Cardiac and gastric effects of histamine H2 receptor antagonists: No evidence for a correlation between lipophilicity and receptor affinity

British Journal of Pharmacology

Volumn 118, Issue 7, 1996, Pages 1813-1821

  Coruzzi, G ^a   Adami, M ^a   Pozzoli, C ^b   Giorgi, F ^a   Bertaccini, G ^a  

^a UNIVERSITY OF PARMA   (Italy)

^b Sigma Tau SpA   (Italy)

Author keywords

Aminopotentidine; Compound SK and F 92857; Heart; Histamine H2 receptors; Iodoaminopotentidine; Lipophilicity; Stomach

Indexed keywords

AMINOPOTENTIDINE; HISTAMINE; HISTAMINE H2 RECEPTOR ANTAGONIST; IODOAMINOPOTENTIDINE I 125; RANITIDINE; SKF 92857; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; COMPETITIVE INHIBITION; CONCENTRATION RESPONSE; CONTROLLED STUDY; FEMALE; GUINEA PIG; HEART; HEART PAPILLARY MUSCLE; IONIZATION; LIPOPHILICITY; MALE; MOLECULE; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY; REVERSED PHASE HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; STOMACH; STOMACH ACID SECRETION; STOMACH FUNDUS;

EID: 0030012401     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1476-5381.1996.tb15608.x     Document Type: Article

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