New methods for determining dissociation constants of agonist-receptor complexes

European Journal of Pharmacology

Volumn 303, Issue 3, 1996, Pages 235-246

  Venter, Daniel P ^a  

^a NORTH WEST UNIVERSITY   (South Africa)

Author keywords

agonist affinity; agonist antagonist combination, fixed; carbachol; new methods; spare receptor; tripitramine

Indexed keywords

CARBACHOL; MUSCARINIC M3 RECEPTOR; PARTIAL AGONIST; RECEPTOR RESERVE; TRIPITRAMINE;

AGONIST; ARTICLE; COMPETITIVE INHIBITION; CONCENTRATION RESPONSE; DISSOCIATION CONSTANT; DRUG ACTIVITY; DRUG ANTAGONISM; GUINEA PIG; ILEUM; PRIORITY JOURNAL; RECEPTOR AFFINITY; RECEPTOR BINDING; RECEPTOR INTRINSIC ACTIVITY; RECEPTOR OCCUPANCY; TECHNIQUE; THEORY;

EID: 0030008864     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(96)00075-1     Document Type: Article

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