Synthesis of new 1H-tetrazoles and 1,2,3-triazoles via reactions of 3(,5)-(di)chloro-2H-1,4-(benz)oxazin-2-ones with sodium azide or diazocompounds

Tetrahedron

Volumn 52, Issue 26, 1996, Pages 8813-8826

  Medaer, Bart P ^a   Van Aken, Koen J ^a   Hoornaert, Georges J ^a  

^a UNIVERSITY OF LEUVEN   (Belgium)

Author keywords

[No Author keywords available]

Indexed keywords

1,2,3 TRIAZOLE DERIVATIVE; 1,4 OXAZINE DERIVATIVE; TETRAZOLE DERIVATIVE;

ARTICLE; DRUG SYNTHESIS; PRIORITY JOURNAL; REACTION ANALYSIS;

EID: 0029951475     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/0040-4020(96)00423-1     Document Type: Article

References (13)

1. Medaer, B.; Van Aken, K.; Hoornaert, G. Tetrahedron Lett. 1994, 66, 9767.
2. Shimorori, H. et. al. Jpn. Kokai Tokkyo Koho, JP 01,113,372 1989, CA 111: 194777n.
3. Georgiev, S.; Loev, B.; Musser, J. U.S. Patent, US 4,276,292 1981.
4. Klaubert, D. J. Med. Chem. 1981, 24, 748.
5. Meerpoel, L.; Hoornaert, G. Synthesis 1990, 305.
6. Dickoré, K.; Sasse, K.; Bode, K.-D. Liebigs Ann. Chem. 1970, 70, 733.
7. Tisler, M. Synthesis 1973 123.
8. (a) Maury, G.; Paugam, J.; Paugam, R. J. Het. Chem. 1978, 15, 1041.
9. (b) Tennant, G.; Vevers, R. J. Chem. Soc., Chem. Commun. 1974, 671.
10. Lwowski, W. in "1,3-Dipolar Cycloaddition Chemistry"; Padwa, A. Ed.; Wiley Interscience: New York, 1984, volume 1, 559.
11. Könnecke, A.; Lippman E. Z. Chem. 1976, 16, 53.
12. Verhé, R.; DeKimpe, N. in "The chemistry of functional groups"; Patai, S.; Rappoport, Z. Eds, J. Wiley & Sons Ltd, 1983, Supplement D, Chapter 19.
13. Synthetical procedure: see De Kimpe, N.; Verhé, R.; De Buyck, L.; Moëns, L.; Schamp, N. Synthesis 1982, 43.