Antiandrogen. III. 11-Oxapregnane Steroids

Chemical and Pharmaceutical Bulletin

Volumn 44, Issue 4, 1996, Pages 746-748

  Takegawa, Shigehiro ^a   Koizumi, Naoyuki ^a   Mieda, Mamoru ^a   Shibata, Kenyu ^a  

^a Grelan Pharmaceutical Co Ltd   (Japan)

Author keywords

11 oxachlormadinone acetate; 2,11 dioxachlormadinone acetate; antiandrogen; ventral prostate

Indexed keywords

11 OXACHLORMADINONE ACETATE; 2,11 DIOXACHLORMADINONE ACETATE; ANTIANDROGEN; CHLORMADINONE ACETATE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; CASTRATION; DRUG CONFORMATION; DRUG MECHANISM; DRUG POTENCY; DRUG SYNTHESIS; HORMONE INHIBITION; MALE; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION; SUBCUTANEOUS DRUG ADMINISTRATION;

EID: 0029917466     PISSN: 00092363     EISSN: None     Source Type: Journal    
DOI: 10.1248/cpb.44.746     Document Type: Article

References (11)

1. Part II: Takegawa S., Koizumi N., Takahashi H., Shibata K., Chem. Pharm. Bull., 41, 870-875 (1993).
2. Brennan D. M., Kraay R. J., Acta Endocrinol., 44, 367-379 (1963).
3. Honma S., Iwamura S., Iizuka K., Kambegawa A., Shida K., Chem. Pharm. Bull., 25, 2019-2031 (1977).
4. Engel Ch. R., Rastogi R. C., Chowdhury M. N. Roy, Steroids, 19, 1-24 (1972); Engel Ch. R., Mukherjee D., Chowdhury M. N. Roy, Ramani G., Salvi V. S., J. Steroid Biochem., 6, 585-597 (1975).
5. Engel Ch. R., Rastogi R. C., Chowdhury M. N. Roy, Steroids, 19, 1-24 (1972); Engel Ch. R., Mukherjee D., Chowdhury M. N. Roy, Ramani G., Salvi V. S., J. Steroid Biochem., 6, 585-597 (1975).
6. Ringold H. J., Batres E., Bowers A., Edwards J., Zderic J., J. Am. Chem. Soc., 81, 3485-3486 (1959).
7. Agnello E. J., Laubach G. D., J. Am. Chem. Soc., 82, 4293-4299 (1960).
8. Nussbaum A. L., Brabazon G., Popper T. L., Oliveto E. P., J. Am. Chem. Soc., 80, 2722-2725 (1958).
9. Shibata K., Takegawa S., Koizumi N., Yamakoshi N., Simazawa E., Chem. Pharm. Bull., 40, 935-941 (1992).
10. Slomp G., Johnson J. L., Jr., J. Am. Chem. Soc., 80, 915-921 (1958).
11. Dorfmann R. I., "Methods in Hormone Research," Vol. 2, Academic Press, New York, 1962, pp. 315-340.