C-5 functionalization of trisubstituted imidazoles with azodicarbonyl compounds

Journal of Heterocyclic Chemistry

Volumn 33, Issue 1, 1996, Pages 41-44

  Yamazaki, Chiji ^a   Arima, Hideshi ^a   Udagawa, Satoru ^a  

^a KITASATO UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

IMIDAZOLE DERIVATIVE;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; MASS SPECTROMETRY; NUCLEAR MAGNETIC RESONANCE; ULTRAVIOLET SPECTROPHOTOMETRY;

EID: 0029912984     PISSN: 0022152X     EISSN: None     Source Type: Journal    
DOI: 10.1002/jhet.5570330107     Document Type: Article

References (9)

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3. R. Grigg, R. Hayes and J. L. Jackson, Chem. Commun., 1167 (1969); T. Ibata, S. Nakano, H. Nakawa, J. Toyoda and Y. Isogami, Bull. Chem. Soc. Japan. 59, 433 (1986).
4. R. Grigg, R. Hayes and J. L. Jackson, Chem. Commun., 1167 (1969); T. Ibata, S. Nakano, H. Nakawa, J. Toyoda and Y. Isogami, Bull. Chem. Soc. Japan. 59, 433 (1986).
5. B. Abarca-Gonzalez, R. A. Jones, M. Medio-Simon, J. Quilez-Pardo, J. Sepulveda-Arques and E. Zaballos-Garcia, Synth. Commun., 20, 321 (1990).
6. Based on the actually employed azodicarboxylate, subtracting the amount (0.03 g) of unreacted material.
7. C. J. Moody, Adv. Heterocyclic Chem., 30, 1 (1983).
8. This was prepared using α-bromo-α-di-deuterioacetophenone in place of α-bromoacetophenone by the literature method [8]
9. C. Yamazaki, Bull Chem. Soc. Japan, 51, 1846 (1978).