메뉴 건너뛰기




Volumn 28, Issue 5-6, 1996, Pages 591-595

Kinetic evidence for isomerization of the dopamine receptor-raclopride complex

Author keywords

[No Author keywords available]

Indexed keywords

DOPAMINE 2 RECEPTOR BLOCKING AGENT; DOPAMINE RECEPTOR; RACLOPRIDE; RADIOLIGAND;

EID: 0029905350     PISSN: 01970186     EISSN: None     Source Type: Journal    
DOI: 10.1016/0197-0186(95)00123-9     Document Type: Article
Times cited : (30)

References (20)
  • 1
    • 0020512496 scopus 로고
    • Antipsychotic drug action: Clinical, biochemical and pharmacological evidence for site specificity of action
    • Borison R. L., Hitri A., Blowers A. J. and Diamond B. (1983) Antipsychotic drug action: clinical, biochemical and pharmacological evidence for site specificity of action. Clin. Neuropharmac. 76, 137-146.
    • (1983) Clin. Neuropharmac. , vol.76 , pp. 137-146
    • Borison, R.L.1    Hitri, A.2    Blowers, A.J.3    Diamond, B.4
  • 2
    • 0002224681 scopus 로고
    • Functional architecture and dynamics of the nicotinic acetylcholine receptors: An allosteric ligand gated ion channel
    • Raven Press, New York
    • Changeaux J.-P. (1990) Functional architecture and dynamics of the nicotinic acetylcholine receptors: an allosteric ligand gated ion channel. In: Fidia Research Foundation Neuroscience Award Lectures, Vol. 4, pp. 21-36. Raven Press, New York.
    • (1990) Fidia Research Foundation Neuroscience Award Lectures , vol.4 , pp. 21-36
    • Changeaux, J.-P.1
  • 3
    • 0023818443 scopus 로고
    • 3H]spiperone with rat striatal dopamine D-2 receptors: Kinetic evidence for antagonist-induced formation of ternary complex
    • 3H]spiperone with rat striatal dopamine D-2 receptors: kinetic evidence for antagonist-induced formation of ternary complex. Molec. Pharmac. 33, 402-413.
    • (1988) Molec. Pharmac. , vol.33 , pp. 402-413
    • Chatterjee, T.K.1    Scott, C.E.2    Vazquez, D.M.3    Bhatnagar, R.K.4
  • 4
    • 0024472937 scopus 로고
    • 3H]raclopride in rat and rabbit brains. Equilibrium binding, kinetics, distribution and selectivity
    • 3H]raclopride in rat and rabbit brains. Equilibrium binding, kinetics, distribution and selectivity. J. Pharmac. exp. Ther. 250, 696-706.
    • (1989) J. Pharmac. Exp. Ther. , vol.250 , pp. 696-706
    • Dewar, K.M.1    Montreuil, B.2    Grondin, L.3    Reader, T.4
  • 5
    • 0025812324 scopus 로고
    • Model systems for the study of seven-transmembrane-segment receptors
    • Dohlman H. G., Thorner J., Caron M. G. and Lefkowitz R. J. (1991) Model systems for the study of seven-transmembrane-segment receptors. A. Rev. Biochem. 60, 653-688.
    • (1991) A. Rev. Biochem. , vol.60 , pp. 653-688
    • Dohlman, H.G.1    Thorner, J.2    Caron, M.G.3    Lefkowitz R, J.4
  • 6
    • 0023920945 scopus 로고
    • Two-step isomerization of quinuclidinyl benzilate-muscarinic receptor complex
    • Eller M. and Järv, J. (1988) Two-step isomerization of quinuclidinyl benzilate-muscarinic receptor complex. Neurochem. Int. 12, 285-289.
    • (1988) Neurochem. Int. , vol.12 , pp. 285-289
    • Eller, M.1    Järv, J.2
  • 8
    • 0002867860 scopus 로고
    • Strategy and tactics in receptor binding studies
    • Hulme E. C., ed.. IRL Press, Oxford
    • Hulme E. C. and Birdsall N. J. M. (1992) Strategy and tactics in receptor binding studies. In: Receptor-Ligand Interactions. A Practical Approach (Hulme E. C., ed.). pp. 63-176. IRL Press, Oxford.
    • (1992) Receptor-ligand Interactions. A Practical Approach , pp. 63-176
    • Hulme, E.C.1    Birdsall, N.J.M.2
  • 9
    • 0008256977 scopus 로고
    • Neurotoxic agents interacting with the muscarinic acetylcholine receptor
    • Herken H. and Hucho F., eds. Springer, Berlin
    • Järv J. (1992) Neurotoxic agents interacting with the muscarinic acetylcholine receptor. In: Selective Neurotoxicity (Herken H. and Hucho F., eds). pp. 659-680. Springer, Berlin.
    • (1992) Selective Neurotoxicity , pp. 659-680
    • Järv, J.1
  • 10
    • 0024205793 scopus 로고
    • Kinetic aspects of L-quinuclidinyl benzilate interaction with muscarinic receptor
    • Järv J. and Eller M. (1988) Kinetic aspects of L-quinuclidinyl benzilate interaction with muscarinic receptor. Neurochem. Int. 13, 419-428.
    • (1988) Neurochem. Int. , vol.13 , pp. 419-428
    • Järv, J.1    Eller, M.2
  • 11
    • 77956861751 scopus 로고
    • Muscarinic acetylcholine receptors
    • Hucho F., ed., Elsevier Science, Amsterdam
    • Järv J. and Rinken A. (1993) Muscarinic acetylcholine receptors. In: Neurotransmitter Receptors (Hucho F., ed.), pp. 199-220. Elsevier Science, Amsterdam.
    • (1993) Neurotransmitter Receptors , pp. 199-220
    • Järv, J.1    Rinken, A.2
  • 12
    • 0018650387 scopus 로고
    • Isomerization of the muscarinic receptor-antagonist complex
    • Järv J., Hedlund B. and Bartfai T. (1979) Isomerization of the muscarinic receptor-antagonist complex. J. biol. Chem. 254, 5595-5598.
    • (1979) J. Biol. Chem. , vol.254 , pp. 5595-5598
    • Järv, J.1    Hedlund, B.2    Bartfai, T.3
  • 13
    • 0021844076 scopus 로고
    • 3H-raclopride. A potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain
    • 3H-raclopride. A potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain. Biochem. Pharmac. 34, 2251-2259.
    • (1985) Biochem. Pharmac. , vol.34 , pp. 2251-2259
    • Köhler, C.1    Hall, H.2    Ögren, S.-O.3    Gawell, L.4
  • 15
    • 0020669405 scopus 로고
    • Determination of total protein
    • Peterson G. L. (1983) Determination of total protein. Meth. Enzymol. 91, 95-119.
    • (1983) Meth. Enzymol. , vol.91 , pp. 95-119
    • Peterson, G.L.1
  • 16
    • 0029028008 scopus 로고
    • Purification of recombinant porcine m2 muscarinic acetylcholine receptor from Chinese hamster ovary cells. Circular dichroism spectra and ligand binding properties
    • Peterson G. L., Toumadje A., Johnson W. C. and Schimerlik M. I. (1995) Purification of recombinant porcine m2 muscarinic acetylcholine receptor from Chinese hamster ovary cells. Circular dichroism spectra and ligand binding properties. J. biol. Chem. 270, 17,808-17,814.
    • (1995) J. Biol. Chem. , vol.270 , pp. 17808-17814
    • Peterson, G.L.1    Toumadje, A.2    Johnson, W.C.3    Schimerlik, M.I.4
  • 17
    • 0021370898 scopus 로고
    • Kinetics of the interaction of dihydroalperonal with beta-adrenergic receptors in red cerebral cortex
    • Schiliebs R. and Bigl V. (1984) Kinetics of the interaction of dihydroalperonal with beta-adrenergic receptors in red cerebral cortex. Gen. Physiol. Biophys. 3, 31-46.
    • (1984) Gen. Physiol. Biophys. , vol.3 , pp. 31-46
    • Schiliebs, R.1    Bigl, V.2
  • 19
    • 0016749447 scopus 로고
    • Determination of dissociation constants and specific rate constants of enzyme-substrate (or protein-ligand) interactions from rapid reaction kinetic data
    • Strickland S., Palmer G. and Massey V. (1975) Determination of dissociation constants and specific rate constants of enzyme-substrate (or protein-ligand) interactions from rapid reaction kinetic data. J. biol. Chem. 250, 4048-4052.
    • (1975) J. Biol. Chem. , vol.250 , pp. 4048-4052
    • Strickland, S.1    Palmer, G.2    Massey, V.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.