Synthesis and anti-inflammatory evaluation of new sulfamoylheterocarboxylic derivatives

Archiv der Pharmazie

Volumn 329, Issue 5, 1996, Pages 229-238

  Díaz, Juan A ^a,d   Morante, M Esther ^a   Vega, Salvador ^a   Darias, Victoriano ^b   Abdala, Susana ^b   Delgado, Laura ^b   De Las Heras, Beatriz ^c   Villar, Angel ^c   Vivas, José María ^c  

^a INSTITUTO DE QUÍMICA MÉDICA   (Spain)

^b UNIVERSIDAD DE LA LAGUNA   (Spain)

^c UNIVERSIDAD COMPLUTENSE DE MADRID   (Spain)

^d NONE   (Spain)

Author keywords

analgesic activity; anti inflammatory activity; sulfamoylthiophene and sulfamoylpyrazole carboxylic derivatives

Indexed keywords

ACETYLSALICYLIC ACID; AMPHETAMINE; BETAMETHASONE; DEXAMETHASONE; DIAZEPAM; IBUPROFEN; INDOMETACIN; NONSTEROID ANTIINFLAMMATORY AGENT; PIROXICAM; PYRAZOLE DERIVATIVE; THIOPHENE DERIVATIVE;

ANALGESIA; ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIINFLAMMATORY ACTIVITY; ARTICLE; BEHAVIOR; BLEEDING TIME; CONTROLLED STUDY; DRUG SCREENING; DRUG SYNTHESIS; LOCOMOTION; MOUSE; NONHUMAN; ORAL DRUG ADMINISTRATION; PRIORITY JOURNAL; RAT;

ANALGESICS; ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; BLOOD COAGULATION; CARBOXYLIC ACIDS; FEMALE; MALE; MICE; MOTOR ACTIVITY; MUSCLE RELAXANTS, CENTRAL; RATS; RATS, WISTAR;

EID: 0029934819     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/ardp.19963290503     Document Type: Article

References (22)

1. J.E. Wallace, Gastroenterol. Clin. North. Am. 1992, 21, 631-641.
2. S. Vega, R. Madroñero, J.A. Díaz, F. Junquera, J. Alonso, V. Darias, L. Bravo, S. Abdallah, Eur. J. Med. Chem. 1988, 23, 329-334.
3. S. Vega, J. Alonso, J.A. Díaz, F. Junquera, C. Pérez, V. Darias, L. Bravo, S. Abdallah, Eur. J. Med. Chem. 1991, 26, 323-329.
4. V. Darias, S. Abdallah, M.L. Tello, L.D. Delgado, S. Vega, Arch. Pharm. 1994, 327, 779-783.
5. T.Y. Shen in Burger's Medicinal Chemistry (Ed.: M. E. Wolf), 4th ed., Wiley, New York, 1981, part 3.
6. th International Symposium on Medicinal Chemistry in Paris, France, September 19-23, 1994.
7. J.A. Díaz, S. Vega, J. Heterocyclic Chem. 1994, 31, 93-96.
8. S. Vega, J.A. Díaz, J. Heterocyclic Chem. 1993, 30, 1509-1512.
9. P.A. Rossy, W. Hoffmann, N. Müller, J. Org. Chem. 1980, 45, 617-620.
10. S. Irwin, Psychopharmacology (Berlin), 1968, 13, 222-257.
11. G. Levy, T. Tuschima, L.P. Amsel, Clin. Pharmacol. Ther. 1972, 13, 258-262.
12. C. A. Winter, E.A. Risler, G.W. Nuss, Proc. Soc. Exptl. Biol. Med. 1962, 111, 544-547.
13. K. Charalambous, B. de las Heras, J.R.S. Hoult, Agents Actions 1994, 41, 101-104.
14. W.E.C. Waker, D.D. Ulmer, B.L. Vallee, New Engl. J. Med. 1956, 225, 449-456.
15. M. Paya, P.A. Goodwin, B. de las Heras, J.R.S. Hoult, Biochem. Pharmacol. 1994, 48 (3), 445-451.
16. C. Corral, J. Lissavetzky, A. Valdeolmillos, L. Bravo, V. Darias, C. Sánchez-Mateo, Arzneim.-Forsch. 1992, 42, 896-900.
17. S. Courvoisier, R. Ducrot, L. Julou, in Psychotropic Drugs, (Eds: S. Garattini, V. Ghetti), Elsevier Publishing Co., Amsterdam, 1975, p. 373.
18. J.R. Boissier, J. Tardy, J.C. Diverres, Med. Exp. 1960, 3, 81-84.
19. J.T. Litchfield, F. and J. Wilcoxon, Pharmacol. Exptl. Ther. 1949, 96, 99-113.
20. E. Siegmund, R. Cadmus, G. Lu, Proc. Soc. Exptl. Biol. Med. 1957, 95, 729-731.
21. R.P. Carlson, L.O'Neill-Davis, J. Chang, A.J. Lewis, Agents and Actions 1985, 17, 2-12.
22. W.W. Duke, J. Am. Med. Assoc. 1910, 15, 1185-1193.