Threedimensional solubility parameters and their use in characterising the permeation of drugs through the skin

Pharmazie

Volumn 51, Issue 5, 1996, Pages 337-341

  Groning R ^a   Braun, F J ^a  

^a UNIVERSITY OF MÜNSTER   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

ATROPINE; CHLORPHENIRAMINE; CODEINE; CORTICOSTEROID; CORTICOSTERONE; CORTISONE; DEXAMETHASONE; DIETHYLCARBAMAZINE; DIGITOXIN; ESTRADIOL; FENTANYL; GLYCERYL TRINITRATE; HYDROCORTISONE; HYDROMORPHONE; MORPHINE; PETHIDINE; PROGESTERONE; SCOPOLAMINE; SUFENTANIL; TESTOSTERONE;

ARTICLE; CONTROLLED STUDY; DRUG ABSORPTION; DRUG SOLUBILITY; HUMAN; IN VITRO STUDY; SKIN PERMEABILITY; THEORY;

ANALGESICS; CHEMISTRY, PHYSICAL; DIFFUSION; KINETICS; MODELS, CHEMICAL; SKIN ABSORPTION; SOLUBILITY; STEROIDS;

EID: 0030004786     PISSN: 00317144     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (38)

1. Kubinyi, H.. Pharm. Ztg. Wiss 4, 265 (1991)
2. Taylor, P. J.; in: Hansch, C. (Ed.): Comprehensive Medicinal Chemistry, vol. 4, p. 241, Pergamon Press, Oxford 1990
3. Baker, R.: Controlled Release of Biologically Active Agents, p. 33, Wiley, New York 1987
4. Leo, A.; Hansch, C ; Elkins, D.: Chem. Rev. 71, 525 (1971)
5. Chou, J. T.; Jurs, P. C.; in: Yalkowsky; Sinkula; Valvani (Eds.): Physical Chemical Properties of Drugs, p. 163, Marcel Dekker, New York 1980
6. Rekker, R. F.: The Hydrophobic Fragment Constant, Elsevier, New York 1977
7. Shinoda, K.: Principles of Solution and Solubility, Marcel Dekker, New York 1978
8. Hildebrand, J. H.; Prausnitz, J. M ; Scott, R L.: Regular and Related Solutions, Van Nostrand Reinhold, New York 1970
9. Hildebrand, J. H., Scott, R. L : The Solubility of Nonelectrolytes, Reinhold, New York 1950
10. Khali, S A.; Martin, A. N.. J Pharm. Sci. 56, 1225 (1967)
11. Micheals, A. S. et al.: AICHE J. 21, 1073 (1975)
12. Adjei, A. et al.: J. Pharm. Sci. 73, 742 (1984)
13. Liron, Z.; Cohen, S.. J. Pharm. Sci. 73, 538 (1984)
14. Barton, A. F. M.: CRC-Handbook of Solubility Parameters and Other Cohesion Parameters, CRC Press, Boca Raton 1983
15. Barton, A. F. M.: Pure Appl. Chem. 57, 905 (1985)
16. Snyder, L.: Chemtech. 10, 188 (1980)
17. Hansen, C.: I & EC Product Res. Devel. 8, 2 (1969)
18. Wu, P. L.; Beerbower, A.; Martin, A.: J. Pharm. Sci. 71, 1285 (1982)
19. Lhoest, G.: Pharm. Acta Helv. 48, 549 (1973)
20. Siddiqui, S. A.; Needles, H. L.: Textile Res. J 52, 570 (1982)
21. Roy, S. D.; Flynn, G. L.: Pharm. Res. 6, 825 (1989)
22. Scheuplein, R. J.; Blank, I H.: J. Invest. Dermatol. 60, 286 (1973)
23. Van Krevelen, D. W.; Hoftyzer, P. J.: Properties of Polymers, their Estimation and Correlation with Chemical Structure, Elsevier, Amsterdam 1976
24. Snyder, L.: Chemtech 9, 750 (1979)
25. Fuhrhop, J. H.: Bip-organische Chemie, Struktur, Reaktivität und Wechselwirkungen von Naturstoffen, Thieme, Stuttgart 1982
26. Moore, J. W.; Hummel, D O : Physikalische Chemie, de Gryter, Berlin 1983
27. Bagley, E. B.; Nelson, T. P.; Scigliano, J. M.: J. Paint Technol. 43, 35 (1971)
28. Fedor, R. F.. Polymer Engin. Sci. 14, 147 (1974)
29. Loth, H.: Acta Pharm Technol. 33, 3 (1987)
30. Lippold, B. C.: Acta Pharm. Technol. 27, 1 (1981)
31. Landmann, L.: Pharmazie uns Zeit 20, 155 (1991)
32. Stüttgen, G.; in: Rietbrock, N. (Ed.): Die Haut als Transportorgan für Arzneistoffe, p. 1, Steinkopff, Darmstadt 1990
33. Ebert, G.: Biopolymere, p. 102, Steinkopff, Darmstadt 1980
34. Osborne, D. W.: Pharm. Manuf. 41 (1986)
35. Feldman, R. J.; Maibach, H. I.: J. Invest. Dermatol. 52, 89 (1969)
36. Sachs, L.: Angewandte Statistik, Springer, Berlin-Heidelberg 1992
37. Michaels, A. S.; Chandrasekaran, S. K ; Shaw, J. E.: AICHE J. 21, 985 (1975)
38. Scheuplein, R. J.; Blank, I. H.; Brauner, G. J ; Mac Farlane, D. J.: J. Invest. Dermatol. 52, 63 (1969)