메뉴 건너뛰기




Volumn 40, Issue 2, 1996, Pages 473-476

Mode of action of GR122222X, a novel inhibitor of bacterial DNA gyrase

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINE TRIPHOSPHATASE; CIPROFLOXACIN; COUMARIN; GR 122222X; GYRASE INHIBITOR; NOVOBIOCIN; QUINOLINE DERIVED ANTIINFECTIVE AGENT; UNCLASSIFIED DRUG;

EID: 0030053504     PISSN: 00664804     EISSN: None     Source Type: Journal    
DOI: 10.1128/aac.40.2.473     Document Type: Article
Times cited : (21)

References (31)
  • 1
    • 0027419771 scopus 로고
    • The 43-kDa N-terminal fragment of the gyrase B protein hydrolyses ATP and binds coumarin drugs
    • Ali, J. A., A. P. Jackson, A. J. Howells, and A. Maxwell. 1993. The 43-kDa N-terminal fragment of the gyrase B protein hydrolyses ATP and binds coumarin drugs. Biochemistry 32:2717-2724.
    • (1993) Biochemistry , vol.32 , pp. 2717-2724
    • Ali, J.A.1    Jackson, A.P.2    Howells, A.J.3    Maxwell, A.4
  • 2
    • 0029166885 scopus 로고
    • Nucleotide binding to the 43-kilodalton N-terminal fragment of the DNA gyrase B protein
    • Ali, J. A., G. Orphanides, and A. Maxwell. 1995 Nucleotide binding to the 43-kilodalton N-terminal fragment of the DNA gyrase B protein Biochemistry. 34:9801-9808.
    • (1995) Biochemistry , vol.34 , pp. 9801-9808
    • Ali, J.A.1    Orphanides, G.2    Maxwell, A.3
  • 3
    • 0026648204 scopus 로고
    • gyrB mutations which confer coumarin resistance also affect DNA supercoiling and ATP hydrolysis by Escherichia coli DNA gyrase
    • Contreras, A., and A. Maxwell. 1992. gyrB mutations which confer coumarin resistance also affect DNA supercoiling and ATP hydrolysis by Escherichia coli DNA gyrase Mol. Microbiol. 6:1617-1624
    • (1992) Mol. Microbiol. , vol.6 , pp. 1617-1624
    • Contreras, A.1    Maxwell, A.2
  • 4
    • 0024383245 scopus 로고
    • Cloning and characterization of a DNA gyrase A gene from Escherichia coli that confers clinical resistance to 4-quinolones
    • Cullen, M. E., A. W. Wyke, R. Kuroda, and L. M. Fisher. 1989. Cloning and characterization of a DNA gyrase A gene from Escherichia coli that confers clinical resistance to 4-quinolones. Antimicrob. Agents Chemother. 33:886-894
    • (1989) Antimicrob. Agents Chemother. , vol.33 , pp. 886-894
    • Cullen, M.E.1    Wyke, A.W.2    Kuroda, R.3    Fisher, L.M.4
  • 6
    • 0024429631 scopus 로고
    • Inhibitors of DNA gyrase
    • Drlica, K., and S. Coughlin. 1989. Inhibitors of DNA gyrase. Pharmacol. Ther. 44:107-121.
    • (1989) Pharmacol. Ther. , vol.44 , pp. 107-121
    • Drlica, K.1    Coughlin, S.2
  • 8
    • 0001373485 scopus 로고
    • Nalidixic acid resistance: A second genetic character involved in DNA gyrase activity
    • Gellert, M., K. Mizuuchi, M. H. O'Dea, T. Itoh, and J. Tomizawa. 1977. Nalidixic acid resistance: a second genetic character involved in DNA gyrase activity. Proc. Natl. Acad. Sci. USA 74:4772-4776.
    • (1977) Proc. Natl. Acad. Sci. USA , vol.74 , pp. 4772-4776
    • Gellert, M.1    Mizuuchi, K.2    O'Dea, M.H.3    Itoh, T.4    Tomizawa, J.5
  • 9
    • 0028363364 scopus 로고
    • The 24 kDa N-terminal sub domain of the DNA gyrase B protein binds coumarin drugs
    • Gilbert, E. J., and A. Maxwell. 1994. The 24 kDa N-terminal sub domain of the DNA gyrase B protein binds coumarin drugs Mol Microbiol. 12:365-373.
    • (1994) Mol Microbiol. , vol.12 , pp. 365-373
    • Gilbert, E.J.1    Maxwell, A.2
  • 13
    • 0019812210 scopus 로고
    • Mechanism of action of cinodine, a glycocinnamoylspermidine antibiotic
    • Greenstein, M., J. L. Speth, and W. M. Maise. 1981. Mechanism of action of cinodine, a glycocinnamoylspermidine antibiotic. Antimicrob. Agents Chemother. 20:425-432.
    • (1981) Antimicrob. Agents Chemother. , vol.20 , pp. 425-432
    • Greenstein, M.1    Speth, J.L.2    Maise, W.M.3
  • 14
    • 0025155773 scopus 로고
    • Cloning of the DNA gyrase genes under tac promoter control overproduction of the gyrase A and B proteins
    • Hallett, P., A. J. Grimshaw, D. B. Wigley, and A. Maxwell. 1990. Cloning of the DNA gyrase genes under tac promoter control overproduction of the gyrase A and B proteins. Gene 93:139-142
    • (1990) Gene , vol.93 , pp. 139-142
    • Hallett, P.1    Grimshaw, A.J.2    Wigley, D.B.3    Maxwell, A.4
  • 15
    • 0028068693 scopus 로고
    • Crystallisation of inhibitor complexes of an N-terminal fragment of the DNA gyrase B protein
    • Lewis, R. J., O. M. P. Singh, C. V. Smith, A. Maxwell, A. J. Wonacott, and D. B. Wigley. 1994. Crystallisation of inhibitor complexes of an N-terminal fragment of the DNA gyrase B protein. J. Mol. Biol. 241:128-130.
    • (1994) J. Mol. Biol. , vol.241 , pp. 128-130
    • Lewis, R.J.1    Singh, O.M.P.2    Smith, C.V.3    Maxwell, A.4    Wonacott, A.J.5    Wigley, D.B.6
  • 16
    • 85088673636 scopus 로고    scopus 로고
    • The nature of inhibition of DNA gyrase by the coumarins and the cyclothialidines revealed by X-ray crystallography
    • in press
    • Lewis, R. J., O. M. P. Singh, C. V. Smith, T. Skarynski, A. Maxwell, A. J. Wonacott, and D. B. Wigley. The nature of inhibition of DNA gyrase by the coumarins and the cyclothialidines revealed by X-ray crystallography. EMBO J., in press.
    • EMBO J.
    • Lewis, R.J.1    Singh, O.M.P.2    Smith, C.V.3    Skarynski, T.4    Maxwell, A.5    Wonacott, A.J.6    Wigley, D.B.7
  • 17
    • 0026468457 scopus 로고
    • The molecular basis of quinolone action
    • Maxwell, A. 1992. The molecular basis of quinolone action. J. Antimicrob. Chemother. 30:409-416.
    • (1992) J. Antimicrob. Chemother. , vol.30 , pp. 409-416
    • Maxwell, A.1
  • 18
    • 0027200479 scopus 로고
    • The interaction between coumarin drugs and DNA gyrase
    • Maxwell, A. 1993. The interaction between coumarin drugs and DNA gyrase. Mol. Microbiol. 9:681-686.
    • (1993) Mol. Microbiol. , vol.9 , pp. 681-686
    • Maxwell, A.1
  • 20
    • 0021139129 scopus 로고
    • Cloning and simplified purification of Escherichia coli DNA gyrase A and B proteins
    • Mizuuchi, K., M. Mizuuchi, M. H. O'Dea, and M. Gellert. 1984. Cloning and simplified purification of Escherichia coli DNA gyrase A and B proteins. J Biol. Chem 259:9199-9201
    • (1984) J Biol. Chem , vol.259 , pp. 9199-9201
    • Mizuuchi, K.1    Mizuuchi, M.2    O'Dea, M.H.3    Gellert, M.4
  • 21
    • 13344265875 scopus 로고    scopus 로고
    • Unpublished observation
    • Moult, A. B., and K. Duncan. Unpublished observation
    • Moult, A.B.1    Duncan, K.2
  • 22
    • 0027933357 scopus 로고
    • Mechanism of inhibition of DNA gyrase by cyclothialidine, a novel DNA gyrase inhibitor
    • Nakada, N., H. Gmünder, T. Hirata, and M. Arisana. 1994. Mechanism of inhibition of DNA gyrase by cyclothialidine, a novel DNA gyrase inhibitor. Antimicrob. Agents Chemother 38:1966-1973.
    • (1994) Antimicrob. Agents Chemother , vol.38 , pp. 1966-1973
    • Nakada, N.1    Gmünder, H.2    Hirata, T.3    Arisana, M.4
  • 24
    • 0025348759 scopus 로고
    • In vitro inhibition of bacterial DNA gyrase by cinodine, a glycocinnamoylspermidine antibiotic
    • Osburne, M. S., W. M. Maiese, and M. Greenstein. 1990. In vitro inhibition of bacterial DNA gyrase by cinodine, a glycocinnamoylspermidine antibiotic. Antimicrob. Agents Chemother. 34:1450-1452.
    • (1990) Antimicrob. Agents Chemother. , vol.34 , pp. 1450-1452
    • Osburne, M.S.1    Maiese, W.M.2    Greenstein, M.3
  • 25
    • 0025091073 scopus 로고
    • Structure-activity relationships in DNA gyrase inhibitors
    • Rádl, S. 1990. Structure-activity relationships in DNA gyrase inhibitors. Pharmacol. Ther. 48:1-17.
    • (1990) Pharmacol. Ther. , vol.48 , pp. 1-17
    • Rádl, S.1
  • 26
    • 0024398661 scopus 로고
    • Tryptic fragments of the Escherichia coli DNA gyrase A protein
    • Reece, R. J., and A. Maxwell. 1989. Tryptic fragments of the Escherichia coli DNA gyrase A protein. J. Biol. Chem. 264:19648-19653.
    • (1989) J. Biol. Chem. , vol.264 , pp. 19648-19653
    • Reece, R.J.1    Maxwell, A.2
  • 27
    • 0026015132 scopus 로고
    • DNA gyrase: Structure and function Crit
    • Reece, R. J., and A. Maxwell. 1991. DNA gyrase: structure and function Crit. Rev Biochem Mol Biol. 26:335-375.
    • (1991) Rev Biochem Mol Biol. , vol.26 , pp. 335-375
    • Reece, R.J.1    Maxwell, A.2
  • 28
    • 0019878168 scopus 로고
    • DNA gyrase: Affinity Chromatography on novobiocin-Sepharose and catalytic properties
    • Staudenbauer, W. L., and E. Orr. 1981. DNA gyrase: affinity Chromatography on novobiocin-Sepharose and catalytic properties. Nucleic Acids Res 9:3589-3603.
    • (1981) Nucleic Acids Res , vol.9 , pp. 3589-3603
    • Staudenbauer, W.L.1    Orr, E.2
  • 29
    • 0025964113 scopus 로고
    • The peptide antibiotic microcin B17 induces double-strand cleavage of DNA mediated by E. coli DNA gyrase
    • Vizan, J., C. Hernandex-Chico, I. Castillo, and F. Moreno. 1991. The peptide antibiotic microcin B17 induces double-strand cleavage of DNA mediated by E. coli DNA gyrase. EMBO J. 10:467-476.
    • (1991) EMBO J. , vol.10 , pp. 467-476
    • Vizan, J.1    Hernandex-Chico, C.2    Castillo, I.3    Moreno, F.4
  • 30
    • 0026428621 scopus 로고
    • Crystal structure of an N-terminal fragment of the DNA gyrase B protein
    • Wigley, D. B., G. J. Davies, E. J. Dodson, A. Maxwell, and G. Dodson. 1991 Crystal structure of an N-terminal fragment of the DNA gyrase B protein. Nature (London) 351:624-629.
    • (1991) Nature (London) , vol.351 , pp. 624-629
    • Wigley, D.B.1    Davies, G.J.2    Dodson, E.J.3    Maxwell, A.4    Dodson, G.5
  • 31
    • 0023906965 scopus 로고
    • Quinolone-resistant mutations of the gyrA gene of Escherichia coli
    • Yoshida, H., T. Kojima, J. Yamagishi, and S. Nakamura. 1988. Quinolone-resistant mutations of the gyrA gene of Escherichia coli. Mol Gen. Genet. 211:1-7.
    • (1988) Mol Gen. Genet. , vol.211 , pp. 1-7
    • Yoshida, H.1    Kojima, T.2    Yamagishi, J.3    Nakamura, S.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.