (1995) J Neurosci Res , vol.42 , pp. 666-673
    • Galvez-Ruano, E.1    Aprison, M.H.2    Robertson, D.H.3    Lipkowitz, K.B.4
  • 17
    • 0025346780 scopus 로고
    • Identification of a novel amino acid α-Tyrosine 93 within the cholmergic ligands-binding sites of the acetylcholine receptor by photoaffinity labeling
    • Galzi JL, Revah F, Black D, Goeldner M, Hirth C, Changeux JP (1990): Identification of a novel amino acid α-Tyrosine 93 within the cholmergic ligands-binding sites of the acetylcholine receptor by photoaffinity labeling. J Biol Chem 265:10430-10437.
    • (1990) J Biol Chem , vol.265 , pp. 10430-10437
    • Galzi, J.L.1    Revah, F.2    Black, D.3    Goeldner, M.4    Hirth, C.5    Changeux, J.P.6
  • 18
    • 0019918111 scopus 로고
    • - conductance in inhibitory synaptic channels
    • - conductance in inhibitory synaptic channels. Nature 299: 828-830.
    • (1982) Nature , vol.299 , pp. 828-830
    • Gold, M.R.1    Martin, A.R.2
  • 22
    • 0001022354 scopus 로고
    • Hydrogen-bond length in homomolecular organic crystals
    • Kuleshova LN, Zorkii PM (1980): Hydrogen-bond length in homomolecular organic crystals. Acta Crystallogr B 37:1363-1366.
    • (1980) Acta Crystallogr B , vol.37 , pp. 1363-1366
    • Kuleshova, L.N.1    Zorkii, P.M.2
  • 23
    • 0026011344 scopus 로고
    • Ion channel formation by synthetic transmembrane segments of the inhibitory glycine receptor - A model study
    • Langosch D, Hartung K, Grell E, Bamberg E, Betz H (1991): Ion channel formation by synthetic transmembrane segments of the inhibitory glycine receptor - a model study. Biochem Biophys Acta 1063.36-44.
    • (1991) Biochem Biophys Acta , vol.1063 , pp. 36-44
    • Langosch, D.1    Hartung, K.2    Grell, E.3    Bamberg, E.4    Betz, H.5
  • 24
    • 0027764470 scopus 로고
    • Importance of ARG-219 for correct biogenesis of αI homooligomeric glycine receptors
    • Langosch D, Herbold A, Schmieden V, Borman J, Kirsch J (1993): Importance of ARG-219 for correct biogenesis of αI homooligomeric glycine receptors. FEBS Lett 3:540-544.
    • (1993) FEBS Lett , vol.3 , pp. 540-544
    • Langosch, D.1    Herbold, A.2    Schmieden, V.3    Borman, J.4    Kirsch, J.5
  • 25
    • 0028016521 scopus 로고
    • Decreased agonist affinity and chloride conductance of mutant glycine receptors associated with human hereditary hyperkeplexia
    • Langosch D, Laube B, Rundström N, Schmieden V, Bormann J, Betz H (1994): Decreased agonist affinity and chloride conductance of mutant glycine receptors associated with human hereditary hyperkeplexia. EMBO J 13:4223-4228.
    • (1994) EMBO J , vol.13 , pp. 4223-4228
    • Langosch, D.1    Laube, B.2    Rundström, N.3    Schmieden, V.4    Bormann, J.5    Betz, H.6
  • 26
    • 0001972149 scopus 로고
    • Electronic and structural features of γ-aminobutyric acid (GABA) and four of its direct agonists
    • Lipkowitz KB, Gilardi RD, Aprison MH (1989): Electronic and structural features of γ-aminobutyric acid (GABA) and four of its direct agonists. J Mol Struct 195:65-77.
    • (1989) J Mol Struct , vol.195 , pp. 65-77
    • Lipkowitz, K.B.1    Gilardi, R.D.2    Aprison, M.H.3
  • 28
    • 85050517685 scopus 로고
    • Molecular surfaces
    • Lipkowitz K, Boyd D (eds): New York: VCH
    • Mezey PG (1990): Molecular surfaces. In Lipkowitz K, Boyd D (eds): "Reviews in Computational Chemistry." Vol. 1. New York: VCH, pp 265-294.
    • (1990) Reviews in Computational Chemistry , vol.1 , pp. 265-294
    • Mezey, P.G.1
  • 29
    • 0025819979 scopus 로고
    • 3H] nicotine as an agonist photoaffinity label
    • 3H] nicotine as an agonist photoaffinity label. Biochemistry 30:6987-6997.
    • (1991) Biochemistry , vol.30 , pp. 6987-6997
    • Middleton, R.E.1    Cohen, J.B.2
  • 30
    • 9044246221 scopus 로고
    • MSI, 16 New England Executive Park, Burlington, MA 01803-5297 (Telephone no. 800-756-4674)
    • Molecular Simulations Incorporated, Quanta/CHARMm, version 4.1, 1995, MSI, 16 New England Executive Park, Burlington, MA 01803-5297 (Telephone no. 800-756-4674).
    • (1995) Molecular Simulations Incorporated, Quanta/CHARMm, Version 4.1
  • 31
    • 0026758178 scopus 로고
    • Mutational analysis of ligand-induced actrvation of the torpedo acetylcholine receptor
    • O'Leary ME, White MM (1992): Mutational analysis of ligand-induced actrvation of the torpedo acetylcholine receptor. J Biol Chem 207:8360-8365.
    • (1992) J Biol Chem , vol.207 , pp. 8360-8365
    • O'Leary, M.E.1    White, M.M.2
  • 32
    • 0001198076 scopus 로고
    • Molecular electrostatic potentials and chemical reactivity
    • Lipkowitz K, Boyd D (eds): New York: VCH
    • Politzer P, Murray J (1991): Molecular electrostatic potentials and chemical reactivity. In Lipkowitz K, Boyd D (eds): "Reviews in Computational Chemistry." Vol. 2. New York: VCH.
    • (1991) Reviews in Computational Chemistry , vol.2
    • Politzer, P.1    Murray, J.2
  • 33
    • 0027424165 scopus 로고
    • Mutation of glycine receptor subunit creates β-alanine receptor responsive to GABA
    • Schmieden V, Kuhse J, Betz H (1993): Mutation of glycine receptor subunit creates β-alanine receptor responsive to GABA. Science 282:256-258.
    • (1993) Science , vol.282 , pp. 256-258
    • Schmieden, V.1    Kuhse, J.2    Betz, H.3
  • 35
    • 0039808378 scopus 로고
    • Quantun Chemistry Program Exchange
    • Stewart JJP (1993): MOPAC version 7, Quantun Chemistry Program Exchange 23:40-43.
    • (1993) MOPAC Version 7 , vol.23 , pp. 40-43
    • Stewart, J.J.P.1
  • 36
    • 0027506299 scopus 로고
    • Nicotinic acetylcholine receptor at 9Å resolution
    • Unwin N (1993). Nicotinic acetylcholine receptor at 9Å resolution. J Mol Biol 229:1101-1124.
    • (1993) J Mol Biol , vol.229 , pp. 1101-1124
    • Unwin, N.1
  • 37
    • 0028921479 scopus 로고
    • Acetylcholine receptor channel imaged in the open state
    • Unwin N (1995): Acetylcholine receptor channel imaged in the open state. Nature 373:37-43.
    • (1995) Nature , vol.373 , pp. 37-43
    • Unwin, N.1
  • 38
    • 0026787189 scopus 로고
    • Distinct agonist- and antagonist-binding sites on the glycine receptor
    • Vandenberg RJ, Handford CA, Schofield PR (1992): Distinct agonist- and antagonist-binding sites on the glycine receptor. Neuron 9:491-496.
    • (1992) Neuron , vol.9 , pp. 491-496
    • Vandenberg, R.J.1    Handford, C.A.2    Schofield, P.R.3
  • 39
    • 0024073762 scopus 로고
    • 3 receptors mediate rapid response in cultured hippocampus and a clonal cell line
    • 3 receptors mediate rapid response in cultured hippocampus and a clonal cell line. Neuron 1:615-621.
    • (1988) Neuron , vol.1 , pp. 615-621
    • Yakel, J.L.1    Jackson, M.B.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.