Kinetic properties of fluorinated substrate analogues on 5′-methylthioadenosine nucleosidase from Escherichia coli

European Journal of Medicinal Chemistry

Volumn 31, Issue 1, 1996, Pages 37-41

  Gatel, M ^a   Muzard, M ^a   Guillerm, D ^a   Guillerm, G ^a  

^a UNIVERSITÉ DE REIMS CHAMPAGNE ARDENNE   (France)

Author keywords

Fluorinated substrate analogue; MTA nucleosidase

Indexed keywords

5' DEOXY 5' (FLUOROMETHYLTHIO)ADENOSINE; 5' DEOXY 5' [(DIFLUOROMETHYL)THIO]ADENOSINE; 5' DEOXY 5' [(TRIFLUOROMETHYL)THIO]ADENOSINE; ADENOSINE DERIVATIVE; NUCLEOSIDASE; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; ENZYME ACTIVITY; ENZYME BINDING; ENZYME KINETICS; ESCHERICHIA COLI; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; NONHUMAN;

EID: 0030032316     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0223-5234(96)80004-3     Document Type: Article

References (24)

1. Ferro AJ (1979) Transmethylation (Usdin E, Borchart RT, Creveling CR, eds) Elsevier/North-Holland, New York, 117-126
2. Zappia V, Pegg AE (1988) Advances in Experimental Medicine and Biology (Zappia V, Peeg AE, eds) Plenum Press, New York, Vol 250
3. Williams-Ashman HG, Seidenfeld J, Galletti P (1982) Biochem Pharmacol 31, 277-288
4. Peeg AE, Williams-Ashman HG (1969) Biochem J 115, 241-247
5. Duerre JA (1962) J Biol Chem 237, 3737-3741
6. Ferro AJ, Barrett A, Shapiro SK (1976) Biochim Biophys Acta 438, 487-494
7. Della Ragione F, Porcelli M, Carteni-Farina M, Zappia V, Pegg AE (1985) Biochem J 232, 335-341
8. Ferro AJ, Barrett A, Shapiro SK (1978) J Biol Chem 253, 6021-6025
9. Backlund PS, Smith RA (1981) J Biol Chem 256, 1533-1535
10. Shapiro SK, Barrett A (1981) Biochem Biophy Res Commun 102, 302-307
11. Myer RW, Abeles RH (1990) J Biol Chem 265, 16913-16921
12. Savarese TM, Ghoda LY, Parks RE Jr (1983) Development of Target-Oriented Anticancer Drugs (Cheng YC, Goz B, Minkoff M, eds) Raven Press, NY, 129-142
13. Riscoe MK, Ferro AJ, Fitchen JH (1988) Antimicrob Agents Chemother 32, 1904-1906
14. Riscoe MK, Ferro AJ, Fitchen JH (1989) Parasitol Today 5, 330-333
15. Gianotti AJ, Tower PA, Sheley JH et al (1990) J Biol Chem 265, 831-837
16. Winter RW, Cornell KA, Johnson LL, Riscoe MK (1993) Bioorg Med Chem Lett 3, 2079-2082
17. Robins MJ, Wnuk SF (1988) Tetrahedron Lett 29, 5729-5732
18. Guillerm G, Gatel M (1994) J Chem Soc Perkin Trans 12, 153-154
19. Sufrin JR, Spiess AJ, Kramer DL, Libby PR, Porter CW (1989) J Med Chem 32, 997-1001
20. Houston ME, Vander Jagt DL, Honek JF (1991) Bioorg Med Chem Lett 11, 623-628
21. Ramachandran PV, Teodrorovic AV, Brown HC (1993) Tetrahedron 49, 1725-1738
22. York JL (1981) J Org Chem 46, 2171-2173
23. Nishikawa S, Ueno A, Inoue H, Takeda Y (1987) J Cell Physiol 133, 372-376
24. Guillerm G, Galas MC, Le Goffic F (1986) J Labelled Compds Radiopharm 23, 845-851