Potent α-ketocarbonyl and boronic ester derived inhibitors of proteasome

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 3, 1996, Pages 287-290

  Iqbal, Mohamed ^a   Chatterjee, Sankar ^a   Kauer, James C ^a   Mallamo, John P ^a   Messina, Patricia A ^a   Reiboldt, Alyssa ^a   Siman, Robert ^a  

^a CEPHALON INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ENZYME INHIBITOR; OLIGOPEPTIDE; PROTEASOME; PROTEINASE INHIBITOR;

ARTICLE; AUTOPSY; BRAIN; CONTROLLED STUDY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; HUMAN TISSUE; LIVER;

EID: 0030020338     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0960-894X(96)00014-5     Document Type: Article

References (10)

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7. Shenvi, A. B.; US patent 4,537,773 (Aug. 27, 1985).
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10. Abbreviations used: BOP: benzotriazol-1-yloxy-tris(dimethylamino)phosphonium hexafluorophosphate HOBt: 1-hydroxybenzotriazole; NMM: N-methylmorpholine; DMF: N,N-dimethylformamide.