Derivatives of kynurenine as inhibitors of rat brain kynurenine aminotransferase

European Journal of Medicinal Chemistry

Volumn 31, Issue 1, 1996, Pages 11-21

  Varasi, M ^a   Della Torre, A ^a   Heidempergher, F ^a   Pevarello, P ^a   Speciale, C ^a   Guidetti, P ^b   Wells, D R ^b   Schwarcz, R ^b  

^a PFIZER INC   (United States)

^b UNIVERSITY OF MARYLAND SCHOOL OF MEDICINE   (United States)

Author keywords

Enzyme inhibition; Kynurenic acid; Kynurenine; Kynurenine aminotransferase; Neuroprotection

Indexed keywords

5 CHLOROKYNURENINE; KYNURENIC ACID DERIVATIVE; KYNURENINE AMINOTRANSFERASE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BRAIN; BRAIN HOMOGENATE; BRAIN TISSUE; CONTROLLED STUDY; DRUG SYNTHESIS; ENZYME ACTIVE SITE; ENZYME INHIBITION; MALE; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION;

EID: 0030030058     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0223-5234(96)80002-X     Document Type: Article

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