Peptidyl vinyl sulphones: A new class of potent and selective cysteine protease inhibitors: S2P2 specificity of human cathepsin 02 in comparison with cathepsins S and L

Biochemical Journal

Volumn 315, Issue 1, 1996, Pages 85-89

  Brömme, Dieter ^a   Klaus, Jeff L ^a   Okamoto, Kathleen ^a   Rasnick, David ^a   Palmer, James T ^a  

^a Khepri Pharmaceuticals Inc   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINOCAPROIC ACID; CATHEPSIN L; CATHEPSIN S; CYSTEINE PROTEINASE INHIBITOR; ENZYME VARIANT; NORLEUCINE; PHENYLALANINE; SULFONE DERIVATIVE;

ANIMAL CELL; ARTICLE; COMPARATIVE STUDY; ENZYME SPECIFICITY; HUMAN; INHIBITION KINETICS; NONHUMAN; PRIORITY JOURNAL;

AMINO ACID SEQUENCE; CATHEPSINS; CYSTEINE ENDOPEPTIDASES; CYSTEINE PROTEINASE INHIBITORS; ENDOPEPTIDASES; ENZYME ACTIVATION; HUMANS; KINETICS; MOLECULAR SEQUENCE DATA; SUBSTRATE SPECIFICITY; SULFONES; VINYL COMPOUNDS;

EID: 0029911570     PISSN: 02646021     EISSN: None     Source Type: Journal    
DOI: 10.1042/bj3150085     Document Type: Article

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