메뉴 건너뛰기




Volumn 39, Issue 1-2, 1996, Pages 198-206

Regional variability in changes in 5-HT2A receptor mRNA levels in rat brain following irreversible inactivation with EEDQ 1

Author keywords

5 HT2A mRNA; 5 HT2A receptor; Autoradiography; Hybridization, in situ; N ethoxycarbonyl 2 ethoxy 1,2 dihydroquinoline; Receptor regulation

Indexed keywords

2 ETHOXY 1(2H) QUINOLINECARBOXYLIC ACID ETHYL ESTER; KETANSERIN; MESSENGER RNA; PHOSPHORUS; SEROTONIN 2A RECEPTOR; TRITIUM;

EID: 0029938668     PISSN: 0169328X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0169-328X(96)00024-1     Document Type: Article
Times cited : (5)

References (46)
  • 4
    • 0023162109 scopus 로고
    • 2 receptor recovery in mature and senescent rat brain after irreversible receptor modification: Effect of chronic reserpine treatment
    • 2 receptor recovery in mature and senescent rat brain after irreversible receptor modification: effect of chronic reserpine treatment, J. Pharmacol. Exp. Ther., 243 (1987) 69-75.
    • (1987) J. Pharmacol. Exp. Ther. , vol.243 , pp. 69-75
    • Battaglia, G.1    Norman, A.B.2    Creese, I.3
  • 6
    • 0014511179 scopus 로고
    • The mechanism of irreversible adrenergic blockade by N-carbethoxydihydroquinolines. Model studies with typical serine hydrolases
    • Belleau, B., DiTullio, V. and Godin, D., The mechanism of irreversible adrenergic blockade by N-carbethoxydihydroquinolines. Model studies with typical serine hydrolases. Biochem. Pharmacol., 18 (1969) 1039-1044.
    • (1969) Biochem. Pharmacol. , vol.18 , pp. 1039-1044
    • Belleau, B.1    DiTullio, V.2    Godin, D.3
  • 7
    • 0025944626 scopus 로고
    • 2 receptor mRNA in response to haloperidol treatment: A quantitative in situ hybridization study
    • 2 receptor mRNA in response to haloperidol treatment: a quantitative in situ hybridization study. Neuroscience, 45 (1991) 117-126.
    • (1991) Neuroscience , vol.45 , pp. 117-126
    • Bernard, V.1    Le Moine, C.2    Bloch, B.3
  • 8
    • 0019843739 scopus 로고
    • Multiple serotonin receptors: Regional distribution and effect of raphe lesions
    • Blackshear, M.A., Steranka, L.R. and Sanders-Bush, E., Multiple serotonin receptors: regional distribution and effect of raphe lesions. Eur. J. Pharmacol., 76 (1981) 325-334.
    • (1981) Eur. J. Pharmacol. , vol.76 , pp. 325-334
    • Blackshear, M.A.1    Steranka, L.R.2    Sanders-Bush, E.3
  • 13
    • 0022183592 scopus 로고
    • The influence of ritanserin, a serotonin antagonist, in anxiety disorders: A double-blind placebo-controlled study versus lorazepam
    • Ceulemans, D.L.S., Hoppenbrouwers, M.-L.J.A., Gelders, Y.G. amd Reyntjens, A.J.M., The influence of ritanserin, a serotonin antagonist, in anxiety disorders: a double-blind placebo-controlled study versus lorazepam. Pharmacopsychiatry, 18 (1985) 303-305.
    • (1985) Pharmacopsychiatry , vol.18 , pp. 303-305
    • Ceulemans, D.L.S.1    Hoppenbrouwers, M.-L.J.A.2    Gelders, Y.G.3    Reyntjens, A.J.M.4
  • 14
    • 0039166383 scopus 로고
    • Mechanism of cholinergic antagonism by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ)
    • Chang, K.J., Moran, J.F. and Triggle, D.J., Mechanism of cholinergic antagonism by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ). Pharmacol. Res. Commun., 2 (1970) 63-66.
    • (1970) Pharmacol. Res. Commun. , vol.2 , pp. 63-66
    • Chang, K.J.1    Moran, J.F.2    Triggle, D.J.3
  • 15
    • 0023275768 scopus 로고
    • Central serotonin receptors: Effector systems, physiological roles and regulation
    • Conn, P.J. and Sanders-Bush, E., Central serotonin receptors: effector systems, physiological roles and regulation, Psychopharmacology, 92 (1987) 267-277.
    • (1987) Psychopharmacology , vol.92 , pp. 267-277
    • Conn, P.J.1    Sanders-Bush, E.2
  • 16
    • 0023952199 scopus 로고
    • Ketanserin binds to the monoamine transporter of chromaffin granules and of synaptic vesicles
    • Darchen, F., Scherman, D., Laduron, P.M. and Henry, J. -P., Ketanserin binds to the monoamine transporter of chromaffin granules and of synaptic vesicles. Mol. Pharmacol., 33 (1988) 672-677.
    • (1988) Mol. Pharmacol. , vol.33 , pp. 672-677
    • Darchen, F.1    Scherman, D.2    Laduron, P.M.3    Henry, J.-P.4
  • 17
    • 0024380377 scopus 로고
    • 2 and beta-adrenergic receptors following noradrenergic or serotonergic denervation
    • 2 and beta-adrenergic receptors following noradrenergic or serotonergic denervation. J. Neural Transm., 44 (1989) 1419-1427.
    • (1989) J. Neural Transm. , vol.44 , pp. 1419-1427
    • Eison, A.S.1    Eison, M.S.2    Yocca, F.D.3    Gianutsos, G.4
  • 18
    • 0027944168 scopus 로고
    • 2A receptors in P11 cells through a post-transcriptional mechanism requiring activation of protein kinase C
    • 2A receptors in P11 cells through a post-transcriptional mechanism requiring activation of protein kinase C. J. Biol. Chem., 269 (1994) 31850-31857.
    • (1994) J. Biol. Chem. , vol.269 , pp. 31850-31857
    • Ferry, R.C.1    Unsworth, C.D.2    Artymyshyn, R.3    Molinoff, P.B.4
  • 19
    • 0023630323 scopus 로고
    • 2 receptors throughout the rat central nervous system using quantitative autoradiography
    • 2 receptors throughout the rat central nervous system using quantitative autoradiography. Brain Res., 421 (1987) 263-279.
    • (1987) Brain Res. , vol.421 , pp. 263-279
    • Fischette, C.T.1    Nock, B.2    Renner, K.3
  • 20
    • 0002867336 scopus 로고
    • Regulation of serotonin receptors and responsiveness in the brain
    • E. Sanders-Bush (Rd.), Humana Press
    • Frazer, A., Offord, S.J. and Lucki, I., Regulation of serotonin receptors and responsiveness in the brain. In: E. Sanders-Bush (Rd.), The Serotonin Receptors, Humana Press, 1988, pp. 319-362.
    • (1988) The Serotonin Receptors , pp. 319-362
    • Frazer, A.1    Offord, S.J.2    Lucki, I.3
  • 21
    • 0024366801 scopus 로고
    • Thymosthenic agents, a novel approach in the treatment of schizophrenia
    • Gelders, Y.G., Thymosthenic agents, a novel approach in the treatment of schizophrenia. Br. J. Psychiat., Suppl. 11 (1989) 33-36.
    • (1989) Br. J. Psychiat. , vol.11 , Issue.SUPPL. 11 , pp. 33-36
    • Gelders, Y.G.1
  • 22
    • 0028290841 scopus 로고
    • Differential effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on various 5-HT receptor binding sites in the rat brain
    • Gozlan, H., Laporte, A.-M., Thibault, S., Schechter, L.E., Bolanos, F. and Hamon, M., Differential effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on various 5-HT receptor binding sites in the rat brain, Neuropharmacology, 33 (1994) 423-431.
    • (1994) Neuropharmacology , vol.33 , pp. 423-431
    • Gozlan, H.1    Laporte, A.-M.2    Thibault, S.3    Schechter, L.E.4    Bolanos, F.5    Hamon, M.6
  • 23
    • 0024341172 scopus 로고
    • Agonist-induced destabilization of β-adrenergic receptor mRNA
    • Hadcock, J.R., Wang, H.-Y. and Malbon, C.C., Agonist-induced destabilization of β-adrenergic receptor mRNA. J. Biol. Chem., 264 (1989) 19928-19933.
    • (1989) J. Biol. Chem. , vol.264 , pp. 19928-19933
    • Hadcock, J.R.1    Wang, H.-Y.2    Malbon, C.C.3
  • 27
    • 0021893269 scopus 로고
    • 2 dopamine receptors by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline in vivo: Selective protection by neuroleptics
    • 2 dopamine receptors by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline in vivo: selective protection by neuroleptics. J. Pharmacol. Exp. Ther., 233 (1985) 656-662.
    • (1985) J. Pharmacol. Exp. Ther. , vol.233 , pp. 656-662
    • Meller, E.1    Bohmaker, K.2    Goldstein, M.3    Friedhoff, A.J.4
  • 28
    • 0025124833 scopus 로고
    • 2 receptor by in situ hybridization histochemistry. Correlation with the distribution of receptor sites
    • 2 receptor by in situ hybridization histochemistry. Correlation with the distribution of receptor sites. Brain Res., 524 (1990) 139-143.
    • (1990) Brain Res. , vol.524 , pp. 139-143
    • Mengod, G.1    Pompeiano, M.2    Martinez-Mir, I.3    Palacios, J.M.4
  • 30
    • 0022401097 scopus 로고
    • Quantitative autoradiographic mapping of serotonin receptors in rat brain. II. Serotonin-2 receptors
    • Pazos, A., Cortes, R. and Palacios, J.M., Quantitative autoradiographic mapping of serotonin receptors in rat brain. II. Serotonin-2 receptors. Brain Res., 346 (1985) 231-249.
    • (1985) Brain Res. , vol.346 , pp. 231-249
    • Pazos, A.1    Cortes, R.2    Palacios, J.M.3
  • 31
    • 0027382098 scopus 로고
    • In vivo EEDQ dose-dependently inactivates rat brain 5-HT receptors but not 5-HT uptake sites
    • Pinto, W. and G. Battaglia., In vivo EEDQ dose-dependently inactivates rat brain 5-HT receptors but not 5-HT uptake sites. NeuroReport, 5 (1993) 61-64.
    • (1993) NeuroReport , vol.5 , pp. 61-64
    • Pinto, W.1    Battaglia, G.2
  • 33
    • 0025923909 scopus 로고
    • 2 receptors in rat cortex. Studies with a putative selective agonist and an antagonist
    • 2 receptors in rat cortex. Studies with a putative selective agonist and an antagonist, Biochem. Pharmacol., 45 (1991) 1099-1105.
    • (1991) Biochem. Pharmacol. , vol.45 , pp. 1099-1105
    • Pranzatelli, M.R.1
  • 43
    • 0021683773 scopus 로고
    • Aortic recognition sites for serotonin (5-HT) are coupled to phospholipase C and modulate phosphatidylinositol turnover
    • Roth, B.L., Nakaki, T., Chuang, D.-M. and Costa, E., Aortic recognition sites for serotonin (5-HT) are coupled to phospholipase C and modulate phosphatidylinositol turnover. Neuropharmacology, 23 (1984) 1223-1225.
    • (1984) Neuropharmacology , vol.23 , pp. 1223-1225
    • Roth, B.L.1    Nakaki, T.2    Chuang, D.-M.3    Costa, E.4
  • 44
    • 0028290842 scopus 로고
    • Lack of effects of antidepressant drugs on the levels of mRNAs encoding serotonergic receptors, synthetic enzymes and 5-HT transporter
    • Spurlock, G., Buckland, P., O'Donovan, M. and McGuffin, P., Lack of effects of antidepressant drugs on the levels of mRNAs encoding serotonergic receptors, synthetic enzymes and 5-HT transporter, Neuropharmacology, 3 (1994) 433-440.
    • (1994) Neuropharmacology , vol.3 , pp. 433-440
    • Spurlock, G.1    Buckland, P.2    O'Donovan, M.3    McGuffin, P.4
  • 45
    • 0028235547 scopus 로고
    • Antagonist-mediated down-regulation of 5-hydroxytryptamine type 2 receptor gene expression: Modulation of transcription
    • Toth, M. and Shenk, T., Antagonist-mediated down-regulation of 5-hydroxytryptamine type 2 receptor gene expression: modulation of transcription, Mol. Pharmacol., 45 (1994) 1095-1100.
    • (1994) Mol. Pharmacol. , vol.45 , pp. 1095-1100
    • Toth, M.1    Shenk, T.2
  • 46
    • 0026610708 scopus 로고
    • 2 dopamine receptor mRNA during ontogenesis, lesion and chronic antagonist treatment
    • 2 dopamine receptor mRNA during ontogenesis, lesion and chronic antagonist treatment. Life Sci., 50 (1991) 383-396.
    • (1991) Life Sci. , vol.50 , pp. 383-396
    • Xu, S.1    Monsma F.J., Jr.2    Sibley, D.R.3    Creese, I.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.