Kinetics of the interaction of nonsteroidal antiinflammatory drugs with prostaglandin endoperoxide synthase-1 studied by limited proteolysis

Biochemistry

Volumn 35, Issue 28, 1996, Pages 9076-9082

  Kalgutkar, Amit S ^a   Crews, Brenda C ^a   Marnett, Lawrence J ^a  

^a VANDERBILT UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

NONSTEROID ANTIINFLAMMATORY AGENT; PROSTAGLANDIN SYNTHASE;

ARTICLE; DRUG EFFECT; DRUG PROTEIN BINDING; ENZYME CONFORMATION; ENZYME KINETICS; INFLAMMATION; NONHUMAN; PRIORITY JOURNAL; PROTEIN DEGRADATION;

ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; ARACHIDONIC ACID; CYCLOOXYGENASE INHIBITORS; HEMIN; IBUPROFEN; KINETICS; MOLECULAR STRUCTURE; NITROBENZENES; PROSTAGLANDIN-ENDOPEROXIDE SYNTHASES; PROSTANOIC ACIDS; PROTEIN BINDING; PROTEIN CONFORMATION; SULFONAMIDES; THIAZOLES; TRYPSIN;

EID: 0029893612     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi9605752     Document Type: Article

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