메뉴 건너뛰기




Volumn 117, Issue 8, 1996, Pages 1645-1652

KW-3902, a selective high affinity antagonist for adenosine A1 receptors

Author keywords

8 (Noradamantan 3 yl) 1,3 dipropylxanthine (KW 3902); A1 and A2 receptors; A1 antagonists; Adenosine receptors; Cyclic AMP; DPCPX

Indexed keywords

2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); 8 (2 NOR 1 ADAMANTYL) 1,3 DIPROPYLXANTHINE; ADENOSINE A1 RECEPTOR; ADENOSINE A1 RECEPTOR ANTAGONIST; ADENOSINE A2 RECEPTOR; CYCLIC AMP; FORSKOLIN; RADIOLIGAND;

EID: 0030011960     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1476-5381.1996.tb15335.x     Document Type: Article
Times cited : (38)

References (46)
  • 2
    • 0023161116 scopus 로고
    • 1 muscarinic receptor subtype between peripheral lung and cerebral cortex demonstrated by the selective antagonist AF-DX 116
    • 1 muscarinic receptor subtype between peripheral lung and cerebral cortex demonstrated by the selective antagonist AF-DX 116. Life Sci., 41, 491-496.
    • (1987) Life Sci. , vol.41 , pp. 491-496
    • Bloom, J.W.1    Halonen, M.2    Seaver, N.A.3    Yamamura, H.I.4
  • 11
    • 0022997406 scopus 로고
    • Adenosine A1 receptors in mammalian brain: Species differences in their interactions with agonists and antagonists
    • FERKANY, J.W., VALENTINE, H.L., STONE, G.A. & WILLIAMS, M. (1986). Adenosine A1 receptors in mammalian brain: Species differences in their interactions with agonists and antagonists. Drug Dev. Res., 9, 85-93.
    • (1986) Drug Dev. Res. , vol.9 , pp. 85-93
    • Ferkany, J.W.1    Valentine, H.L.2    Stone, G.A.3    Williams, M.4
  • 16
    • 0017159337 scopus 로고
    • Alpha-noradrenergic receptor binding in mammalian brain: Differential labeling of agonist and antagonist states
    • GREENBERG, D.A., U'PRICHARD, D.C. & SNYDER, S.H. (1976). Alpha-noradrenergic receptor binding in mammalian brain: differential labeling of agonist and antagonist states. Life Sci., 19, 69-76.
    • (1976) Life Sci. , vol.19 , pp. 69-76
    • Greenberg, D.A.1    U'Prichard, D.C.2    Snyder, S.H.3
  • 17
    • 0022544512 scopus 로고
    • 3H]Xanthine amine congener of 1,3-dipropyl-8-phenylxanthine: An antagonist radioligand for adenosine receptors
    • 3H]Xanthine amine congener of 1,3-dipropyl-8-phenylxanthine: an antagonist radioligand for adenosine receptors. Proc. Natl. Acad. Sci. U.S.A., 83, 4089-4093.
    • (1986) Proc. Natl. Acad. Sci. U.S.A. , vol.83 , pp. 4089-4093
    • Jacobson, K.A.1    Ukena, D.2    Kirk, K.L.3    Daly, J.W.4
  • 19
    • 0023795507 scopus 로고
    • Assay of cyclic nucleotide phosphodiesterase using radiolabeled and fluorescent substrates
    • ed. Corbin J.D. & Johnson, R.A. New York: Academic Press
    • KINCAID, R.L. & MANGANIELLO, V.C. (1988). Assay of cyclic nucleotide phosphodiesterase using radiolabeled and fluorescent substrates. In Methods in Enzymology. ed. Corbin J.D. & Johnson, R.A. Vol. 159, pp. 457-462. New York: Academic Press.
    • (1988) Methods in Enzymology , vol.159 , pp. 457-462
    • Kincaid, R.L.1    Manganiello, V.C.2
  • 21
    • 0025897566 scopus 로고
    • CD3-dependent increase in cyclic AMP in human T-cells following stimulation of the CD2 receptor
    • KVANTA, A., JONDAL, M. & FREDHOLM, B.B. (1991). CD3-dependent increase in cyclic AMP in human T-cells following stimulation of the CD2 receptor. Biochim. Biophys. Acta, 1093, 178-183.
    • (1991) Biochim. Biophys. Acta , vol.1093 , pp. 178-183
    • Kvanta, A.1    Jondal, M.2    Fredholm, B.B.3
  • 22
    • 0019394690 scopus 로고
    • 3H]spiperone to rat striatal membranes: Involvement of surface phenomena versus multiple binding sites
    • 3H]spiperone to rat striatal membranes: Involvement of surface phenomena versus multiple binding sites. J. Neurochem., 36, 201-219.
    • (1981) J. Neurochem. , vol.36 , pp. 201-219
    • Leysen, J.E.1    Gommeren, W.2
  • 25
    • 0023751273 scopus 로고
    • Identification of putative high affinity nicotinic receptors on cultured cortical neurons
    • LIPPIELLO, P.M. & FERNANDES, K.G. (1988). Identification of putative high affinity nicotinic receptors on cultured cortical neurons. J. Pharmacol. Exp. Ther., 246, 409-416.
    • (1988) J. Pharmacol. Exp. Ther. , vol.246 , pp. 409-416
    • Lippiello, P.M.1    Fernandes, K.G.2
  • 29
    • 0022005744 scopus 로고
    • Analysis of radioligand binding experiments: A collection of computer programs for the IBM PC
    • MCPHERSON, G.A. (1995). Analysis of radioligand binding experiments: A collection of computer programs for the IBM PC. J. Pharmacol. Methods, 14, 213-228.
    • (1995) J. Pharmacol. Methods , vol.14 , pp. 213-228
    • Mcpherson, G.A.1
  • 30
    • 0025395303 scopus 로고
    • Expression of human beta-interferon in Namalwa KJM-1 which was adapted to serum-free medium
    • MIYAJI, H., MIZUKAMI, T., HOSOI, S., SATO, S., FUJIYOSHI, N. & ITOH, S. (1990). Expression of human beta-interferon in Namalwa KJM-1 which was adapted to serum-free medium. Cytotechnology, 3, 133-140.
    • (1990) Cytotechnology , vol.3 , pp. 133-140
    • Miyaji, H.1    Mizukami, T.2    Hosoi, S.3    Sato, S.4    Fujiyoshi, N.5    Itoh, S.6
  • 32
    • 0019061918 scopus 로고
    • LIGAND, a versatile computerized approach for characterization of ligand-binding systems
    • MUNSON, P.J. & RODBARD, D. (1980). LIGAND, a versatile computerized approach for characterization of ligand-binding systems. Anal. Biochem., 107, 220-239.
    • (1980) Anal. Biochem. , vol.107 , pp. 220-239
    • Munson, P.J.1    Rodbard, D.2
  • 37
    • 0026024245 scopus 로고
    • Adenosine receptors and signaling in the kidney
    • SPIELMAN, W.S. & AREND, L.J. (1991). Adenosine receptors and signaling in the kidney. Hypertension, 17, 117-130.
    • (1991) Hypertension , vol.17 , pp. 117-130
    • Spielman, W.S.1    Arend, L.J.2
  • 38
    • 4244042273 scopus 로고
    • A proposed role for adenosine in the regulation of renal hemodynamics and renin release
    • SPIELMAN, W.S. & THOMPSON, C.I. (1982). A proposed role for adenosine in the regulation of renal hemodynamics and renin release. Am. J. Physiol., 242, F423-F435.
    • (1982) Am. J. Physiol. , vol.242
    • Spielman, W.S.1    Thompson, C.I.2
  • 39
    • 0025092063 scopus 로고
    • Characterization and selective inhibition of cyclic nucleotide phosphodiesterase isozymes in canine tracheal smooth muscle
    • TORPHY, T.J. & CIESLINSKI, L.B. (1990). Characterization and selective inhibition of cyclic nucleotide phosphodiesterase isozymes in canine tracheal smooth muscle. Mol. Pharmacol., 37, 206-214.
    • (1990) Mol. Pharmacol. , vol.37 , pp. 206-214
    • Torphy, T.J.1    Cieslinski, L.B.2
  • 42
    • 0018634064 scopus 로고
    • Adenosine regulates via two different types of receptors, the accumulation of cyclic AMP in cultured brain cells
    • VAN CALKER, D., MÜLLER, M. & HAMPRECHT, B. (1979). Adenosine regulates via two different types of receptors, the accumulation of cyclic AMP in cultured brain cells. J. Neurochem., 33, 999-1005.
    • (1979) J. Neurochem. , vol.33 , pp. 999-1005
    • Van Calker, D.1    Müller, M.2    Hamprecht, B.3
  • 44
    • 0021971160 scopus 로고
    • Nitrobenzylthioinosine binding in brain: An interspecies study
    • VERMA, A. & MARANGOS, P.J. (1985). Nitrobenzylthioinosine binding in brain: an interspecies study. Life Sci., 36, 283-290.
    • (1985) Life Sci. , vol.36 , pp. 283-290
    • Verma, A.1    Marangos, P.J.2
  • 45
    • 0018332925 scopus 로고
    • 3H]muscimol, a potent γ-aminobutyric acid agonist, to rat brain synaptosomal membranes using a filtration assay
    • 3H]muscimol, a potent γ-aminobutyric acid agonist, to rat brain synaptosomal membranes using a filtration assay. J. Neurochem., 32, 713-718.
    • (1979) J. Neurochem. , vol.32 , pp. 713-718
    • Williams, M.1    Risley, E.A.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.