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Volumn 109, Issue 4, 1996, Pages 957-962

Partial vs Full ß-Receptor Agonism: A Clinical Study of Inhaled Albuterol and Fenoterol

Author keywords

Cardiovascular effects; Intrinsic activity; agonist

Indexed keywords

BETA ADRENERGIC RECEPTOR STIMULATING AGENT; CYCLIC AMP; FENOTEROL; PARTIAL AGONIST; POTASSIUM ION; SALBUTAMOL;

EID: 0029924030     PISSN: 00123692     EISSN: None     Source Type: Journal    
DOI: 10.1378/chest.109.4.957     Document Type: Article
Times cited : (32)

References (41)
  • 1
    • 0027255641 scopus 로고
    • Beta-adrenergic agonist toxicity: Less of a problem, more of a perception
    • Ziment I. Beta-adrenergic agonist toxicity: less of a problem, more of a perception. Chest 1993; 103:1591-97
    • (1993) Chest , vol.103 , pp. 1591-1597
    • Ziment, I.1
  • 2
    • 0028142160 scopus 로고
    • Regular beta-adrenergic agonists: Evidence, not reassurance, is what is needed
    • Taylor DR, Sears MR. Regular beta-adrenergic agonists: evidence, not reassurance, is what is needed. Chest 1994; 106:552-59
    • (1994) Chest , vol.106 , pp. 552-559
    • Taylor, D.R.1    Sears, M.R.2
  • 3
    • 0024515162 scopus 로고
    • Prescribed fenoterol and death from asthma in New Zealand, 1981-83: Case control study
    • Crane J, Flatt A, Jackson R, et al. Prescribed fenoterol and death from asthma in New Zealand, 1981-83: case control study. Lancet 1989; 1:917-22
    • (1989) Lancet , vol.1 , pp. 917-922
    • Crane, J.1    Flatt, A.2    Jackson, R.3
  • 4
    • 0025797080 scopus 로고
    • Case control study of prescribed fenoterol and death from asthma in New Zealand, 1981-1987: A further case control study
    • Grainger J, Woodman K, Pearce NE, et al. Case control study of prescribed fenoterol and death from asthma in New Zealand, 1981-1987: a further case control study. Thorax 1991; 46:105-11
    • (1991) Thorax , vol.46 , pp. 105-111
    • Grainger, J.1    Woodman, K.2    Pearce, N.E.3
  • 5
    • 0025318713 scopus 로고
    • Case control study of prescribed fenoterol and death from asthma in New Zealand, 1977-1981
    • Pearce NE, Grainger J, Atkinson M, et al. Case control study of prescribed fenoterol and death from asthma in New Zealand, 1977-1981. Thorax 1990; 45:170-75
    • (1990) Thorax , vol.45 , pp. 170-175
    • Pearce, N.E.1    Grainger, J.2    Atkinson, M.3
  • 6
    • 0026595475 scopus 로고
    • The use of beta agonists and the risk of death and near death from asthma
    • Spitzer WO, Suissa S, Ernst P, et al. The use of beta agonists and the risk of death and near death from asthma. N Engl J Med 1992; 326:501-06
    • (1992) N Engl J Med , vol.326 , pp. 501-506
    • Spitzer, W.O.1    Suissa, S.2    Ernst, P.3
  • 7
    • 0000406736 scopus 로고
    • Use of beta agonists and mortality in patients with stable COPD
    • Criée C-P, Quast C-H, Lüdtke R, et al. Use of beta agonists and mortality in patients with stable COPD. Eur Respir J 1993; 6(suppl 17):426s
    • (1993) Eur Respir J , vol.6 , Issue.17 SUPPL.
    • Criée, C.-P.1    Quast, C.-H.2    Lüdtke, R.3
  • 8
    • 0025902196 scopus 로고
    • Beta agonists and asthma mortality: Déjà-vu
    • Pearce N, Crane J, Burgess C, et al. Beta agonists and asthma mortality: déjà-vu. Clin Exp Allergy 1991; 21:401-10
    • (1991) Clin Exp Allergy , vol.21 , pp. 401-410
    • Pearce, N.1    Crane, J.2    Burgess, C.3
  • 9
    • 0026241776 scopus 로고
    • Asthma mortality and inhaled beta agonist therapy
    • Beasley R, Pearce N, Crane J, et al. Asthma mortality and inhaled beta agonist therapy. Aust NZ J Med 1991; 21:753-63
    • (1991) Aust NZ J Med , vol.21 , pp. 753-763
    • Beasley, R.1    Pearce, N.2    Crane, J.3
  • 10
    • 0027313429 scopus 로고
    • The β-agonist controversy: A perspective
    • Crane J, Burgess C, Pearce N, et al. The β-agonist controversy: a perspective. Eur Respir Rev 1993; 3:475-82
    • (1993) Eur Respir Rev , vol.3 , pp. 475-482
    • Crane, J.1    Burgess, C.2    Pearce, N.3
  • 11
    • 0025223381 scopus 로고
    • Regular inhaled beta-agonist treatment in bronchial asthma
    • Sears MR, Taylor DR, Print CG, et al. Regular inhaled beta-agonist treatment in bronchial asthma. Lancet 1990; 336:1391-96
    • (1990) Lancet , vol.336 , pp. 1391-1396
    • Sears, M.R.1    Taylor, D.R.2    Print, C.G.3
  • 12
    • 0015348479 scopus 로고
    • Asthma mortality: Why the United States was spared an epidemic of deaths due to asthma
    • Stolley PD. Asthma mortality: why the United States was spared an epidemic of deaths due to asthma. Am Rev Respir Dis 1972; 105:883-90
    • (1972) Am Rev Respir Dis , vol.105 , pp. 883-890
    • Stolley, P.D.1
  • 13
    • 0018246383 scopus 로고
    • Association between asthma mortality and isoproterenol aerosols: A review
    • Stolley PD, Schinnar R. Association between asthma mortality and isoproterenol aerosols: a review. Prev Med 1978; 7:519-38
    • (1978) Prev Med , vol.7 , pp. 519-538
    • Stolley, P.D.1    Schinnar, R.2
  • 14
    • 0642325775 scopus 로고
    • Sympathomimetic bronchodilating drugs
    • Widdicombe J, ed. Oxford, NY: Oxford Pergamon Press
    • Brittain RT, Dean CM, Jack D. Sympathomimetic bronchodilating drugs. In: Widdicombe J, ed. Respiratory pharmacology. Oxford, NY: Oxford Pergamon Press, 1991; 613-52
    • (1991) Respiratory Pharmacology , pp. 613-652
    • Brittain, R.T.1    Dean, C.M.2    Jack, D.3
  • 15
    • 0015391826 scopus 로고
    • An examination of some β-adrenoceptor stimulants for selectivity using the isolated trachea and atria of the guinea-pig
    • O'Donnell SR. An examination of some β-adrenoceptor stimulants for selectivity using the isolated trachea and atria of the guinea-pig. Eur J Pharmacol 1972; 19:371-79
    • (1972) Eur J Pharmacol , vol.19 , pp. 371-379
    • O'Donnell, S.R.1
  • 16
    • 34447558006 scopus 로고
    • Mechanisms of drug action
    • Edinburgh: Churchill Livingstone
    • Rang HP, Dale MM. Mechanisms of drug action. In: Pharmacology. Edinburgh: Churchill Livingstone, 1987; 33
    • (1987) Pharmacology , pp. 33
    • Rang, H.P.1    Dale, M.M.2
  • 17
    • 0016189843 scopus 로고
    • Non-catechol phenylethanolamines: Agonistic actions on β-adrenoceptors in isolated tissues from the guinea-pig
    • Malta E, Raper C. Non-catechol phenylethanolamines: agonistic actions on β-adrenoceptors in isolated tissues from the guinea-pig. Clin Exp Pharmacol Physiol 1974; 1:259-68
    • (1974) Clin Exp Pharmacol Physiol , vol.1 , pp. 259-268
    • Malta, E.1    Raper, C.2
  • 18
    • 0015797496 scopus 로고
    • Salbutamol: Agonistic and antagonistic activity at β-adrenoceptor sites
    • Raper C, Malta E. Salbutamol: agonistic and antagonistic activity at β-adrenoceptor sites. J Pharm Pharmacol 1973; 25:661-63
    • (1973) J Pharm Pharmacol , vol.25 , pp. 661-663
    • Raper, C.1    Malta, E.2
  • 19
    • 0019165681 scopus 로고
    • β-adrenoceptors in human lung, bronchus and lymphocytes
    • Davis C, Conolly ME, Greenacre JK. β-adrenoceptors in human lung, bronchus and lymphocytes. Br J Clin Pharmacol 1980; 10:425-32
    • (1980) Br J Clin Pharmacol , vol.10 , pp. 425-432
    • Davis, C.1    Conolly, M.E.2    Greenacre, J.K.3
  • 20
    • 0025119788 scopus 로고
    • Guidelines for the management of asthma in adults
    • British Thoracic Society. Guidelines for the management of asthma in adults. BMJ 1990; 301:797-800
    • (1990) BMJ , vol.301 , pp. 797-800
  • 21
    • 0017666391 scopus 로고
    • A critical review of the systolic time intervals
    • Lewis RP, Rittgers SE, Forester WF, et al. A critical review of the systolic time intervals. Circulation 1977; 56:146-58
    • (1977) Circulation , vol.56 , pp. 146-158
    • Lewis, R.P.1    Rittgers, S.E.2    Forester, W.F.3
  • 22
    • 0024062758 scopus 로고
    • Correction of systolic time intervals for heart rate: A comparison of individual with population derived regression equations
    • Warrington SJ, Weerasuriya K, Burgess CD. Correction of systolic time intervals for heart rate: a comparison of individual with population derived regression equations. Br J Clin Pharmacol 1988; 26:155-65
    • (1988) Br J Clin Pharmacol , vol.26 , pp. 155-165
    • Warrington, S.J.1    Weerasuriya, K.2    Burgess, C.D.3
  • 23
    • 0642264538 scopus 로고
    • Evaluation of the Ionetics electrolyte analyser for plasma potassium measurement in whole blood
    • Siebers RWL, Bremner P, Woodman K, et al. Evaluation of the Ionetics electrolyte analyser for plasma potassium measurement in whole blood. NZ J Med Lab Technol 1990; 44:85-6
    • (1990) NZ J Med Lab Technol , vol.44 , pp. 85-86
    • Siebers, R.W.L.1    Bremner, P.2    Woodman, K.3
  • 24
    • 0023585102 scopus 로고
    • Hypokalaemia and other nonbronchial effects of inhaled fenoterol and salbutamol: A placebo-controlled dose-response study in healthy volunteers
    • Scheinin M, Koulu M, Laurikainen E, et al. Hypokalaemia and other nonbronchial effects of inhaled fenoterol and salbutamol: a placebo-controlled dose-response study in healthy volunteers. Br J Clin Pharmacol 1987; 24:645-53
    • (1987) Br J Clin Pharmacol , vol.24 , pp. 645-653
    • Scheinin, M.1    Koulu, M.2    Laurikainen, E.3
  • 25
    • 0022978869 scopus 로고
    • In vitro responsiveness of human asthmatic bronchus to carbachol, histamine, β-adrenoceptor agonists and theophvlline
    • Goldie RG, Spina D, Henry PJ, et al. In vitro responsiveness of human asthmatic bronchus to carbachol, histamine, β-adrenoceptor agonists and theophvlline. Br J Clin Pharmacol 1986; 22:669-76
    • (1986) Br J Clin Pharmacol , vol.22 , pp. 669-676
    • Goldie, R.G.1    Spina, D.2    Henry, P.J.3
  • 26
    • 0017885580 scopus 로고
    • Evidence that the efficacy (intrinsic activity) of fenoterol is higher than that of salbutamol on β-adrenoceptors in guinea-pig trachea
    • O'Donnell SR, Wanstall JC. Evidence that the efficacy (intrinsic activity) of fenoterol is higher than that of salbutamol on β-adrenoceptors in guinea-pig trachea. Eur J Clin Pharmacol 1978; 47:333-40
    • (1978) Eur J Clin Pharmacol , vol.47 , pp. 333-340
    • O'Donnell, S.R.1    Wanstall, J.C.2
  • 27
    • 0025237868 scopus 로고
    • On the physiological role of beta-2 adrenoceptors in the human heart: In vitro and in vivo studies
    • Motomura S, Zerkowski HR, Daul A, et al. On the physiological role of beta-2 adrenoceptors in the human heart: in vitro and in vivo studies. Am Heart J 1990; 119:608-19
    • (1990) Am Heart J , vol.119 , pp. 608-619
    • Motomura, S.1    Zerkowski, H.R.2    Daul, A.3
  • 28
    • 0021929608 scopus 로고
    • Effects of the beta-2 adrenoceptor agonists fenoterol and salbutamol on force of confraction in isolated human ventricular myocardium
    • Mugge A, Posselt D, Reimer U, et al. Effects of the beta-2 adrenoceptor agonists fenoterol and salbutamol on force of confraction in isolated human ventricular myocardium. Klin Wochenschr 1985; 63:26-31
    • (1985) Klin Wochenschr , vol.63 , pp. 26-31
    • Mugge, A.1    Posselt, D.2    Reimer, U.3
  • 29
    • 0023808883 scopus 로고
    • The functional importance of beta-1 and beta-2 adrenoceptors in the human heart
    • Brodde OE. The functional importance of beta-1 and beta-2 adrenoceptors in the human heart. Am J Cardiol 1988; 62:24C-9C
    • (1988) Am J Cardiol , vol.62
    • Brodde, O.E.1
  • 30
    • 0022547778 scopus 로고
    • The role of cardiac beta-1 receptors in the haemodynamic response to a beta-2 agonist
    • Strauss MH, Reeves RA, Smith DL, et al. The role of cardiac beta-1 receptors in the haemodynamic response to a beta-2 agonist. Clin Pharmacol Ther 1986; 40:108-15
    • (1986) Clin Pharmacol Ther , vol.40 , pp. 108-115
    • Strauss, M.H.1    Reeves, R.A.2    Smith, D.L.3
  • 31
    • 0018908946 scopus 로고
    • Beta-1 and beta-2 adrenergic receptors responsible for cyclic AMP accumulation in isolated heart and lung cells
    • Hazeki O, Ui M. Beta-1 and beta-2 adrenergic receptors responsible for cyclic AMP accumulation in isolated heart and lung cells. Mol Pharmacol 1980; 17:8-13
    • (1980) Mol Pharmacol , vol.17 , pp. 8-13
    • Hazeki, O.1    Ui, M.2
  • 32
    • 0025851462 scopus 로고
    • 2 -adrenoceptors in the human heart: Properties, function and alternations in chronic heart failure
    • 2 -adrenoceptors in the human heart: properties, function and alternations in chronic heart failure. Pharmacol Rev 1991; 43:204-42
    • (1991) Pharmacol Rev , vol.43 , pp. 204-242
    • Brodde, O.E.1
  • 33
  • 34
    • 0016224315 scopus 로고
    • Further observations on the cardiotoxicity of isoprenaline during hypoxia
    • McDevitt DG, Shanks RG, Swanton JG. Further observations on the cardiotoxicity of isoprenaline during hypoxia. Br J Pharmacol 1974; 50:335-44
    • (1974) Br J Pharmacol , vol.50 , pp. 335-344
    • McDevitt, D.G.1    Shanks, R.G.2    Swanton, J.G.3
  • 35
    • 0028130173 scopus 로고
    • The myoardial effects of fenoterol, isoprenaline and salbutamol in normoxic and hypoxic sheep
    • Pack RJ, Alley MR, Dallimore JA, et al. The myoardial effects of fenoterol, isoprenaline and salbutamol in normoxic and hypoxic sheep. Int J Exp Pathol 1994; 75:357-62
    • (1994) Int J Exp Pathol , vol.75 , pp. 357-362
    • Pack, R.J.1    Alley, M.R.2    Dallimore, J.A.3
  • 37
    • 0025816779 scopus 로고
    • Respiratory arrest in fatal asthma
    • Beasley R, Burgess C, Crane J, et al. Respiratory arrest in fatal asthma. N Engl J Med 1991; 325:205-06
    • (1991) N Engl J Med , vol.325 , pp. 205-206
    • Beasley, R.1    Burgess, C.2    Crane, J.3
  • 38
    • 0026479923 scopus 로고
    • The cardiovascular effects of fenoterol under conditions of hypoxaemia
    • Bremner P, Burgess C, Crane J, et al. The cardiovascular effects of fenoterol under conditions of hypoxaemia. Thorax 1992; 47:814-17
    • (1992) Thorax , vol.47 , pp. 814-817
    • Bremner, P.1    Burgess, C.2    Crane, J.3
  • 39
    • 0017819204 scopus 로고
    • Fenoterol: A review of its pharmacological properties and therapeutic efficacy in asthma
    • Heel RC, Brogden TM, Avery GS. Fenoterol: a review of its pharmacological properties and therapeutic efficacy in asthma. Drugs 1978; 15:3-32
    • (1978) Drugs , vol.15 , pp. 3-32
    • Heel, R.C.1    Brogden, T.M.2    Avery, G.S.3
  • 40
    • 0028888460 scopus 로고
    • Comparison of the relative airways and systemic potencies of inhaled fenoterol and salbutamol in asthmatic patients
    • Lipworth BJ, Newnham DM, Clark RA, et al. Comparison of the relative airways and systemic potencies of inhaled fenoterol and salbutamol in asthmatic patients. Thorax 1995; 50:54-61
    • (1995) Thorax , vol.50 , pp. 54-61
    • Lipworth, B.J.1    Newnham, D.M.2    Clark, R.A.3
  • 41
    • 0025159925 scopus 로고
    • The self-administration of inhaled beta agonist drugs during severe asthma
    • Windom HH, Burgess CD, Crane J, et al. The self-administration of inhaled beta agonist drugs during severe asthma. NZ Med J 1990; 103:205-07
    • (1990) NZ Med J , vol.103 , pp. 205-207
    • Windom, H.H.1    Burgess, C.D.2    Crane, J.3


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