Quinoline-substituted dihydroindoles as cysLT1 (LTD4 receptor) antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 3, 1996, Pages 249-252

  Sawyer, J Scott ^a   Thrasher, K Jeff ^a   Bach, Nicholas J ^a   Stengel, Peter W ^a   Cockerham, Sandra L ^a   Silbaugh, Steven A ^a   Roman, Carlos R ^a   Froelich, Larry L ^a   Fleisch, Jerome H ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1 [3 [2,3 DIHYDRO 7 (5 TETRAZOLYLMETHYL)INDOL 1 YL]PHENYL] 2 (7 CHLOROQUINOLIN 2 YL) ETHENE; INDOLE DERIVATIVE; LEUKOTRIENE D4; LEUKOTRIENE D4 RECEPTOR; LEUKOTRIENE RECEPTOR BLOCKING AGENT; LY 290324; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BRONCHOSPASM; CONTROLLED STUDY; DOSE RESPONSE; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; GUINEA PIG; ILEUM; LUNG; NONHUMAN; ORAL DRUG ADMINISTRATION; QUANTITATIVE STRUCTURE ACTIVITY RELATION; TRACHEA;

EID: 0030022067     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0960-894x(96)00013-3     Document Type: Article

References (10)

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