메뉴 건너뛰기




Volumn 117, Issue 6, 1996, Pages 1171-1180

Evidence for human thromboxane receptor heterogeneity using a novel series of 9,11-cyclic carbonate derivatives of prostaglandin F2α

Author keywords

AGN191976; AGN192093; Human platelets; Human uterus; Prostanoid receptors; Rat aorta; Smooth muscle; TP receptor heterogeneity; TxA2 mimetics; U 46619

Indexed keywords

15 HYDROXY 11ALPHA,9ALPHA EPOXYMETHANOPROSTA 5,13 DIENOIC ACID; 7 [3 [(4 PHENYLSEMICARBAZIDO)METHYL] 7 OXABICYCLO[2.2.1]HEPT 2 YL] 5 HEPTENOIC ACID; 7 [7 (3 HYDROXY 1 OCTENYL) 3 OXO 2,4 DIOXABICYCLO[3.2.1]OCT 6 YL] 5 HEPTENOIC ACID; 7 [7 (3 HYDROXY 1 OCTENYL) 3 OXO 2,4 DIOXABICYCLO[3.2.1]OCT 6 YL] 5 HEPTENOL; ADENOSINE DIPHOSPHATE; ARACHIDONIC ACID; PROSTAGLANDIN F2 ALPHA DERIVATIVE; PROSTANOID RECEPTOR; RECEPTOR SUBTYPE; THROMBOXANE RECEPTOR; UNCLASSIFIED DRUG;

EID: 0029918957     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1476-5381.1996.tb16712.x     Document Type: Article
Times cited : (22)

References (42)
  • 4
    • 0016681589 scopus 로고
    • The synthesis of prostaglandin endoperoxide analogs
    • BUNDY, G.L. (1975). The synthesis of prostaglandin endoperoxide analogs. Tetrahedron Lett., 24, 1957-1960.
    • (1975) Tetrahedron Lett. , vol.24 , pp. 1957-1960
    • Bundy, G.L.1
  • 5
    • 0028023008 scopus 로고
    • Synthesis of a novel series of 3-oxo-2,4-dioxobicyclo[3.2.1]octanes: Additional evidence for two thromboxane receptor subtypes
    • BURK, R.M., GAC, T.S., GARST, M.E., GIBSON, L.L., KRAUSS, A.H., PROTZMAN, C.E. & WOODWARD, D.F. (1994). Synthesis of a novel series of 3-oxo-2,4-dioxobicyclo[3.2.1]octanes: additional evidence for two thromboxane receptor subtypes. Bioorg. Med. Chem. Lett., 4, 2103-2106.
    • (1994) Bioorg. Med. Chem. Lett. , vol.4 , pp. 2103-2106
    • Burk, R.M.1    Gac, T.S.2    Garst, M.E.3    Gibson, L.L.4    Krauss, A.H.5    Protzman, C.E.6    Woodward, D.F.7
  • 8
    • 0024592289 scopus 로고
    • Prostanoid-induced contraction of human bronchial smooth muscle is mediated by TP-receptors
    • COLEMAN, R.A. & SHELDRICK, R.L.G. (1989). Prostanoid-induced contraction of human bronchial smooth muscle is mediated by TP-receptors. Br. J. Pharmacol., 96, 688-692.
    • (1989) Br. J. Pharmacol. , vol.96 , pp. 688-692
    • Coleman, R.A.1    Sheldrick, R.L.G.2
  • 9
    • 0028930443 scopus 로고
    • Chromosomal localization of the human prostanoid receptor gene family
    • DUNCAN, A.M.V., ANDERSON, L.L., FUNK, C.D., ABRAMOVITZ, M. & ADAM, M. (1995). Chromosomal localization of the human prostanoid receptor gene family. Genomics, 25, 740-742.
    • (1995) Genomics , vol.25 , pp. 740-742
    • Duncan, A.M.V.1    Anderson, L.L.2    Funk, C.D.3    Abramovitz, M.4    Adam, M.5
  • 10
    • 0025923520 scopus 로고
    • 2 receptors: Distinct subtypes mediate vascular smooth muscle contraction and platelet aggregation
    • 2 receptors: distinct subtypes mediate vascular smooth muscle contraction and platelet aggregation. J. Pharmacol. Exp. Ther., 258, 74-81.
    • (1991) J. Pharmacol. Exp. Ther. , vol.258 , pp. 74-81
    • Furci, L.1    Fitzgerald, D.J.2    Fitzgerald, G.A.3
  • 13
    • 0019969438 scopus 로고
    • Antagonism of the thromboxane-sensitive systems of the rabbit aorta, dog saphenous vein and guinea-pig trachea
    • JONES, R.L., PEESAPATI, V. & WILSON, N.H. (1982). Antagonism of the thromboxane-sensitive systems of the rabbit aorta, dog saphenous vein and guinea-pig trachea. Br. J. Pharmacol., 76, 423-438.
    • (1982) Br. J. Pharmacol. , vol.76 , pp. 423-438
    • Jones, R.L.1    Peesapati, V.2    Wilson, N.H.3
  • 14
    • 0024604978 scopus 로고
    • 2-mimetic, the actions of which are slowly reversed by receptor blockade
    • 2-mimetic, the actions of which are slowly reversed by receptor blockade. Br. J. Pharmacol., 96, 875-887.
    • (1989) Br. J. Pharmacol. , vol.96 , pp. 875-887
    • Jones, R.L.1    Wilson, N.H.2    Lawrence, R.A.3
  • 16
    • 0020398514 scopus 로고
    • Studies on the characterisation of prostanoid receptors: A proposed classification
    • KENNEDY, I., COLEMAN, RA., HUMPHREY, P.P.A., LEVY, G.P. & LUMLEY, P. (1982). Studies on the characterisation of prostanoid receptors: a proposed classification. Prostaglandins, 24, 667-689.
    • (1982) Prostaglandins , vol.24 , pp. 667-689
    • Kennedy, I.1    Coleman, R.A.2    Humphrey, P.P.A.3    Levy, G.P.4    Lumley, P.5
  • 20
    • 0024348514 scopus 로고
    • 2 receptor blocking drug on platelets and vascular and airways smooth muscle in vitro
    • 2 receptor blocking drug on platelets and vascular and airways smooth muscle in vitro. Br. J. Pharmacol., 97, 783-794.
    • (1989) Br. J. Pharmacol. , vol.97 , pp. 783-794
    • Lumley, P.1    White, B.P.2    Humphrey, P.P.A.3
  • 24
    • 0023740545 scopus 로고
    • Characterisation of receptors mediating the contractile effects of prostanoids in guinea-pig and human airways
    • MCKENNIFF, M., RODGER, I.W., NORMAN, P. & GARDINER, P.J. (1988). Characterisation of receptors mediating the contractile effects of prostanoids in guinea-pig and human airways. Eur. J. Pharmacol., 153, 149-159.
    • (1988) Eur. J. Pharmacol. , vol.153 , pp. 149-159
    • Mckenniff, M.1    Rodger, I.W.2    Norman, P.3    Gardiner, P.J.4
  • 25
    • 0026617018 scopus 로고
    • 2α, a potent agonist of the vascular thromboxane/endoperoxide receptor, is a platelet thromboxane/endoperoxide receptor antagonist
    • 2α, a potent agonist of the vascular thromboxane/endoperoxide receptor, is a platelet thromboxane/endoperoxide receptor antagonist. Prostaglandins, 44, 155-163.
    • (1992) Prostaglandins , vol.44 , pp. 155-163
    • Morrow, J.D.1    Minton, T.A.2    Roberts III, L.J.3
  • 27
    • 0022612678 scopus 로고
    • Binding of radioiodinated 13-azapinane thromboxane antagonist to platelets: Correlation with antiaggregatory activity in different species
    • NARUMIYA, S., OKUMA, M. & USHIKUBI, F. (1986). Binding of radioiodinated 13-azapinane thromboxane antagonist to platelets: correlation with antiaggregatory activity in different species. Br. J. Pharmacol., 88, 323-331.
    • (1986) Br. J. Pharmacol. , vol.88 , pp. 323-331
    • Narumiya, S.1    Okuma, M.2    Ushikubi, F.3
  • 29
    • 0025938084 scopus 로고
    • Inhibitory effects of BAY u3405 on prostanoid-induced contractions in human isolated bronchial and pulmonary arterial muscle preparations
    • NOREL, X., LABAT, C., GARDINER, P.J. & BRINK, C. (1991). Inhibitory effects of BAY u3405 on prostanoid-induced contractions in human isolated bronchial and pulmonary arterial muscle preparations. Br. J. Pharmacol., 104, 591-595.
    • (1991) Br. J. Pharmacol. , vol.104 , pp. 591-595
    • Norel, X.1    Labat, C.2    Gardiner, P.J.3    Brink, C.4
  • 34
    • 0026071419 scopus 로고
    • In vitro characterization of prostanoid EP-receptors in the non-pregnant human myometrium
    • SENIOR, J., MARSHALL, K., BAXTER, G.S. SANGHA, R. & CLAYTON, J.K. (1991). In vitro characterization of prostanoid EP-receptors in the non-pregnant human myometrium. Br. J. Pharmacol., 102, 747-753.
    • (1991) Br. J. Pharmacol. , vol.102 , pp. 747-753
    • Senior, J.1    Marshall, K.2    Baxter, G.S.3    Sangha, R.4    Clayton, J.K.5
  • 35
    • 0026698153 scopus 로고
    • In vitro characterization of prostanoid FP-, DP-, IP- and TP-receptors on the non-pregnant human myometrium
    • SENIOR, J., SANGHA, R., BAXTER, G.S., MARSHALL, K. & CLAYTON, J.K. (1992). In vitro characterization of prostanoid FP-, DP-, IP- and TP-receptors on the non-pregnant human myometrium. Br. J. Pharmacol. 107, 215-221.
    • (1992) Br. J. Pharmacol. , vol.107 , pp. 215-221
    • Senior, J.1    Sangha, R.2    Baxter, G.S.3    Marshall, K.4    Clayton, J.K.5
  • 37
    • 0025193358 scopus 로고
    • 2 analogues in human platelets. Discrimination of two binding sites linked to distinct effector systems
    • 2 analogues in human platelets. Discrimination of two binding sites linked to distinct effector systems. J. Biol. Chem., 265, 6836-6844.
    • (1990) J. Biol. Chem. , vol.265 , pp. 6836-6844
    • Takahara, K.1    Murray, R.2    Fitzgerald, G.A.3    Fitzgerald, D.J.4
  • 40
    • 0028915988 scopus 로고
    • Molecular evolution of receptors for eicosanoids
    • TOH, H., ICHIKAWA, A. & NARUMIYA, S. (1995). Molecular evolution of receptors for eicosanoids. FEBS Lett., 361, 17-21.
    • (1995) FEBS Lett. , vol.361 , pp. 17-21
    • Toh, H.1    Ichikawa, A.2    Narumiya, S.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.