Radiolabeled antimalarials: Synthesis of 14C-artemisinin

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 38, Issue 3, 1996, Pages 263-267

  Avery, Mitchell A ^a,b   Bonk, Jason D ^a   Bupp, James ^c  

^a UNIVERSITY OF MISSISSIPPI   (United States)

^b UNIVERSITY OF MISSISSIPPI   (United States)

^c SRI INTERNATIONAL   (United States)

Author keywords

Artemisinin; Carbon 14; Malaria; Radiolabeled

Indexed keywords

ANTIMALARIAL AGENT; ARTEMISININ; CARBON 14; MALARIA; RADIOCHEMICAL YIELD; RADIOLABELED; STEREO-SELECTIVE; TOTAL SYNTHESIS;

CARBON;

ANTIMALARIAL AGENT; ARTEMISININ; CARBON 14;

ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; ISOTOPE LABELING;

EID: 0029918074     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199603)38:3<263::AID-JLCR839>3.0.CO;2-O     Document Type: Article

References (12)

1. Krogstad, D.J.; Herwaldt, B.L. New Eng. J. Med. 319: 1538 (1988)
2. Marshall, E. Science 247: 399 (1990)
3. Miller, K.D.; Greenberg, A.E.; Campbell, C.C. New Eng. J. Med. 321: 65 (1989)
4. Werdsdorfer, W., ed. World Health Organization Report on Drug-Resistant Malaria. (1982)
5. Luo, X.D.; Shen, C.C. Med. Res. Rev. 7: 29 (1987)
6. Hien, T.T. Trans. Royal Soc. Trop. Med. Hyg. 88, Supplement 1: 7 (1994)
7. Klayman, D.L. Science 228: 1049 (1985)
8. Avery, M.A.; Gao, F.; Chong, W.K.M.; Mehrotra, S.; Jennings-White, C. Trends in Organic Chemistry, Trivandrum, India. Vol. 4: 413 (1993)
9. Brossi, A.; Venugopalan, B.; Dominguez Gerpe, L.; Yeh, H.J.C.; Flippen-Anderson, J.L.; Buchs, P.; Luo, X.D.; Milhous, W.; Peters, W. J. Med. Chem. 31: 645 (1988)
10. China Cooperative Research Group on Qinghaosu and its Derivatives and Antimalarials. J. Trad. Chin. Med. 2: 45 (1982)
11. China Cooperative Research Group on Qinghaosu and its Derivatives and Antimalarials. J. Trad. Chin. Med. 2: 9 (1982)
12. Avery, M.A.; Chong, W.K.M.; Jennings-White, C. J. Am. Chem. Soc. 114: 974 (1992)