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Volumn 276, Issue 1, 1996, Pages 84-92

YM90K: Pharmacological characterization as a selective and potent α-amino-3-hydroxy-5-methylisoxazole-4-propionate/kainate receptor antagonist

Author keywords

[No Author keywords available]

Indexed keywords

6 (1 IMIDAZOLYL) 7 NITRO 2,3 QUINOXALINEDIONE; 6 CYANO 7 NITRO 2,3 QUINOXALINEDIONE; 6 NITRO 7 SULFAMOYLBENZO[F]QUINOXALINE 2,3 DIONE; ALPHA AMINO 3 HYDROXY 5 METHYL 4 ISOXAZOLEPROPIONIC ACID; AMPA RECEPTOR; KAINIC ACID; KAINIC ACID RECEPTOR; RECEPTOR BLOCKING AGENT;

EID: 0029927472     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (94)

References (65)
  • 2
    • 0018139770 scopus 로고
    • Muscimol binding in rat brain: Association with synaptic GABA receptors
    • BEAUMONT, K., CHILTON, W. S., YAMAMURA, H. I. AND ENNA, S. J.: Muscimol binding in rat brain: Association with synaptic GABA receptors. Brain Res. 148: 153-162, 1978.
    • (1978) Brain Res. , vol.148 , pp. 153-162
    • Beaumont, K.1    Chilton, W.S.2    Yamamura, H.I.3    Enna, S.J.4
  • 3
    • 0023856682 scopus 로고
    • The N-methyl-D-aspartate antagonists CGS 19755 and CPP reduce ischemic brain damage in gerbils
    • BOAST, C. A., GERHARDT, S. C., PASTOR, G., LEHMANN, J., ETIENNE, P. E. AND LIEBMAN, J. M.: The N-methyl-D-aspartate antagonists CGS 19755 and CPP reduce ischemic brain damage in gerbils. Brain Res. 442: 345-348, 1988.
    • (1988) Brain Res. , vol.442 , pp. 345-348
    • Boast, C.A.1    Gerhardt, S.C.2    Pastor, G.3    Lehmann, J.4    Etienne, P.E.5    Liebman, J.M.6
  • 5
    • 0023162156 scopus 로고
    • 3H]-kainic acid receptor binding by divalent cations correlates with ion affinity for the calcium channel
    • 3H]-kainic acid receptor binding by divalent cations correlates with ion affinity for the calcium channel. Neuropharmacology 26: 1247-1251, 1987.
    • (1987) Neuropharmacology , vol.26 , pp. 1247-1251
    • Braitman, D.J.1    Coyle, J.T.2
  • 6
    • 0025779342 scopus 로고
    • Delayed AMPA receptor blockade reduces cerebral infarction induced by focal ischemia
    • BUCHAN, A. M., XUE, D., HUANG, Z-G., SMITH, K. H. AND LESIUK, H.: Delayed AMPA receptor blockade reduces cerebral infarction induced by focal ischemia. Neuroreport 2: 473-476, 1991.
    • (1991) Neuroreport , vol.2 , pp. 473-476
    • Buchan, A.M.1    Xue, D.2    Huang, Z.-G.3    Smith, K.H.4    Lesiuk, H.5
  • 7
    • 0026752304 scopus 로고
    • Memory formation in day-old chicks requires NMDA but not non-NMDA glutamate receptors
    • BURCHULADZE, R. AND ROSE, S. P. R.: Memory formation in day-old chicks requires NMDA but not non-NMDA glutamate receptors. Eur. J. Neurosci. 4: 533-538, 1992.
    • (1992) Eur. J. Neurosci. , vol.4 , pp. 533-538
    • Burchuladze, R.1    Rose, S.P.R.2
  • 8
    • 0025603178 scopus 로고
    • Correlation between amino acid release and neuropathologic outcome in rat brain following middle cerebral artery occlusion
    • BUTCHER, S. P., BULLOCK, R., GRAHAM, D. I. AND MCCULLOCH, J.: Correlation between amino acid release and neuropathologic outcome in rat brain following middle cerebral artery occlusion. Stroke 21: 1727-1733, 1990.
    • (1990) Stroke , vol.21 , pp. 1727-1733
    • Butcher, S.P.1    Bullock, R.2    Graham, D.I.3    Mcculloch, J.4
  • 9
    • 0025789026 scopus 로고
    • The anticonvulsant effect of the non-NMDA antagonists, NBQX and GYKI 52466, in mice
    • CHAPMAN, A. G., SMITH, S. E. AND MELDRUM, B. S.: The anticonvulsant effect of the non-NMDA antagonists, NBQX and GYKI 52466, in mice. Epilepsy Res. 9: 92-96, 1991.
    • (1991) Epilepsy Res. , vol.9 , pp. 92-96
    • Chapman, A.G.1    Smith, S.E.2    Meldrum, B.S.3
  • 10
    • 0024829451 scopus 로고
    • Excitatory amino acid receptors in the vertebrate central nervous system
    • COLLINGRIDGE, G. L. AND LESTER, R. A. J.: Excitatory amino acid receptors in the vertebrate central nervous system. Pharmacol. Rev. 40: 143-210, 1989.
    • (1989) Pharmacol. Rev. , vol.40 , pp. 143-210
    • Collingridge, G.L.1    Lester, R.A.J.2
  • 11
    • 0023264133 scopus 로고
    • Anatomical organization of excitatory amino acid receptors and their pathways
    • COTMAN, C. W., MONAGHAN, D. T. AND OTTERSEN, O. P.: Anatomical organization of excitatory amino acid receptors and their pathways. Trends Neurosci. 10: 273-279, 1987.
    • (1987) Trends Neurosci. , vol.10 , pp. 273-279
    • Cotman, C.W.1    Monaghan, D.T.2    Ottersen, O.P.3
  • 12
    • 0023867358 scopus 로고
    • Anticonvulsant effects of some calcium entry blockers in DBA/2 mice
    • DE SARRO, G. B , MELDRUM, B. S. AND NISTICO, G.: Anticonvulsant effects of some calcium entry blockers in DBA/2 mice. Br. J. Pharmacol. 93: 247-256, 1988.
    • (1988) Br. J. Pharmacol. , vol.93 , pp. 247-256
    • De Sarro, G.B.1    Meldrum, B.S.2    Nistico, G.3
  • 14
    • 0026505691 scopus 로고
    • Inhibition of cisplatin-induced emesis in ferrets by the non-NMDA receptor antagonists NBQX and CNQX
    • FINK-JENSEN, A., JUDGE, M. E., HANSEN, J. B., JACOBSEN, P., TURSKI, L., OLNEY, J. AND HONORE, T.: Inhibition of cisplatin-induced emesis in ferrets by the non-NMDA receptor antagonists NBQX and CNQX. Neurosci. Lett. 137: 173-177, 1992.
    • (1992) Neurosci. Lett. , vol.137 , pp. 173-177
    • Fink-Jensen, A.1    Judge, M.E.2    Hansen, J.B.3    Jacobsen, P.4    Turski, L.5    Olney, J.6    Honore, T.7
  • 16
    • 0025784436 scopus 로고
    • The neuroprotective action of dizocilpine (MK-801) in the rat middle cerebral artery occlusion model of focal ischaemia
    • GILL, R., BHAZELL, C., WOODRUFF, G. N., KEMP, J. A.: The neuroprotective action of dizocilpine (MK-801) in the rat middle cerebral artery occlusion model of focal ischaemia. Br. J. Pharmacol. 103: 2030-2036, 1991.
    • (1991) Br. J. Pharmacol. , vol.103 , pp. 2030-2036
    • Gill, R.1    Bhazell, C.2    Woodruff, G.N.3    Kemp, J.A.4
  • 17
    • 0026710232 scopus 로고
    • The neuroprotective actions of 2,3-dihydroxy-6-nitro-7-sulfamoyl-benzo(F)quinoxaline (NBQX) in a rat focal ischaemia model
    • GILL, R., NORDHOLM, L. AND LODGE, D.: The neuroprotective actions of 2,3-dihydroxy-6-nitro-7-sulfamoyl-benzo(F)quinoxaline (NBQX) in a rat focal ischaemia model. Brain Res. 580: 35-43, 1992.
    • (1992) Brain Res. , vol.580 , pp. 35-43
    • Gill, R.1    Nordholm, L.2    Lodge, D.3
  • 18
    • 0025141246 scopus 로고
    • Changes in extracellular amino acid neurotransmitters produced by focal cerebral ischemia
    • GRAHAM, S. H., SHIRAISHI, K., PANTER, S. S., SIMON, R. P. AND FADEN, A. L.: Changes in extracellular amino acid neurotransmitters produced by focal cerebral ischemia. Neurosci. Lett. 110: 124-130, 1990.
    • (1990) Neurosci. Lett. , vol.110 , pp. 124-130
    • Graham, S.H.1    Shiraishi, K.2    Panter, S.S.3    Simon, R.P.4    Faden, A.L.5
  • 19
    • 0025923461 scopus 로고
    • 2+ permeability of KA-/ AMPA-gated glutamate receptor channels depends on subunit composition
    • 2+ permeability of KA-/ AMPA-gated glutamate receptor channels depends on subunit composition. Science 252: 851-853, 1991.
    • (1991) Science , vol.252 , pp. 851-853
    • Hollmann, M.1    Hartley, M.2    Heinemann, S.3
  • 23
    • 0021965716 scopus 로고
    • Highly sensitive assay for choline acetyltransferase activity by high-performance liquid chromatography with electrochemical detection
    • KANEDA, N. AND NAGATSU, T.: Highly sensitive assay for choline acetyltransferase activity by high-performance liquid chromatography with electrochemical detection. J. Chromatogr. 341: 23-30, 1985.
    • (1985) J. Chromatogr. , vol.341 , pp. 23-30
    • Kaneda, N.1    Nagatsu, T.2
  • 24
    • 1842366535 scopus 로고
    • Postischemic administration of YM900, a selective and potent α-amino-3-hydroxy-5-methylisoxazole-4-propionate (AMPA) receptor antagonist, prevents delayed neuronal death in gerbil hippocampus
    • KAWASAKI, S., YATSUGI, S., TAKAHASHI, M., KATO, M., KOSHIYA, K., SAKAMOTO, S. AND SHIMIZU-SASAMATA, M.: Postischemic administration of YM900, a selective and potent α-amino-3-hydroxy-5-methylisoxazole-4-propionate (AMPA) receptor antagonist, prevents delayed neuronal death in gerbil hippocampus. Jpn. J. Pharmacol. 60(suppl. 1): 284, 1993
    • (1993) Jpn. J. Pharmacol. , vol.60 , Issue.1 SUPPL. , pp. 284
    • Kawasaki, S.1    Yatsugi, S.2    Takahashi, M.3    Kato, M.4    Koshiya, K.5    Sakamoto, S.6    Shimizu-Sasamata, M.7
  • 25
    • 0020051129 scopus 로고
    • Delayed neuronal death in the gerbil hippocampus following ischemia
    • KIRINO, T.: Delayed neuronal death in the gerbil hippocampus following ischemia. Brain Res. 239: 57-69, 1982.
    • (1982) Brain Res. , vol.239 , pp. 57-69
    • Kirino, T.1
  • 26
    • 0026074931 scopus 로고
    • The AMPA receptor antagonist NBQX has antiparkinsonian effects in monoamine-depleted rats and MPTP-treated monkeys
    • KLOCKGETHER, T., TURSKI, L., HONORE, T., ZHANG, Z., GASH, D.M., KURLAN, R. AND GEEENMYRE, J. T.: The AMPA receptor antagonist NBQX has antiparkinsonian effects in monoamine-depleted rats and MPTP-treated monkeys. Ann. Neurol. 30: 717-723, 1991.
    • (1991) Ann. Neurol. , vol.30 , pp. 717-723
    • Klockgether, T.1    Turski, L.2    Honore, T.3    Zhang, Z.4    Gash, D.M.5    Kurlan, R.6    Geeenmyre, J.T.7
  • 27
    • 0023901123 scopus 로고
    • MK-801, a proposed noncompetitive antagonist of excitatory amino acid neurotransmission produces phencyclidine-like behavioral effects in pigeons, rats and rhesus monkeys
    • KOEK, W., WOOD, J. H. AND WINGER, G. D.: MK-801, a proposed noncompetitive antagonist of excitatory amino acid neurotransmission produces phencyclidine-like behavioral effects in pigeons, rats and rhesus monkeys. J. Pharmacol Exp. Ther. 245: 969-974, 1988.
    • (1988) J. Pharmacol Exp. Ther. , vol.245 , pp. 969-974
    • Koek, W.1    Wood, J.H.2    Winger, G.D.3
  • 29
    • 0026670676 scopus 로고
    • The non-NMDA glutamate antagonist NBQX blocks the local hippocampal toxicity of kainic acid, but not the diffuse extrahippocampal damage
    • LEES, G. J. AND LEONG, W.: The non-NMDA glutamate antagonist NBQX blocks the local hippocampal toxicity of kainic acid, but not the diffuse extrahippocampal damage. Neurosci Lett. 143: 39-42, 1992.
    • (1992) Neurosci Lett. , vol.143 , pp. 39-42
    • Lees, G.J.1    Leong, W.2
  • 30
    • 0025740632 scopus 로고
    • Kynurenic acid derivatives. Structure-activity relationships for excitatory amino acid antagonism and identification of potent and selective antagonists at the glycine site on the N-methyl-D-aspartate receptor
    • LEESON, P. D., BAKER, R , CARLING, R. W., CURTIS, N. R., MOORE, K. W., WILLIAMS, B. J., FOSTER, A. C., DONALD, A. E., KEMP, J. A. AND MARSHALL, G. R.: Kynurenic acid derivatives. Structure-activity relationships for excitatory amino acid antagonism and identification of potent and selective antagonists at the glycine site on the N-methyl-D-aspartate receptor. J. Med. Chem. 34: 1243-1252, 1991.
    • (1991) J. Med. Chem. , vol.34 , pp. 1243-1252
    • Leeson, P.D.1    Baker, R.2    Carling, R.W.3    Curtis, N.R.4    Moore, K.W.5    Williams, B.J.6    Foster, A.C.7    Donald, A.E.8    Kemp, J.A.9    Marshall, G.R.10
  • 32
    • 0027445864 scopus 로고
    • Treatment with an AMPA antagonist 12 hours following severe normothermic forebrain ischemia prevents CA1 neuronal injury
    • LI, H. AND BUCHAN, A M.: Treatment with an AMPA antagonist 12 hours following severe normothermic forebrain ischemia prevents CA1 neuronal injury. J. Cereb. Blood Flow Metab. 13: 933-939, 1993.
    • (1993) J. Cereb. Blood Flow Metab. , vol.13 , pp. 933-939
    • Li, H.1    Buchan, A.M.2
  • 33
    • 0025720689 scopus 로고
    • Inhibitory effect of 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX) on the micturition reflex in rat
    • MATSUMOTO, G., KAWATANI, M. AND TAKESHIGE, C.: Inhibitory effect of 6-cyano-7-nitroquinoxaline-2,3-dione (CNQX) on the micturition reflex in rat. Neurosci. Lett. 133: 211-214, 1991.
    • (1991) Neurosci. Lett. , vol.133 , pp. 211-214
    • Matsumoto, G.1    Kawatani, M.2    Takeshige, C.3
  • 34
    • 0027405774 scopus 로고
    • Cyclothiazide treatment unmasks AMPA excitotoxicity in rat primary hippocampal cultures
    • MAY, P. C. AND ROBINSON, P. M.: Cyclothiazide treatment unmasks AMPA excitotoxicity in rat primary hippocampal cultures. J. Neurochem. 60: 1171-1174, 1993.
    • (1993) J. Neurochem. , vol.60 , pp. 1171-1174
    • May, P.C.1    Robinson, P.M.2
  • 35
    • 0020516359 scopus 로고
    • A comparison of the anticonvulsant potency of (±)-2-amino-5-phosphonopentanoic acid and 2-amino-7-phosphonoheptanoic acid
    • MELDRUM, B. S., CROUCHER, M. J., CZUCZWAR, S. J., COLLINS, J. F., CURRY, K., JOSEPH, M. AND STONE, T. W.: A comparison of the anticonvulsant potency of (±)-2-amino-5-phosphonopentanoic acid and 2-amino-7-phosphonoheptanoic acid. Neuroscience. 9: 925-930, 1983.
    • (1983) Neuroscience , vol.9 , pp. 925-930
    • Meldrum, B.S.1    Croucher, M.J.2    Czuczwar, S.J.3    Collins, J.F.4    Curry, K.5    Joseph, M.6    Stone, T.W.7
  • 36
    • 0023176489 scopus 로고
    • 3H]-glutamate recognition site in synaptic plasma membranes
    • 3H]-glutamate recognition site in synaptic plasma membranes. J. Neurochem. 48: 1699-1708, 1987.
    • (1987) J. Neurochem. , vol.48 , pp. 1699-1708
    • Monahan, J.B.1    Michel, J.2
  • 38
    • 0025831124 scopus 로고
    • Non-NMDA antagonists protect against kainate more than AMPA toxicity in the rat hippocampus
    • MONCADA, C., ARVIN, B., LE PEILLET, E. AND MELDRUM, B. S.: Non-NMDA antagonists protect against kainate more than AMPA toxicity in the rat hippocampus. Neurosci. Lett 133: 287-290, 1991.
    • (1991) Neurosci. Lett , vol.133 , pp. 287-290
    • Moncada, C.1    Arvin, B.2    Le Peillet, E.3    Meldrum, B.S.4
  • 39
    • 0022650213 scopus 로고
    • Selective impairment of learning and blockade of long-term potentiation by an N-methyl-D-aspartate receptor antagonist, AP5
    • MORRIS, R. G. M., ANDERSON, E., LYNCH, G. S. AND BAUDRY, M.: Selective impairment of learning and blockade of long-term potentiation by an N-methyl-D-aspartate receptor antagonist, AP5. Nature 319: 774-776, 1986.
    • (1986) Nature , vol.319 , pp. 774-776
    • Morris, R.G.M.1    Anderson, E.2    Lynch, G.S.3    Baudry, M.4
  • 40
    • 0026505401 scopus 로고
    • Postischemic blockade of AMPA but not NMDA receptors mitigates neuronal damage in the rat brain following transient severe cerebral ischemia
    • NELLGȦRD, B. AND WIELOCH, T.: Postischemic blockade of AMPA but not NMDA receptors mitigates neuronal damage in the rat brain following transient severe cerebral ischemia. J. Cereb. Blood Flow Metab. 12: 2-11, 1992.
    • (1992) J. Cereb. Blood Flow Metab. , vol.12 , pp. 2-11
    • Nellgard, B.1    Wieloch, T.2
  • 41
    • 0028314957 scopus 로고
    • 6-(1H-Imidazol-1-yl)-7-nitro-2,3(1H, 4H)-quinoxalinedione hydrochloride (YM90K) and related compounds: Structure-activity relationships for the AMPA-type non-NMDA receptor
    • OHMORI, J., SAKAMOTO, S., KUBOTA, H., SHIMIZU-SASAMATA, M., OKADA, M., KAWASAKI, S., HIDAKA, K., TOGAMI, J., FURUYA, T. AND MURASE, K.: 6-(1H-Imidazol-1-yl)-7-nitro-2,3(1H, 4H)-quinoxalinedione hydrochloride (YM90K) and related compounds: Structure-activity relationships for the AMPA-type non-NMDA receptor. J. Med. Chem. 37: 467-475, 1994
    • (1994) J. Med. Chem. , vol.37 , pp. 467-475
    • Ohmori, J.1    Sakamoto, S.2    Kubota, H.3    Shimizu-Sasamata, M.4    Okada, M.5    Kawasaki, S.6    Hidaka, K.7    Togami, J.8    Furuya, T.9    Murase, K.10
  • 42
    • 1842339166 scopus 로고
    • α-Amino-3-hydroxy-5-methylisoxazole-4-propionate (AMPA) excitatory amino acid receptor antagonistic properties of YM900 (6-(1-imidazolyl)-7-nitroquinoxaline-2,3-(1H, 4H)-dione)
    • OKADA, M., HIDAKA, K., TOGAMI, J., OHNO, K., TADA, S., OHMORI, J., SAKAMOTO, S. AND YAMAGUCHI, T.: α-Amino-3-hydroxy-5-methylisoxazole-4-propionate (AMPA) excitatory amino acid receptor antagonistic properties of YM900 (6-(1-imidazolyl)-7-nitroquinoxaline-2,3-(1H, 4H)-dione). Soc. Neurosci. Abst. 18: 87, 1992.
    • (1992) Soc. Neurosci. Abst. , vol.18 , pp. 87
    • Okada, M.1    Hidaka, K.2    Togami, J.3    Ohno, K.4    Tada, S.5    Ohmori, J.6    Sakamoto, S.7    Yamaguchi, T.8
  • 43
    • 0024338054 scopus 로고
    • Pathological changes induced in cerebrocortical neurons by phencyclidine and related drugs
    • OLNEY, J. W., LABRUYERE, J. AND PRICE, M. T.: Pathological changes induced in cerebrocortical neurons by phencyclidine and related drugs. Science 244: 1360-1362, 1989.
    • (1989) Science , vol.244 , pp. 1360-1362
    • Olney, J.W.1    Labruyere, J.2    Price, M.T.3
  • 44
    • 0026633793 scopus 로고
    • NBQX does not affect learning and memory tasks in mice: A comparison with D-CPPene and ifenprodil
    • PARADA, J., CZUCZWAR, S. J. AND TURSKI, W. A.: NBQX does not affect learning and memory tasks in mice: A comparison with D-CPPene and ifenprodil. Cognitive Brain Res. 1: 67-71, 1992.
    • (1992) Cognitive Brain Res. , vol.1 , pp. 67-71
    • Parada, J.1    Czuczwar, S.J.2    Turski, W.A.3
  • 45
    • 4244030354 scopus 로고
    • The dose-dependency of the antiischemic efficacy and of the side effects of a novel NMDA antagonist, CNS 1102
    • PARK, C. K., MCBURNEY, R. N., HOLT, W. F., COTTER, R. E., MCCULLOCH, J., KANG, J. K. AND CHOI, C. R.: The dose-dependency of the antiischemic efficacy and of the side effects of a novel NMDA antagonist, CNS 1102 J Cereb Blood Flow Metab. 13(suppl. 1): S641, 1993.
    • (1993) J Cereb Blood Flow Metab. , vol.13 , Issue.1 SUPPL.
    • Park, C.K.1    Mcburney, R.N.2    Holt, W.F.3    Cotter, R.E.4    Mcculloch, J.5    Kang, J.K.6    Choi, C.R.7
  • 46
    • 0023788688 scopus 로고
    • The glutamate antagonist MK-801 reduces focal ischemic brain damage in the rat
    • PARK, C. K., NEHLS, D. G., GRAHAM, D. I., TEASDALE, G. M. AND MCCULLOCH, J.: The glutamate antagonist MK-801 reduces focal ischemic brain damage in the rat. Ann. Neurol. 24: 543-551, 1988
    • (1988) Ann. Neurol. , vol.24 , pp. 543-551
    • Park, C.K.1    Nehls, D.G.2    Graham, D.I.3    Teasdale, G.M.4    Mcculloch, J.5
  • 48
    • 0026501717 scopus 로고
    • Pathophysiology of acute ischemic stroke
    • PULSINELLI, W. Pathophysiology of acute ischemic stroke. Lancet 339: 533-536, 1992.
    • (1992) Lancet , vol.339 , pp. 533-536
    • Pulsinelli, W.1
  • 49
    • 0026532928 scopus 로고
    • Quinoxaline derivatives: Structure-activity relationships and physiological implications of inhibition of N-methyl-D-aspartate and non-N-Methyl-D-aspartate receptor-mediated currents and synaptic potentials
    • RANDLE, J. C. R., GUET, T., BOBICHON, C., MOREAU, C., CURUTCHET, P., LAMBOLEZ, B., CARVALHO, L. P. D., CORDI, A., LEPAGNOL, J. M.: Quinoxaline derivatives: Structure-activity relationships and physiological implications of inhibition of N-methyl-D-aspartate and non-N-Methyl-D-aspartate receptor-mediated currents and synaptic potentials. Mol. Pharmacol. 41: 337-345, 1992.
    • (1992) Mol. Pharmacol. , vol.41 , pp. 337-345
    • Randle, J.C.R.1    Guet, T.2    Bobichon, C.3    Moreau, C.4    Curutchet, P.5    Lambolez, B.6    Carvalho, L.P.D.7    Cordi, A.8    Lepagnol, J.M.9
  • 50
    • 0026080080 scopus 로고
    • Ontogeny of the benzodiazepine receptor in human brain: Fluorographic, immunochemical and reversible binding studies
    • REICHELT, R , HOFMANN, D., FODISH, H. J., MOHLER, H., KNAPP, M. AND HEBEBRAND, J.: Ontogeny of the benzodiazepine receptor in human brain: Fluorographic, immunochemical and reversible binding studies. J. Neurochem. 57: 1128-1135, 1991.
    • (1991) J. Neurochem. , vol.57 , pp. 1128-1135
    • Reichelt, R.1    Hofmann, D.2    Fodish, H.J.3    Mohler, H.4    Knapp, M.5    Hebebrand, J.6
  • 52
    • 0025117827 scopus 로고
    • 2,3-Dihydroxy-6-nitro-7-sulfamoyl-benzo(F)quinoxaline: A neuroprotectant for cerebral ischemia
    • SHEARDOWN, M. J., NIELSEN, E.Ø., HANSEN, A. J., JACOBSEN, P. AND HONORE, T.: 2,3-Dihydroxy-6-nitro-7-sulfamoyl-benzo(F)quinoxaline: A neuroprotectant for cerebral ischemia. Science 247: 571-574, 1990.
    • (1990) Science , vol.247 , pp. 571-574
    • Sheardown, M.J.1    Nielsen, E.Ø.2    Hansen, A.J.3    Jacobsen, P.4    Honore, T.5
  • 53
    • 0027336469 scopus 로고
    • AMPA, but not NMDA, receptor antagonism is neuroprotective in gerbil global ischaemia, even when delayed 24 h
    • SHEARDOWN, M. J., SUZDAK, P. D. AND NORDHOLM, L.: AMPA, but not NMDA, receptor antagonism is neuroprotective in gerbil global ischaemia, even when delayed 24 h. Eur. J. Pharmacol. 236: 347-353, 1993.
    • (1993) Eur. J. Pharmacol. , vol.236 , pp. 347-353
    • Sheardown, M.J.1    Suzdak, P.D.2    Nordholm, L.3
  • 54
    • 1842370130 scopus 로고
    • The neuroprotective actions of YM900, a novel and potent α-amino-3-hydroxy-5-methylisoxazole-4-propionate (AMPA) receptor antagonist, in a gerbil global ischemia model and a rat focal ischemia model
    • SHIMIZU-SASAMATA, M., KAWASAKI, S., YATSUGI, S., OHMORI, J., SAKAMOTO, S., KOSHIYA, K., USUDA, S. AND MURASE, K.: The neuroprotective actions of YM900, a novel and potent α-amino-3-hydroxy-5-methylisoxazole-4-propionate (AMPA) receptor antagonist, in a gerbil global ischemia model and a rat focal ischemia model. Soc. Neurosci. Abst. 18: 87, 1992.
    • (1992) Soc. Neurosci. Abst. , vol.18 , pp. 87
    • Shimizu-Sasamata, M.1    Kawasaki, S.2    Yatsugi, S.3    Ohmori, J.4    Sakamoto, S.5    Koshiya, K.6    Usuda, S.7    Murase, K.8
  • 56
    • 1842289029 scopus 로고
    • The discovery of YM900 and its pharmacological characterization as a selective and potent α-amino-3-hydroxy-5-methylisoxazole-4-propionate (AMPA) receptor antagonist
    • SHIMIZU-SASAMATA, M., OKADA, M., SAKAMOTO, S , KAWASAKI, S., KOSHIYA, K., USUDA, S. AND MURASE, K.: The discovery of YM900 and its pharmacological characterization as a selective and potent α-amino-3-hydroxy-5-methylisoxazole-4-propionate (AMPA) receptor antagonist. Jpn. J. Pharmacol. 60(suppl. 1): 164, 1993b.
    • (1993) Jpn. J. Pharmacol. , vol.60 , Issue.1 SUPPL. , pp. 164
    • Shimizu-Sasamata, M.1    Okada, M.2    Sakamoto, S.3    Kawasaki, S.4    Koshiya, K.5    Usuda, S.6    Murase, K.7
  • 57
    • 0024556434 scopus 로고
    • Calcium fluxes, calcium antagonists, and calcium related pathology in brain ischemia, hypoglycemia, and spreading depression: A unifying hypothesis
    • SIESJO, B. K. AND BENGTSSON, F.: Calcium fluxes, calcium antagonists, and calcium related pathology in brain ischemia, hypoglycemia, and spreading depression: A unifying hypothesis. J. Cereb. Blood Flow Metab. 9: 127-140, 1989.
    • (1989) J. Cereb. Blood Flow Metab. , vol.9 , pp. 127-140
    • Siesjo, B.K.1    Bengtsson, F.2
  • 58
    • 0026623418 scopus 로고
    • Cerebroprotective effect of a non-N-methyl-D-aspartate antagonist, GYKI 52466, after focal ischemia in the rat
    • SMITH, S. E. AND MELDRUM, B. S.: Cerebroprotective effect of a non-N-methyl-D-aspartate antagonist, GYKI 52466, after focal ischemia in the rat. Stroke 23: 861-864, 1992.
    • (1992) Stroke , vol.23 , pp. 861-864
    • Smith, S.E.1    Meldrum, B.S.2
  • 59
    • 0019868418 scopus 로고
    • Focal cerebral ischemia in the rat: Description of technique and early neuropathological consequences following middle cerebral artery occlusion
    • TAMUSA, A., GRAHAM, D. I., MCCULLOCH, J. AND TEASDALE, G. M.: Focal cerebral ischemia in the rat: Description of technique and early neuropathological consequences following middle cerebral artery occlusion. J. Cereb. Blood Flow Metab. 1: 53-60, 1981.
    • (1981) J. Cereb. Blood Flow Metab. , vol.1 , pp. 53-60
    • Tamusa, A.1    Graham, D.I.2    Mcculloch, J.3    Teasdale, G.M.4
  • 60
    • 0025999656 scopus 로고
    • Selective increase of AMPA binding to the AMPA/quisqualate receptor in the hippocampus in response to acute stress
    • TOCCO, G., SHORS, T. J., BAUDRY, M. AND THOMPSON, R. F.: Selective increase of AMPA binding to the AMPA/quisqualate receptor in the hippocampus in response to acute stress. Brain Res. 559: 168-171, 1991.
    • (1991) Brain Res. , vol.559 , pp. 168-171
    • Tocco, G.1    Shors, T.J.2    Baudry, M.3    Thompson, R.F.4
  • 61
    • 0025024016 scopus 로고
    • Cortical neurons containing somatostatin- or parvalbumin-like immunoreactivity are atypically vulnerable to excitotoxic injury in vitro
    • WEISS, J. H., KOH, J-Y., BAIMBRIDGE, K. G. AND CHOI, D. W.: Cortical neurons containing somatostatin- or parvalbumin-like immunoreactivity are atypically vulnerable to excitotoxic injury in vitro. Neurology 40: 1288-1292, 1990.
    • (1990) Neurology , vol.40 , pp. 1288-1292
    • Weiss, J.H.1    Koh, J.-Y.2    Baimbridge, K.G.3    Choi, D.W.4
  • 62
    • 0026542967 scopus 로고
    • NBQX, an AMPA antagonist, reduces glutamate-mediated brain edema
    • WESTERGREN, I. AND JOHANSSON, B. B.: NBQX, an AMPA antagonist, reduces glutamate-mediated brain edema. Brain Res. 573: 324-326, 1992.
    • (1992) Brain Res. , vol.573 , pp. 324-326
    • Westergren, I.1    Johansson, B.B.2
  • 64
    • 0000708928 scopus 로고
    • Effects of a novel AMPA antagonist YM900 and other excitatory amino acid antagonists on the delayed neuronal death in the gerbil hippocampus
    • YATSUGI, S., KAWASAKI, S., KATOH, M., TAKABASHI, M., KOSHIYA, K. AND SHIMIZU-SASAMATA, M.: Effects of a novel AMPA antagonist YM900 and other excitatory amino acid antagonists on the delayed neuronal death in the gerbil hippocampus. J. Cereb. Blood Flow Metab. 13 (suppl. 1): S635, 1993.
    • (1993) J. Cereb. Blood Flow Metab. , vol.13 , Issue.1 SUPPL.
    • Yatsugi, S.1    Kawasaki, S.2    Katoh, M.3    Takabashi, M.4    Koshiya, K.5    Shimizu-Sasamata, M.6
  • 65
    • 0027464959 scopus 로고
    • A benzodiazepine recognition site associated with the non-NMDA glutamate receptor
    • ZORUMSKI, C. F., YAMADA, K. A., PRICE, M. T. AND OLNEY, J. W.: A benzodiazepine recognition site associated with the non-NMDA glutamate receptor. Neuron 10: 61-67, 1993.
    • (1993) Neuron , vol.10 , pp. 61-67
    • Zorumski, C.F.1    Yamada, K.A.2    Price, M.T.3    Olney, J.W.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.