메뉴 건너뛰기




Volumn 75, Issue 1, 1996, Pages 154-160

Inhibition by argatroban, a specific thrombin inhibitor, of platelet activation by fibrin clot-associated thrombin

Author keywords

[No Author keywords available]

Indexed keywords

ANTITHROMBIN III; ARGATROBAN; FIBRINOGEN; HEPARIN; LEPIRUDIN; THROMBIN; THROMBIN INHIBITOR; THROMBOXANE B2;

EID: 0030052674     PISSN: 03406245     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-0038-1650236     Document Type: Article
Times cited : (41)

References (44)
  • 2
    • 0021035369 scopus 로고
    • Studies on the mechanism of thrombin interaction with fibrin
    • Kaminski M, McDonagh J. Studies on the mechanism of thrombin interaction with fibrin. J Biol Chem 1983, 258: 7627-30.
    • (1983) J Biol Chem , vol.258 , pp. 7627-7630
    • Kaminski, M.1    McDonagh, J.2
  • 3
    • 9044224657 scopus 로고
    • Inhibited thrombins: Interactions with fibrinogen and fibrin
    • Kaminski M, McDonagh J Inhibited thrombins: Interactions with fibrinogen and fibrin. J Biol Chem 1987; 262: 881-7.
    • (1987) J Biol Chem , vol.262 , pp. 881-887
    • Kaminski, M.1    McDonagh, J.2
  • 4
    • 0022369895 scopus 로고
    • Human α-thrombin binding to fibrinsepharose: Evidence for an anionic binding site
    • Berliner LJ, Sugawara Y, Fenton JW II. Human α-thrombin binding to fibrinsepharose: Evidence for an anionic binding site. Biochemistry 1985; 24: 7005-9.
    • (1985) Biochemistry , vol.24 , pp. 7005-7009
    • Berliner, L.J.1    Sugawara, Y.2    Fenton II, J.W.3
  • 7
    • 0023918947 scopus 로고
    • The localization of the binding site on fibrin for the secondary binding site of thrombin
    • Vali Z, Scheraga H. The localization of the binding site on fibrin for the secondary binding site of thrombin. Biochemistry, 1988, 27: 1956-63.
    • (1988) Biochemistry , vol.27 , pp. 1956-1963
    • Vali, Z.1    Scheraga, H.2
  • 8
    • 0024345758 scopus 로고
    • Evaluation of the inhibition by heparin and hirudin of coagulation activation during r-t-PA-induced thrombolysis
    • Mirshahi M, Soria J, Soria C, Faivre R, Lu H, Courtney M, Roitsch C, Tripier D, Caen JP. Evaluation of the inhibition by heparin and hirudin of coagulation activation during r-t-PA-induced thrombolysis. Blood 1989; 74: 1025-30.
    • (1989) Blood , vol.74 , pp. 1025-1030
    • Mirshahi, M.1    Soria, J.2    Soria, C.3    Faivre, R.4    Lu, H.5    Courtney, M.6    Roitsch, C.7    Tripier, D.8    Caen, J.P.9
  • 9
    • 0027393953 scopus 로고
    • Inhibition of concomitant thrombin-mediated fibrin formation enhances clot lysis in whole blood
    • Haskel EJ, Eisenberg PR, Abendschein DR. Inhibition of concomitant thrombin-mediated fibrin formation enhances clot lysis in whole blood. Blood Coagulation Fibrinolysis 1993; 4: 7-13.
    • (1993) Blood Coagulation Fibrinolysis , vol.4 , pp. 7-13
    • Haskel, E.J.1    Eisenberg, P.R.2    Abendschein, D.R.3
  • 10
    • 0027538598 scopus 로고
    • α-Thrombin within fibrin clots: Inactivation of thrombin by antithrombin-III
    • Naski MC, Shafer JA. α-Thrombin within fibrin clots: Inactivation of thrombin by antithrombin-III. Thromb Res 1993; 69: 453-65.
    • (1993) Thromb Res , vol.69 , pp. 453-465
    • Naski, M.C.1    Shafer, J.A.2
  • 11
    • 0025146426 scopus 로고
    • Clot bound thrombin is protected from inhibition by heparin-antithrombin III but is susceptible to inactivation by antithrombin III independent inhibitors
    • Weitz JI, Hudoba M, Masel D, Maraganore J, Hirsh J. Clot bound thrombin is protected from inhibition by heparin-antithrombin III but is susceptible to inactivation by antithrombin III independent inhibitors. J Clin Invest 1990; 86: 385-91.
    • (1990) J Clin Invest , vol.86 , pp. 385-391
    • Weitz, J.I.1    Hudoba, M.2    Masel, D.3    Maraganore, J.4    Hirsh, J.5
  • 12
    • 0027959329 scopus 로고
    • Effects of the synthetic thrombin inhibitor argatroban on fibrin- or clot-incorporated thrombin: Comparison with heparin and recombinant hirudin
    • Berry CN, Girardot C, Lecoffre C, Lunven C. Effects of the synthetic thrombin inhibitor argatroban on fibrin- or clot-incorporated thrombin: comparison with heparin and recombinant hirudin. Thromb Haemost 1994; 72, 381-6.
    • (1994) Thromb Haemost , vol.72 , pp. 381-386
    • Berry, C.N.1    Girardot, C.2    Lecoffre, C.3    Lunven, C.4
  • 13
    • 0018750813 scopus 로고
    • D-Phe-Pro-Arg CH,Cl. A selective affinity label for thrombin
    • Kettner C, Shaw E. D-Phe-Pro-Arg CH,Cl. A selective affinity label for thrombin. Thromb Res 1979, 14: 969-73
    • (1979) Thromb Res , vol.14 , pp. 969-973
    • Kettner, C.1    Shaw, E.2
  • 15
    • 0019891328 scopus 로고
    • Potent inhibition of thrombin by the newly synthesized arginine derivative no. 805. The importance of stereo-structure of its hydrophobic carboxamide portion
    • Okamoto S, Hijikata A, Kikumoto R, Tonomara S, Hara H, Ninomiya K, Maruyama A, Sugano M, Tamao Y. Potent inhibition of thrombin by the newly synthesized arginine derivative no. 805. The importance of stereo-structure of its hydrophobic carboxamide portion. Biochem Biophys Res Commun 1981; 101: 440-6.
    • (1981) Biochem Biophys Res Commun , vol.101 , pp. 440-446
    • Okamoto, S.1    Hijikata, A.2    Kikumoto, R.3    Tonomara, S.4    Hara, H.5    Ninomiya, K.6    Maruyama, A.7    Sugano, M.8    Tamao, Y.9
  • 17
    • 0026692059 scopus 로고
    • Comparative antithrombotic effects of heparin, recombinant hirudin and argatroban in a hamster femoral vein platelet-rich mural thrombosis model
    • Imura Y, Stassen J-M, Collen D. Comparative antithrombotic effects of heparin, recombinant hirudin and argatroban in a hamster femoral vein platelet-rich mural thrombosis model. J Pharm Exp Ther 1992; 261: 895-8.
    • (1992) J Pharm Exp Ther , vol.261 , pp. 895-898
    • Imura, Y.1    Stassen, J.-M.2    Collen, D.3
  • 20
    • 0024411829 scopus 로고
    • Thrombin is an important mediator of platelet aggregation in stenosed canine coronary arteries with endothelial injury
    • Eidt JF, Allison P, Noble S, Ashton J, Golino P, Mcnatt J, Buja LM, Willerson JT. Thrombin is an important mediator of platelet aggregation in stenosed canine coronary arteries with endothelial injury. J Clin Invest 1989; 84: 18-27.
    • (1989) J Clin Invest , vol.84 , pp. 18-27
    • Eidt, J.F.1    Allison, P.2    Noble, S.3    Ashton, J.4    Golino, P.5    Mcnatt, J.6    Buja, L.M.7    Willerson, J.T.8
  • 21
    • 0028004409 scopus 로고
    • Antithrombotic actions of argatroban in rat models of venous, 'mixed' and arterial thrombosis, and its effects on the tail transection bleeding time
    • Berry CN, Girard D, Lochot S, Lecoffre C. Antithrombotic actions of argatroban in rat models of venous, 'mixed' and arterial thrombosis, and its effects on the tail transection bleeding time. Br J Pharmacol 1994; 113: 1209-14.
    • (1994) Br J Pharmacol , vol.113 , pp. 1209-1214
    • Berry, C.N.1    Girard, D.2    Lochot, S.3    Lecoffre, C.4
  • 23
    • 0025648376 scopus 로고
    • In vivo thrombin inhibition enhances and sustains arterial recanalisation with recombinant tissue-type plasminogen activator
    • Jang I-K, Gold HK, Leinbach RC, Fallon JT, Collen D. In vivo thrombin inhibition enhances and sustains arterial recanalisation with recombinant tissue-type plasminogen activator. Circulation Research 1990, 67: 1552-63.
    • (1990) Circulation Research , vol.67 , pp. 1552-1563
    • Jang, I.-K.1    Gold, H.K.2    Leinbach, R.C.3    Fallon, J.T.4    Collen, D.5
  • 24
    • 0026353329 scopus 로고
    • Heparin and the thrombin inhibitor argatroban enhance fibrinolysis by infused or bolus-injected saruplase (r-scu-PA) in rabbit femoral artery thrombosis
    • Schneider J. Heparin and the thrombin inhibitor argatroban enhance fibrinolysis by infused or bolus-injected saruplase (r-scu-PA) in rabbit femoral artery thrombosis. Thrombosis Res 1991; 64: 677-89.
    • (1991) Thrombosis Res , vol.64 , pp. 677-689
    • Schneider, J.1
  • 25
    • 0025143892 scopus 로고
    • Comparative effects of aspirin, a synthetic thrombin inhibitor and a monoclonal antiplatelet glycoprotein IIb/IIIa antibody on coronary artery reperfusion, reocclusion and bleeding with recombinant tissue-type plasminogen activator in a canine preparation
    • Yasuda T, Gold HK, Yaoita H, Leinbach RC, Guerrero JL, Jang IK, Holt R, Fallon JT, Collen D Comparative effects of aspirin, a synthetic thrombin inhibitor and a monoclonal antiplatelet glycoprotein IIb/IIIa antibody on coronary artery reperfusion, reocclusion and bleeding with recombinant tissue-type plasminogen activator in a canine preparation. J Am Coll Cardiol 1990; 16: 714-22.
    • (1990) J Am Coll Cardiol , vol.16 , pp. 714-722
    • Yasuda, T.1    Gold, H.K.2    Yaoita, H.3    Leinbach, R.C.4    Guerrero, J.L.5    Jang, I.K.6    Holt, R.7    Fallon, J.T.8    Collen, D.9
  • 26
    • 0024393955 scopus 로고
    • 2 in reocclusion following coronary thrombolysis with tissue-type plasminogen activator
    • 2 in reocclusion following coronary thrombolysis with tissue-type plasminogen activator. Proc Natl Acad Sci 1989; 86: 7585-9.
    • (1989) Proc Natl Acad Sci , vol.86 , pp. 7585-7589
    • Fitzgerald, D.J.1    Fitzgerald, G.A.2
  • 27
    • 0025676311 scopus 로고
    • Prevention of reocclusion by MCI-9038, a thrombin inhibitor, following t-PA-induced thrombolysis in a canine model of femoral arterial thrombosis
    • Mellot MJ, Connolly TM, York SJ, Bush LR. Prevention of reocclusion by MCI-9038, a thrombin inhibitor, following t-PA-induced thrombolysis in a canine model of femoral arterial thrombosis. Thromb Haemost 1990; 64: 526-34.
    • (1990) Thromb Haemost , vol.64 , pp. 526-534
    • Mellot, M.J.1    Connolly, T.M.2    York, S.J.3    Bush, L.R.4
  • 28
    • 0026344225 scopus 로고
    • Direct observation of platelet adhesion to fibrinogen- and fibrin-coated surfaces
    • Jen CJ, Lin JS. Direct observation of platelet adhesion to fibrinogen- and fibrin-coated surfaces. Am J Physiol 1991; 261: H1457-63.
    • (1991) Am J Physiol , vol.261
    • Jen, C.J.1    Lin, J.S.2
  • 29
    • 0027215042 scopus 로고
    • Spreading of platelets on fibrin is mediated by the amino terminus of the β-chain including peptide β15-42
    • Hamaguchi M, Bunce LA, Sporn LA, Francis CW. Spreading of platelets on fibrin is mediated by the amino terminus of the β-chain including peptide β15-42. Blood 1993; 9: 2348-56.
    • (1993) Blood , vol.9 , pp. 2348-2356
    • Hamaguchi, M.1    Bunce, L.A.2    Sporn, L.A.3    Francis, C.W.4
  • 30
    • 0028007619 scopus 로고
    • The influence of fibrinogen and fibrin on thrombin generation - Evidence for feedback activation of the clotting system by clot-bound thrombin
    • Kumar R, Béguin S, Hemker HC. The influence of fibrinogen and fibrin on thrombin generation - evidence for feedback activation of the clotting system by clot-bound thrombin. Thromb Haemost 1994; 72: 713-21.
    • (1994) Thromb Haemost , vol.72 , pp. 713-721
    • Kumar, R.1    Béguin, S.2    Hemker, H.C.3
  • 31
    • 9044249579 scopus 로고
    • Agonists and receptors: Thrombin
    • Holmsen H, ed. CRC Press, Boca Raton, Florida
    • White GC, Lapetina EG. Agonists and receptors: thrombin. In: Platelet Responses and Metabolism Vol. II. Holmsen H, ed. CRC Press, Boca Raton, Florida, 1987; pp 3-18.
    • (1987) Platelet Responses and Metabolism Vol. II , vol.2 , pp. 3-18
    • White, G.C.1    Lapetina, E.G.2
  • 32
    • 8944254783 scopus 로고
    • Platelet activation by clot-associated thrombin: Inhibition by argatroban, a specific thrombin inhibitor
    • Berry CN, Lunven C, Lecoffre C, O'Brien D, Gauffeny C, Roome NO. Platelet activation by clot-associated thrombin: inhibition by argatroban, a specific thrombin inhibitor Br J Pharmacol 1995; 114 (Procs. Suppl.): 122P.
    • (1995) Br J Pharmacol , vol.114 , Issue.PROCS. SUPPL.
    • Berry, C.N.1    Lunven, C.2    Lecoffre, C.3    O'Brien, D.4    Gauffeny, C.5    Roome, N.O.6
  • 33
    • 0020459977 scopus 로고
    • The use of prostacyclin in the separation from plasma and washing of human platelets
    • Vargas JR., Radomski M, Moncada S. The use of prostacyclin in the separation from plasma and washing of human platelets. Prostaglandins 1982; 23: 929-45.
    • (1982) Prostaglandins , vol.23 , pp. 929-945
    • Vargas, J.R.1    Radomski, M.2    Moncada, S.3
  • 34
    • 3643086579 scopus 로고
    • In vitro platelet responses: Aggregation
    • Holmsen H, ed. CRC Press, Boca Raton, Florida
    • Gear ARL. In vitro platelet responses: aggregation. In: Platelet Responses and Metabolism Vol. I. Holmsen H, ed. CRC Press, Boca Raton, Florida, 1987; pp 97-114.
    • (1987) Platelet Responses and Metabolism Vol. I , vol.1 , pp. 97-114
    • Gear, A.R.L.1
  • 36
    • 0022981986 scopus 로고
    • Effect of argatroban (MD-805) on platelet function
    • Hara H, Tamao Y, Kikumoto R. Effect of argatroban (MD-805) on platelet function. Jap Pharmacol Ther 1986; 14, (Suppl 5): 13-9.
    • (1986) Jap Pharmacol Ther , vol.14 , Issue.5 SUPPL. , pp. 13-19
    • Hara, H.1    Tamao, Y.2    Kikumoto, R.3
  • 37
    • 0026472751 scopus 로고
    • Inhibition of platelet adhesion to fibrin(ogen) in flowing whole blood by Arg-Gly-Asp and fibrinogen γ-chain carboxy terminal peptides
    • Hantgan RR, Endenberg SC, Cavero I, Marguerie G, Uzan A, Sixma JJ, de Groot PG Inhibition of platelet adhesion to fibrin(ogen) in flowing whole blood by Arg-Gly-Asp and fibrinogen γ-chain carboxy terminal peptides. Thromb Haemost 1992; 68: 694-700.
    • (1992) Thromb Haemost , vol.68 , pp. 694-700
    • Hantgan, R.R.1    Endenberg, S.C.2    Cavero, I.3    Marguerie, G.4    Uzan, A.5    Sixma, J.J.6    De Groot, P.G.7
  • 39
    • 0024566520 scopus 로고
    • The effect of trace amounts of tissue factor on thrombin generation in platelet rich plasma, its inhibition by heparin
    • Béguin S, Lindhout T, Hemker HC. The effect of trace amounts of tissue factor on thrombin generation in platelet rich plasma, its inhibition by heparin. Thromb Haemost 1989; 61: 25-9.
    • (1989) Thromb Haemost , vol.61 , pp. 25-29
    • Béguin, S.1    Lindhout, T.2    Hemker, H.C.3
  • 40
    • 0020052831 scopus 로고
    • Generation of prothrombin converting activity and the exposure of phophatidyl-serine at the outer surface of platelets
    • Bevers EM, Comfurius P, Van Rijn JLML. Hemker HC, Zwaal RFA. Generation of prothrombin converting activity and the exposure of phophatidyl-serine at the outer surface of platelets. Eur J Biochem 1982; 122: 429-36.
    • (1982) Eur J Biochem , vol.122 , pp. 429-436
    • Bevers, E.M.1    Comfurius, P.2    Van Rijn, J.3    Hemker, H.C.4    Zwaal, R.F.A.5
  • 42
    • 0025138566 scopus 로고
    • Antithrombotic effects of recombinant hirudin in experimental angioplasty and intravascular thrombolysis
    • Kaiser B, Simon A, Markwardt F. Antithrombotic effects of recombinant hirudin in experimental angioplasty and intravascular thrombolysis. Thromb Haemost 1990; 63: 44-7.
    • (1990) Thromb Haemost , vol.63 , pp. 44-47
    • Kaiser, B.1    Simon, A.2    Markwardt, F.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.