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Volumn 7, Issue 1, 1996, Pages 72-77

Discriminative stimulus effects of the benzodiazepine receptor partial agonist bretazenil in pigeons and in rats

Author keywords

Benzodiazepines; Bretazenil; Diazepam insensitive receptor subtype; Drug discrimination; GABA(A); Partial agonists; Pigeon; Rat

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; BENZODIAZEPINE RECEPTOR; BENZODIAZEPINE RECEPTOR STIMULATING AGENT; BRETAZENIL; FLUMAZENIL; MIDAZOLAM; PARTIAL AGONIST; RECEPTOR SUBTYPE;

EID: 0030033404     PISSN: 09558810     EISSN: None     Source Type: Journal    
DOI: 10.1097/00008877-199601000-00007     Document Type: Article
Times cited : (6)

References (39)
  • 2
    • 0000186261 scopus 로고
    • Discriminative stimulus properties of the benzodiazepine receptor partial agonist β-carbolines abecarnil and ZK 95962: A comparison with chlordiazepoxide
    • Andrews JS and Stephens DN (1991) Discriminative stimulus properties of the benzodiazepine receptor partial agonist β-carbolines abecarnil and ZK 95962: a comparison with chlordiazepoxide. Behavioural Pharmacology, 2, 171-185.
    • (1991) Behavioural Pharmacology , vol.2 , pp. 171-185
    • Andrews, J.S.1    Stephens, D.N.2
  • 3
    • 0011317064 scopus 로고
    • Discriminative stimulus effects of benzodiazepine-receptor partial/selective agonists
    • Ator NA and Griffiths RR (1992) Discriminative stimulus effects of benzodiazepine-receptor partial/selective agonists. Journal of Psychopharmacology, A34.
    • (1992) Journal of Psychopharmacology
    • Ator, N.A.1    Griffiths, R.R.2
  • 4
    • 0021961041 scopus 로고
    • The non-sedating anxiolytic CGS 9896 produces discriminative stimuli that may be related to an anxioselective effect
    • Bennett DA (1985) The non-sedating anxiolytic CGS 9896 produces discriminative stimuli that may be related to an anxioselective effect. Life Sciences, 37, 703-709.
    • (1985) Life Sciences , vol.37 , pp. 703-709
    • Bennett, D.A.1
  • 5
    • 0027241130 scopus 로고
    • Tolerance/cross-tolerance to the discriminative stimulus effects of chlordiazepoxide and bretazenil
    • Bronson ME (1993) Tolerance/cross-tolerance to the discriminative stimulus effects of chlordiazepoxide and bretazenil. Molecular and Chemical Neuropathology, 18, 85-98.
    • (1993) Molecular and Chemical Neuropathology , vol.18 , pp. 85-98
    • Bronson, M.E.1
  • 6
    • 0023709743 scopus 로고
    • Intrinsic activity and discriminative stimu-lus effects of drags
    • Eds FC Colpaert and RL Balster, Springer-Verlag, Berlin
    • Colpaert FC (1988) Intrinsic activity and discriminative stimu-lus effects of drags. In: Transduction Mechanisms of Drug Stimuli (Eds FC Colpaert and RL Balster), pp. 154-160. Springer-Verlag, Berlin.
    • (1988) Transduction Mechanisms of Drug Stimuli , pp. 154-160
    • Colpaert, F.C.1
  • 7
    • 0022361117 scopus 로고
    • The Ro 15-1788 cue: Evidence for benzodiazepine agonist and inverse agonist properties
    • De Vry J and Slangen JL (1985a) The Ro 15-1788 cue: evidence for benzodiazepine agonist and inverse agonist properties. European Journal of Pharmacology, 119, 193-197.
    • (1985) European Journal of Pharmacology , vol.119 , pp. 193-197
    • De Vry, J.1    Slangen, J.L.2
  • 8
    • 0021881057 scopus 로고
    • Stimulus control induced by benzodiazepine antagonist Ro 15-1788 in the rat
    • De Vry J and Slangen JL (1985b) Stimulus control induced by benzodiazepine antagonist Ro 15-1788 in the rat. Psychopharmacology, 85, 483-485.
    • (1985) Psychopharmacology , vol.85 , pp. 483-485
    • De Vry, J.1    Slangen, J.L.2
  • 9
    • 0022638588 scopus 로고
    • Effects of chlordiazepoxide training dose on the mixed agonist-antagonist properties of benzodiazepine receptor antagonist Ro 15-1788, in a drug discrimination procedure
    • De Vry J and Slangen JL (1986) Effects of chlordiazepoxide training dose on the mixed agonist-antagonist properties of benzodiazepine receptor antagonist Ro 15-1788, in a drug discrimination procedure. Psychopharmacology, 88, 177-183.
    • (1986) Psychopharmacology , vol.88 , pp. 177-183
    • De Vry, J.1    Slangen, J.L.2
  • 11
    • 0022656375 scopus 로고
    • Intrinsic actions of the benzodiazepine receptor antagonist Ro 15-1788
    • File SE and Pellow S (1986) Intrinsic actions of the benzodiazepine receptor antagonist Ro 15-1788. Psychopharmacology, 88, 1-11.
    • (1986) Psychopharmacology , vol.88 , pp. 1-11
    • File, S.E.1    Pellow, S.2
  • 12
    • 0022233984 scopus 로고
    • Midazolam cue in rats: Generalization tests with anxiolytics and other drugs
    • Garcha HS, Rose IC and Stolerman IP (1985) Midazolam cue in rats: generalization tests with anxiolytics and other drugs. Psychopharmacology, 87, 233-237.
    • (1985) Psychopharmacology , vol.87 , pp. 233-237
    • Garcha, H.S.1    Rose, I.C.2    Stolerman, I.P.3
  • 13
  • 14
    • 0000107846 scopus 로고
    • a-benzodiazepine receptor: Biology and pharmacology
    • Eds GD Burrows, M Roth and R Noves Jr, Elsevier Science Publishers, Amsterdam
    • A-benzodiazepine receptor: biology and pharmacology. In: Handbook of Anxiety Vol 3: The Neurobiology of Anxiety (Eds GD Burrows, M Roth and R Noves Jr), pp. 165-188. Elsevier Science Publishers, Amsterdam.
    • (1990) Handbook of Anxiety Vol 3: The Neurobiology of Anxiety , pp. 165-188
    • Haefely, W.E.1
  • 15
    • 0002974334 scopus 로고
    • Comparative pharmacology of benzodiazepine receptor ligands with differing intrinsic efficacy
    • Eds EA Barnard and E Costa, Raven Press, New York
    • Haefely WE (1991) Comparative pharmacology of benzodiazepine receptor ligands with differing intrinsic efficacy. In: Transmitter Amino Acids and Receptors: Structures, Transduction and Models for Drug Development (Eds EA Barnard and E Costa), pp. 91-111. Raven Press, New York.
    • (1991) Transmitter Amino Acids and Receptors: Structures, Transduction and Models for Drug Development , pp. 91-111
    • Haefely, W.E.1
  • 16
    • 0025043989 scopus 로고
    • Novel anxiolytics that act as partial agonists at benzodiazepine receptors
    • Haefely WE, Martin JR and Schoch P (1990) Novel anxiolytics that act as partial agonists at benzodiazepine receptors. Trends in Pharmacological Science, 11, 452-456.
    • (1990) Trends in Pharmacological Science , vol.11 , pp. 452-456
    • Haefely, W.E.1    Martin, J.R.2    Schoch, P.3
  • 17
    • 0023856237 scopus 로고
    • Ro 16-6028, a benzodiazepine receptor partial agonist, does not exhibit anticonvulsant tolerance in mice
    • Haigh JRM and Feely M (1988) Ro 16-6028, a benzodiazepine receptor partial agonist, does not exhibit anticonvulsant tolerance in mice. European Journal of Pharmacology, 147, 283-285.
    • (1988) European Journal of Pharmacology , vol.147 , pp. 283-285
    • Haigh, J.R.M.1    Feely, M.2
  • 18
    • 0027283546 scopus 로고
    • Partial agonists, full agonists, antagonists: Dilemmas of definition
    • Hoyer D and Boddeke HWGM (1993) Partial agonists, full agonists, antagonists: dilemmas of definition. Trends in Pharmacological Science, 14, 270-275.
    • (1993) Trends in Pharmacological Science , vol.14 , pp. 270-275
    • Hoyer, D.1    Boddeke, H.W.G.M.2
  • 19
    • 0028217950 scopus 로고
    • Comparison of several benzodiazepine receptor ligands on two models of anxiolytic activity in the mouse: An analysis based on fractional receptor occupancies
    • Jones GH, Schneider C, Schneider HH, Seidler J. Cole BJ and Stephens DN (1994) Comparison of several benzodiazepine receptor ligands on two models of anxiolytic activity in the mouse: an analysis based on fractional receptor occupancies. Psychopharmacology, 114, 191-199.
    • (1994) Psychopharmacology , vol.114 , pp. 191-199
    • Jones, G.H.1    Schneider, C.2    Schneider, H.H.3    Seidler, J.4    Cole, B.J.5    Stephens, D.N.6
  • 21
    • 0027293426 scopus 로고
    • Pharmacological characterization of benzodiazepine receptor ligands with intrinsic efficacies ranging from high to zero
    • Martin JR, Schoch P, Jenck F, Moreau J-L and Haefely WE (1993) Pharmacological characterization of benzodiazepine receptor ligands with intrinsic efficacies ranging from high to zero. Psychopharmacology, 111, 415-422.
    • (1993) Psychopharmacology , vol.111 , pp. 415-422
    • Martin, J.R.1    Schoch, P.2    Jenck, F.3    Moreau, J.-L.4    Haefely, W.E.5
  • 22
    • 0025059553 scopus 로고
    • Physical dependence induced in DBA/2J mice by benzodiazepine receptor full agonists, but not by the partial agonist Ro 16-6028
    • Moreau J-L, Jenck F, Pieri L, Schoch P, Martin JR and Haefely WE (1990) Physical dependence induced in DBA/2J mice by benzodiazepine receptor full agonists, but not by the partial agonist Ro 16-6028. European Journal of Pharmacology, 190, 269-273.
    • (1990) European Journal of Pharmacology , vol.190 , pp. 269-273
    • Moreau, J.-L.1    Jenck, F.2    Pieri, L.3    Schoch, P.4    Martin, J.R.5    Haefely, W.E.6
  • 23
    • 0019983742 scopus 로고
    • Comparison of the degree of discriminability of various drugs using the t-maze drag discrimination paradigm
    • Overton DA (1982) Comparison of the degree of discriminability of various drugs using the t-maze drag discrimination paradigm. Psychopharmacology, 76, 385-395.
    • (1982) Psychopharmacology , vol.76 , pp. 385-395
    • Overton, D.A.1
  • 25
    • 0025818321 scopus 로고
    • The pentylnetetrazole-cue antagonist actions of bretazenil (Ro 16-6028) as compared to midazolam
    • Rijnders HJ, Järbe TUC and Slangen JL (1991) The pentylnetetrazole-cue antagonist actions of bretazenil (Ro 16-6028) as compared to midazolam. Pharmacology Biochemistry and Behavior, 39, 129-132.
    • (1991) Pharmacology Biochemistry and Behavior , vol.39 , pp. 129-132
    • Rijnders, H.J.1    Järbe, T.U.C.2    Slangen, J.L.3
  • 26
    • 0026573402 scopus 로고
    • Discriminative stimulus properties of the benzodiazepine receptor antagonist flumazenil
    • Rowan GA and Lucki I (1992) Discriminative stimulus properties of the benzodiazepine receptor antagonist flumazenil. Psychopharmacology, 107, 103-112.
    • (1992) Psychopharmacology , vol.107 , pp. 103-112
    • Rowan, G.A.1    Lucki, I.2
  • 27
    • 0023200043 scopus 로고
    • Further investigations of the stimulus properties of chlordiazepoxide and zolpidem. Agonism and antagonism by two novel benzodiazepines
    • Sanger DJ (1987) Further investigations of the stimulus properties of chlordiazepoxide and zolpidem. Agonism and antagonism by two novel benzodiazepines. Psychopharmacology, 93, 365-368.
    • (1987) Psychopharmacology , vol.93 , pp. 365-368
    • Sanger, D.J.1
  • 28
    • 0028893945 scopus 로고
    • Drug discrimination analysis of midazolam under a three-lever procedure: 1. Dose-dependent differences in generalization and antagonism
    • Sannerud CA and Ator NA (1995a) Drug discrimination analysis of midazolam under a three-lever procedure: 1. Dose-dependent differences in generalization and antagonism. Journal of Pharmacology and Experimental Therapeutics, 272, 100-111.
    • (1995) Journal of Pharmacology and Experimental Therapeutics , vol.272 , pp. 100-111
    • Sannerud, C.A.1    Ator, N.A.2
  • 29
    • 0028784279 scopus 로고
    • Drug discrimination analysis of midazolam under a three-lever procedure: II. Differential effects of benzodiazepine receptor agonists
    • in press
    • Sannerud CA and Ator NA (1995b) Drug discrimination analysis of midazolam under a three-lever procedure: II. Differential effects of benzodiazepine receptor agonists. Journal of Pharmacology and Experimental Therapeutics (in press).
    • (1995) Journal of Pharmacology and Experimental Therapeutics
    • Sannerud, C.A.1    Ator, N.A.2
  • 32
  • 34
    • 0023766147 scopus 로고
    • Anxiolytic properties of amygdaloid kindling unrelated to benzodiazepine receptors
    • Witkin JM, Lee MA and Walczak DD (1988) Anxiolytic properties of amygdaloid kindling unrelated to benzodiazepine receptors. Psychopharmacology, 96, 296-301.
    • (1988) Psychopharmacology , vol.96 , pp. 296-301
    • Witkin, J.M.1    Lee, M.A.2    Walczak, D.D.3
  • 35
    • 0026585373 scopus 로고
    • High affinity ligands for 'diazepam-insensitive' benzodiazepine receptors
    • Wong G and Skolnick P (1992) High affinity ligands for 'diazepam-insensitive' benzodiazepine receptors. European Journal of Pharmacology, 225, 63-68.
    • (1992) European Journal of Pharmacology , vol.225 , pp. 63-68
    • Wong, G.1    Skolnick, P.2
  • 36
  • 37
    • 0024524925 scopus 로고
    • Discriminative stimulus properties of midazolam: Comparison with other benzodiazepines
    • Woudenberg F and Slangen JL (1989) Discriminative stimulus properties of midazolam: comparison with other benzodiazepines. Psychopharmacology, 97, 466-470.
    • (1989) Psychopharmacology , vol.97 , pp. 466-470
    • Woudenberg, F.1    Slangen, J.L.2
  • 38
    • 0025215169 scopus 로고
    • Characterisation of the discriminative stimulus properties of flumazenil
    • Woudenberg F and Slangen JL (1990) Characterisation of the discriminative stimulus properties of flumazenil. European Journal of Pharmacology, 178, 29-36.
    • (1990) European Journal of Pharmacology , vol.178 , pp. 29-36
    • Woudenberg, F.1    Slangen, J.L.2
  • 39
    • 0026769789 scopus 로고
    • Discriminative stimulus effects of morphine: Effects of training dose on agonist and antagonist effects of mu opioids
    • Young AM, Masaki MA and Geula C (1992) Discriminative stimulus effects of morphine: effects of training dose on agonist and antagonist effects of mu opioids. Journal of Pharmacology and Experimental Therapeutics, 261, 246-257.
    • (1992) Journal of Pharmacology and Experimental Therapeutics , vol.261 , pp. 246-257
    • Young, A.M.1    Masaki, M.A.2    Geula, C.3


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