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Volumn 24, Issue 2, 1996, Pages 216-220

Local absorption kinetics into the portal system using the portal-venous concentration difference after an oral dose of diclofenac in the awakening rat: Accelerative effect of bile on intestinal absorption of diclofenac

Author keywords

[No Author keywords available]

Indexed keywords

DICLOFENAC; NONSTEROID ANTIINFLAMMATORY AGENT;

EID: 0030019765     PISSN: 00909556     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (19)

References (34)
  • 1
    • 0015264301 scopus 로고
    • Influence of route of administration on drug availability
    • M. Rowland: Influence of route of administration on drug availability. J. Pharm. Sci. 61, 70-74 (1972).
    • (1972) J. Pharm. Sci. , vol.61 , pp. 70-74
    • Rowland, M.1
  • 2
    • 0018101672 scopus 로고
    • Theoretical relationships between area under the curve and route of administration of drugs and their precursors for evaluating sites and pathways of metabolism
    • K. S. Pang and J. R. Gillette: Theoretical relationships between area under the curve and route of administration of drugs and their precursors for evaluating sites and pathways of metabolism. J. Pharm. Sci. 67, 703-704 (1978).
    • (1978) J. Pharm. Sci. , vol.67 , pp. 703-704
    • Pang, K.S.1    Gillette, J.R.2
  • 3
    • 0014439831 scopus 로고
    • Influence of the route of administration on the area under the plasma concentration-time curve
    • P. A. Harris and S. Riegelman: Influence of the route of administration on the area under the plasma concentration-time curve. J. Pharm. Sci. 58, 71-75 (1969).
    • (1969) J. Pharm. Sci. , vol.58 , pp. 71-75
    • Harris, P.A.1    Riegelman, S.2
  • 4
    • 0015128465 scopus 로고
    • Influence of first-pass effect on availability of drugs on oral administration
    • M. Gibaldi, R. N. Boyes, and S. Feldman: Influence of first-pass effect on availability of drugs on oral administration. J. Pharm. Sci. 60, 1338-1340 (1971).
    • (1971) J. Pharm. Sci. , vol.60 , pp. 1338-1340
    • Gibaldi, M.1    Boyes, R.N.2    Feldman, S.3
  • 5
    • 0024806363 scopus 로고
    • Oral idazoxan bioavailability in rat: Relevance of intestinal and hepatic first-pass effect
    • J. Valles, J. Prunonosa, A. Menargues, M. Nomen, and R. Obach: Oral idazoxan bioavailability in rat: relevance of intestinal and hepatic first-pass effect. Drug Metab. Dispos. 17, 673-676 (1994).
    • (1994) Drug Metab. Dispos. , vol.17 , pp. 673-676
    • Valles, J.1    Prunonosa, J.2    Menargues, A.3    Nomen, M.4    Obach, R.5
  • 6
    • 0028337470 scopus 로고
    • Determination of bioavailability and systemically available fractions of drugs undergoing reversible metabolism application to 4-amino-5-chloro-2-[2-(methylsulfinyl)ethoxy]-N-[2-(diethylamino)ethyl]benzamide and its sulfide and sulfone metabolites in rats
    • B. Kuo, J. C. Poole, K. Hwang, and H. Cheng: Determination of bioavailability and systemically available fractions of drugs undergoing reversible metabolism application to 4-amino-5-chloro-2-[2-(methylsulfinyl)ethoxy]-N-[2-(diethylamino)ethyl]benzamide and its sulfide and sulfone metabolites in rats. J. Pharm. Sci. 83, 386-390 (1971).
    • (1971) J. Pharm. Sci. , vol.83 , pp. 386-390
    • Kuo, B.1    Poole, J.C.2    Hwang, K.3    Cheng, H.4
  • 7
    • 0027231109 scopus 로고
    • Influence of anesthetic regimens on intestinal absorption in rats
    • H. Yuasa, K. Matsuda, and J. Watanabe: Influence of anesthetic regimens on intestinal absorption in rats. Pharm. Res. 10, 884-888 (1993).
    • (1993) Pharm. Res. , vol.10 , pp. 884-888
    • Yuasa, H.1    Matsuda, K.2    Watanabe, J.3
  • 8
    • 0013883801 scopus 로고
    • Factors affecting the absorption of riboflavin in man
    • G. Levy and W. J. Jusco: Factors affecting the absorption of riboflavin in man. J. Pharm. Sci. 55, 285-289 (1966).
    • (1966) J. Pharm. Sci. , vol.55 , pp. 285-289
    • Levy, G.1    Jusco, W.J.2
  • 9
    • 0014817006 scopus 로고
    • The effects of particle size on the absorption of phenacetine in man et al
    • L. F. Prescott, R. F. Steel, and W. R. Ferrier: The effects of particle size on the absorption of phenacetine in man et al. Clin. Pharmacol. Ther. 11, 496-504 (1970).
    • (1970) Clin. Pharmacol. Ther. , vol.11 , pp. 496-504
    • Prescott, L.F.1    Steel, R.F.2    Ferrier, W.R.3
  • 10
    • 0015124660 scopus 로고
    • Absorption characteristics of solid dispersed and micronized griseofulvin in man
    • W. L. Chiou and S. Riegelman: Absorption characteristics of solid dispersed and micronized griseofulvin in man. J. Pharm. Sci. 60, 1376-1380 (1971).
    • (1971) J. Pharm. Sci. , vol.60 , pp. 1376-1380
    • Chiou, W.L.1    Riegelman, S.2
  • 12
    • 0015123293 scopus 로고
    • Decrease of tetracycline absorption in man by sodium bicarbonate
    • W. H. Barr, J. Adir, and L. Garrettson: Decrease of tetracycline absorption in man by sodium bicarbonate Clin. Pharmacol. Ther. 12, 779-784 (1971).
    • (1971) Clin. Pharmacol. Ther. , vol.12 , pp. 779-784
    • Barr, W.H.1    Adir, J.2    Garrettson, L.3
  • 13
    • 0021233529 scopus 로고
    • Mechanisms of bile formation, hepatic uptake, and biliary excretion
    • C. D. Klaassen and J. B. Watkins: Mechanisms of bile formation, hepatic uptake, and biliary excretion. Pharmacol. Rev. 36, 1-67 (1984).
    • (1984) Pharmacol. Rev. , vol.36 , pp. 1-67
    • Klaassen, C.D.1    Watkins, J.B.2
  • 15
    • 0015257761 scopus 로고
    • The enterohepatic circulation
    • R. H. Dowling: The enterohepatic circulation. Gastroenterology 62, 122-140 (1972).
    • (1972) Gastroenterology , vol.62 , pp. 122-140
    • Dowling, R.H.1
  • 16
    • 0014027584 scopus 로고
    • Rate of dissolution of griseofulvin and hexoesterol in bile salt solutions
    • T. R. Bates, M. Gibaldi, and J. L. Kanig: Rate of dissolution of griseofulvin and hexoesterol in bile salt solutions. Nature 210, 1331-1332 (1966).
    • (1966) Nature , vol.210 , pp. 1331-1332
    • Bates, T.R.1    Gibaldi, M.2    Kanig, J.L.3
  • 17
    • 0013877394 scopus 로고
    • Solubilizing properties of bile salt solution. I. Effect of temperature and bile salt concentration on solubilization of glutethimide. griseofulvin. and hexesterol
    • T. R. Bates, M. Gibaldi, and J. L. Kanig: Solubilizing properties of bile salt solution. I. Effect of temperature and bile salt concentration on solubilization of glutethimide. griseofulvin. and hexesterol. J. Pharm. Sci. 55, 191-199 (1966).
    • (1966) J. Pharm. Sci. , vol.55 , pp. 191-199
    • Bates, T.R.1    Gibaldi, M.2    Kanig, J.L.3
  • 18
    • 0013951569 scopus 로고
    • Solubilizing properties of bile sail solution. II. Effect of inorganic electrolyte, lipids. and a mixed bile salt system on solubulization of glutethimide, griseofulvin, and hexesterol
    • T. R. Bates, M. Gibaldi, and J. L. Kanig: Solubilizing properties of bile sail solution. II. Effect of inorganic electrolyte, lipids. and a mixed bile salt system on solubulization of glutethimide, griseofulvin, and hexesterol. J. Pharm. Sci. 55, 901-906 (1966).
    • (1966) J. Pharm. Sci. , vol.55 , pp. 901-906
    • Bates, T.R.1    Gibaldi, M.2    Kanig, J.L.3
  • 19
    • 0022398863 scopus 로고
    • Influence of bile on the gastrointestinal absorption of phenytoin in rats
    • D. Shinkuma, T. Hamagchi, Y. Yamanaka, N. Mizuno, and N. Yata: Influence of bile on the gastrointestinal absorption of phenytoin in rats. Chem. Pharm. Bull. 33, 5023-5072 (1985).
    • (1985) Chem. Pharm. Bull. , vol.33 , pp. 5023-5072
    • Shinkuma, D.1    Hamagchi, T.2    Yamanaka, Y.3    Mizuno, N.4    Yata, N.5
  • 20
    • 0028069730 scopus 로고
    • Pharmacokinetics analysis of enterohepatic circulation of buprenorphine and its active metabolite, norbuprenorphine, in rats
    • M. Ohtani, H. Kotani, K. Uchino, Y. Sawada, and T. Iga: Pharmacokinetics analysis of enterohepatic circulation of buprenorphine and its active metabolite, norbuprenorphine, in rats. Drug Metab. Dispos. 22, 2-7 (1994).
    • (1994) Drug Metab. Dispos. , vol.22 , pp. 2-7
    • Ohtani, M.1    Kotani, H.2    Uchino, K.3    Sawada, Y.4    Iga, T.5
  • 22
    • 0028244316 scopus 로고
    • A new analysis method for disposition kinetics of enterohepatic circulation of diclofenac in rats
    • T. Fukuyama, K. Yamaoka, Y. Ohata, and T. Nakagawa: A new analysis method for disposition kinetics of enterohepatic circulation of diclofenac in rats. Drug Metab. Dispos. 22, 479-485 (1994).
    • (1994) Drug Metab. Dispos. , vol.22 , pp. 479-485
    • Fukuyama, T.1    Yamaoka, K.2    Ohata, Y.3    Nakagawa, T.4
  • 24
    • 0024259968 scopus 로고
    • Pharmacokinetics and enterohepatic circulation of 2-n-propyl-4-pentenoic acid in the rat
    • K. Singh, J. M. Orr, and F. S. Abbot: Pharmacokinetics and enterohepatic circulation of 2-n-propyl-4-pentenoic acid in the rat. Drug Metab. Dispos. 16, 848-852 (1988).
    • (1988) Drug Metab. Dispos. , vol.16 , pp. 848-852
    • Singh, K.1    Orr, J.M.2    Abbot, F.S.3
  • 25
    • 0023259929 scopus 로고
    • An equation for the systemic availability of drugs undergoing simultaneous enterohepatic cycling, first-pass metabolism, and intestinal elimination
    • T. A. Shepard and R. H. Reuning: An equation for the systemic availability of drugs undergoing simultaneous enterohepatic cycling, first-pass metabolism, and intestinal elimination. Pharm. Res. 4, 195-199 (1987).
    • (1987) Pharm. Res. , vol.4 , pp. 195-199
    • Shepard, T.A.1    Reuning, R.H.2
  • 26
    • 0029032830 scopus 로고
    • Evaluation of intestinal absorption into the portal system in enterohepatic circulation by measuring the difference in portal-venous blood concentrations of diclofenac
    • K. Tabata, K. Yamaoka, T. Fukuyama, and T. Nakagawa: Evaluation of intestinal absorption into the portal system in enterohepatic circulation by measuring the difference in portal-venous blood concentrations of diclofenac. Pharm. Res. 12, 880-883 (1995).
    • (1995) Pharm. Res. , vol.12 , pp. 880-883
    • Tabata, K.1    Yamaoka, K.2    Fukuyama, T.3    Nakagawa, T.4
  • 27
    • 0029011942 scopus 로고
    • Method to estimate the rate and extent of intestinal absorption in conscious rats using an absorption probe and portal blood sampling
    • D. J. Hoffman, T. Seifert, A. Borre, and H. N. Nellans: Method to estimate the rate and extent of intestinal absorption in conscious rats using an absorption probe and portal blood sampling. Pharm. Res. 12, 889-894 (1995).
    • (1995) Pharm. Res. , vol.12 , pp. 889-894
    • Hoffman, D.J.1    Seifert, T.2    Borre, A.3    Nellans, H.N.4
  • 28
    • 0029047852 scopus 로고
    • Active transport of 3-o-methyl-glucose by the small intestines in chronically catheterized rats
    • M. R. Uhing and R. E. Kimura: Active transport of 3-o-methyl-glucose by the small intestines in chronically catheterized rats. J. Clin. Invest. 95, 2799-2805 (1995).
    • (1995) J. Clin. Invest. , vol.95 , pp. 2799-2805
    • Uhing, M.R.1    Kimura, R.E.2
  • 29
    • 0015466662 scopus 로고
    • Drug absorption and metabolism study by use of portal vein infusion in the rat I. Pyloric vein cannulation and its application to study of first-pass effect on bioavailability of propranolol
    • T. Suzuki, Y. Saitoh, S. Isozaki, and R. Ishida: Drug absorption and metabolism study by use of portal vein infusion in the rat I. Pyloric vein cannulation and its application to study of first-pass effect on bioavailability of propranolol Chem. Pharm. Bull. 20, 2731-2735 (1972).
    • (1972) Chem. Pharm. Bull. , vol.20 , pp. 2731-2735
    • Suzuki, T.1    Saitoh, Y.2    Isozaki, S.3    Ishida, R.4
  • 30
    • 0023804452 scopus 로고
    • A rapid and sensitive high-performance liquid Chromatographic method for the determination of diclofenac sodium in serum and its use in pharmacokinetic studies
    • Y. M. El-Sayed, M. E. Abdel-Hameed, M. S. Suleiman, and N. M. Najib: A rapid and sensitive high-performance liquid Chromatographic method for the determination of diclofenac sodium in serum and its use in pharmacokinetic studies. J. Pharm. Pharmacol. 40, 727-729 (1988).
    • (1988) J. Pharm. Pharmacol. , vol.40 , pp. 727-729
    • El-Sayed, Y.M.1    Abdel-Hameed, M.E.2    Suleiman, M.S.3    Najib, N.M.4
  • 31
    • 0027275566 scopus 로고
    • Physiological parameters in laboratory animals and humans
    • B. Davies and T. Morris: Physiological parameters in laboratory animals and humans. Pharm. Res. 10, 1093-1095 (1993).
    • (1993) Pharm. Res. , vol.10 , pp. 1093-1095
    • Davies, B.1    Morris, T.2
  • 34
    • 0025114570 scopus 로고
    • Statistical moment and disposition parameters in a local perfusion system under mammillary nonequilibrium condition
    • T. Kakutani, E. Nara, and M. Hashida: Statistical moment and disposition parameters in a local perfusion system under mammillary nonequilibrium condition. J. Pharmacokinet. Biopharm. 18, 449-458 (1990).
    • (1990) J. Pharmacokinet. Biopharm. , vol.18 , pp. 449-458
    • Kakutani, T.1    Nara, E.2    Hashida, M.3


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