Inhibition of type 4 cyclic nucleotide phosphodiesterase by 8-chloroxanthines

Archiv der Pharmazie

Volumn 329, Issue 4, 1996, Pages 205-208

  Arch, Jonathan R S ^b   Buckle, Derek R ^a   Connolly, Brendan J ^b   Faller, Andrew ^a   Fenwick, Ashley E ^b   Murray, Kenneth J ^b   Rami, Harshad K ^a   Smallridge, Mark S ^a   Smith, David G ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

^b The Frythe   (United Kingdom)

Author keywords

BRL 61063; inflammation; phosphodiesterase inhibition; phosphodiesterase isoenzymes; xanthine

Indexed keywords

8 BROMO 1,3 BIS(CYCLOPROPYLMETHYL) 7 (2 NAPHTHYLMETHYL)XANTHINE; 8 CYCLOPENTYL 1,3 DIPROPYLXANTHINE; ADENOSINE A1 RECEPTOR; BRL 61063; CYCLIC NUCLEOTIDE PHOSPHODIESTERASE; ISOENZYME; PHOSPHODIESTERASE INHIBITOR; ROLIPRAM; UNCLASSIFIED DRUG; XANTHINE DERIVATIVE;

ARTICLE; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; ENZYME INHIBITION; NONHUMAN; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

EID: 0029982441     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/ardp.19963290406     Document Type: Article

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