Microwave-induced 1,3-dipolar cycloaddition of 2-aroyl-aziridines

Tetrahedron Letters

Volumn 37, Issue 24, 1996, Pages 4203-4204

  Boruah, Anima ^a   Baruah, Bipul ^a   Prajapati, Dipak ^a   Sandhu, Jagir S ^a   Ghosh, Anil C ^a  

^a REGIONAL RESEARCH LABORATORY   (India)

Author keywords

[No Author keywords available]

Indexed keywords

2 BENZOYL 1 CYCLOHEXYL 3 PHENYLAZIRIDINE; AZIRIDINE DERIVATIVE; IMIDAZOLIDINE DERIVATIVE; OXAZOLIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG ISOLATION; ENVIRONMENTAL TEMPERATURE; ESTERIFICATION; HYDROLYSIS; INTERMETHOD COMPARISON; MICROWAVE RADIATION; PROTON NUCLEAR MAGNETIC RESONANCE; THIN LAYER CHROMATOGRAPHY;

EID: 0030004708     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/0040-4039(96)00795-2     Document Type: Article

References (11)

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2. For recent reviews on microwave irradiation see: Caddick, S., Tetrahedron, 1995, 51, 10403; Mingos, D.M. and Baghurst, D.R., Chem. Soc. Rev., 1991, 20, 1-47; Giguere, R.J. in Organic Synthesis: Theory and Application, JAI Press, 1989, 1, 103-172; Bose, A.K., Manhas, M.S., Ghosh, M., M., Raju, V.S., Bari, S.S., Newaz, S.N., Banik, B.K., Choudhury, A.G. and Borakat, K.J., J. Org. Chem., 1991, 56, 6968.
3. For recent reviews on microwave irradiation see: Caddick, S., Tetrahedron, 1995, 51, 10403; Mingos, D.M. and Baghurst, D.R., Chem. Soc. Rev., 1991, 20, 1-47; Giguere, R.J. in Organic Synthesis: Theory and Application, JAI Press, 1989, 1, 103-172; Bose, A.K., Manhas, M.S., Ghosh, M., M., Raju, V.S., Bari, S.S., Newaz, S.N., Banik, B.K., Choudhury, A.G. and Borakat, K.J., J. Org. Chem., 1991, 56, 6968.
4. For recent reviews on microwave irradiation see: Caddick, S., Tetrahedron, 1995, 51, 10403; Mingos, D.M. and Baghurst, D.R., Chem. Soc. Rev., 1991, 20, 1-47; Giguere, R.J. in Organic Synthesis: Theory and Application, JAI Press, 1989, 1, 103-172; Bose, A.K., Manhas, M.S., Ghosh, M., M., Raju, V.S., Bari, S.S., Newaz, S.N., Banik, B.K., Choudhury, A.G. and Borakat, K.J., J. Org. Chem., 1991, 56, 6968.
5. For recent reviews on microwave irradiation see: Caddick, S., Tetrahedron, 1995, 51, 10403; Mingos, D.M. and Baghurst, D.R., Chem. Soc. Rev., 1991, 20, 1-47; Giguere, R.J. in Organic Synthesis: Theory and Application, JAI Press, 1989, 1, 103-172; Bose, A.K., Manhas, M.S., Ghosh, M., M., Raju, V.S., Bari, S.S., Newaz, S.N., Banik, B.K., Choudhury, A.G. and Borakat, K.J., J. Org. Chem., 1991, 56, 6968.
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11. The reaction (entry 1) also proceeds smoothly when carried out under ultrasound in homogeneous medium.