New intracellular calcium antagonists. I. Synthesis and pharmacological evaluation of 2,3,4,5-tetrahydro-1,5-benzothiazepine analogs

Yakugaku Zasshi

Volumn 116, Issue 2, 1996, Pages 106-124

  Ueyama, Naoto ^a   Wakabayashi, Shuichi ^a   Tomiyama, Tsuyoshi ^a  

^a Kotobuki Seiyaku Co Ltd   (Japan)

Author keywords

2,3,4,5 tetrahydro 1,5 benzothiazepine; calcium release; intracellular calcium antagonist; structure activity relationship

Indexed keywords

5 [N (3,4 DIMETHOXYPHENETHYL) BETA ALANYL] 2,3,4,5 TETRAHYDRO 1,5 BENZOTHIAZEPINE HYDROGEN FUMARATE; BENZOTHIAZEPINE DERIVATIVE; BENZOTHIAZOLE DERIVATIVE; CAFFEINE; CALCIUM ANTAGONIST; DILTIAZEM; GLYCERYL TRINITRATE; METHOXAMINE; NIFEDIPINE; VERAPAMIL;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTERY CONSTRICTION; ARTICLE; CALCIUM CELL LEVEL; CALCIUM TRANSPORT; CHEMICAL STRUCTURE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; RABBIT; SARCOPLASMIC RETICULUM; STRUCTURE ACTIVITY RELATION;

EID: 0029980725     PISSN: 00316903     EISSN: None     Source Type: Journal    
DOI: 10.1248/yakushi1947.116.2_106     Document Type: Article

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