메뉴 건너뛰기




Volumn 23, Issue 5, 1996, Pages 438-440

Dose dependent in vivo inhibition of human colorectal cancer (LoVo) by the gastrin receptor antagonist, CI-988

Author keywords

Antagonist; CCK B; Cholecystokinin; CI 988; Colon cancer; Gastrin; Gastrin receptor antagonists; In vivo; Receptor

Indexed keywords

4 [[2 [2 [[(2 ADAMANTYLOXY)CARBONYL]AMINO] 3 (1H INDOL 3 YL) 2 METHYLPROPIONAMIDO] 1 PHENYLETHYL]AMINO] 4 OXOBUTYRIC ACID MEGLUMINE; GASTRIN ANTAGONIST;

EID: 0029893577     PISSN: 03051870     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1440-1681.1996.tb02756.x     Document Type: Article
Times cited : (6)

References (24)
  • 1
    • 0021591222 scopus 로고
    • Gastrin receptors in a mouse colon cancer cell line responsive to trophic effects of gastrin
    • Singh P, Townsend CM, Walker JP, Thompson JC. Gastrin receptors in a mouse colon cancer cell line responsive to trophic effects of gastrin. Surg. Forum 1984; 35: 205-6.
    • (1984) Surg. Forum , vol.35 , pp. 205-206
    • Singh, P.1    Townsend, C.M.2    Walker, J.P.3    Thompson, J.C.4
  • 2
    • 0023019897 scopus 로고
    • Stimulation of growth of a colon cancer cell line by gastrin
    • Kusyk CJ, McNeil NO, Johnson LR. Stimulation of growth of a colon cancer cell line by gastrin. Am. J. Physiol. 1986; 251: G597-601.
    • (1986) Am. J. Physiol. , vol.251
    • Kusyk, C.J.1    McNeil, N.O.2    Johnson, L.R.3
  • 3
    • 0022617804 scopus 로고
    • Role of gastrin and gastrin receptors on the growth of a transplantante mouse colon carcinoma (MC-26) in BALB/c mice
    • Singh P, Walker JP, Townsend CM Jr, Thompson JC. Role of gastrin and gastrin receptors on the growth of a transplantante mouse colon carcinoma (MC-26) in BALB/c mice. Cancer Res. 1986; 46: 1612-16.
    • (1986) Cancer Res. , vol.46 , pp. 1612-1616
    • Singh, P.1    Walker, J.P.2    Townsend Jr., C.M.3    Thompson, J.C.4
  • 6
    • 0023882724 scopus 로고
    • Growth-promoting action of gastrin on human colonie and gastric tumor cells cultured in vitro
    • Watson SA, Durrant LG, Morris DL. Growth-promoting action of gastrin on human colonie and gastric tumor cells cultured in vitro. Br. J. Surg. 1988; 75: 342-5.
    • (1988) Br. J. Surg. , vol.75 , pp. 342-345
    • Watson, S.A.1    Durrant, L.G.2    Morris, D.L.3
  • 7
    • 0024517113 scopus 로고
    • The in vitro growth response of primary human colorectal and gastric cancer cells to gastrin
    • Watson SA, Durrant LG, Crosbie JD, Morris DL. The in vitro growth response of primary human colorectal and gastric cancer cells to gastrin. Int. J. Cancer 1989; 43: 692-6.
    • (1989) Int. J. Cancer , vol.43 , pp. 692-696
    • Watson, S.A.1    Durrant, L.G.2    Crosbie, J.D.3    Morris, D.L.4
  • 8
    • 0025008856 scopus 로고
    • Evidence for autocrine growth stimulation of cultured colon tumor cells by gastrin/cholecystokinin-like peptide
    • Hoosein NM, Kiener PA, Curry RC, Brattain MG. Evidence for autocrine growth stimulation of cultured colon tumor cells by gastrin/cholecystokinin-like peptide. Exp. Cell Res. 1990; 186: 15-21.
    • (1990) Exp. Cell Res. , vol.186 , pp. 15-21
    • Hoosein, N.M.1    Kiener, P.A.2    Curry, R.C.3    Brattain, M.G.4
  • 10
    • 0025980628 scopus 로고
    • Inhibition of cell proliferation by the cholecystokinin antagonist L364,718
    • Thumwood CM, Hong J, Baldwin GS. Inhibition of cell proliferation by the cholecystokinin antagonist L364,718. Exp. Cell Res. 1991; 192: 189-92.
    • (1991) Exp. Cell Res. , vol.192 , pp. 189-192
    • Thumwood, C.M.1    Hong, J.2    Baldwin, G.S.3
  • 11
    • 0025936503 scopus 로고
    • Inhibitory effects of the gastrin receptor antagonist (L365,260) on gastrointestinal tumor cells
    • Watson S, Durrant L, Elston P, Morris DL. Inhibitory effects of the gastrin receptor antagonist (L365,260) on gastrointestinal tumor cells. Cancer 1991; 68: 1255-60.
    • (1991) Cancer , vol.68 , pp. 1255-1260
    • Watson, S.1    Durrant, L.2    Elston, P.3    Morris, D.L.4
  • 12
    • 0025064695 scopus 로고
    • The effect of the gastrin receptor antagonist proglumide on survival in gastric carcinoma
    • Harrison JD, Jones JA, Morris DL. The effect of the gastrin receptor antagonist proglumide on survival in gastric carcinoma. Cancer 1990; 66: 1449-52.
    • (1990) Cancer , vol.66 , pp. 1449-1452
    • Harrison, J.D.1    Jones, J.A.2    Morris, D.L.3
  • 13
    • 0025013978 scopus 로고
    • Development of a class of selective cholecystokinin type B receptor antagonists having potent anxiolytic activity
    • Hughes J, Boden P, Costall B et al. Development of a class of selective cholecystokinin type B receptor antagonists having potent anxiolytic activity. Proc. Natl Acad. Sci. USA 1990; 87: 6728-32.
    • (1990) Proc. Natl Acad. Sci. USA , vol.87 , pp. 6728-6732
    • Hughes, J.1    Boden, P.2    Costall, B.3
  • 14
    • 0026649452 scopus 로고
    • Aqueous stability and solubility of CI-988, a novel 'dipeptoid'cholecystokinin-B receptor antagonist
    • Kearney AS, Mehta SC, Radebaugh GW. Aqueous stability and solubility of CI-988, a novel 'dipeptoid'cholecystokinin-B receptor antagonist. Pharm. Res. 1992; 9: 1092-5.
    • (1992) Pharm. Res. , vol.9 , pp. 1092-1095
    • Kearney, A.S.1    Mehta, S.C.2    Radebaugh, G.W.3
  • 15
    • 0029958939 scopus 로고    scopus 로고
    • Gastrin receptor antagonist, CI-988, inhibits basal growth of a human colon cancer cell line both in vivo and in vitro
    • in press
    • Romani R, Howes LG, Morris DL. Gastrin receptor antagonist, CI-988, inhibits basal growth of a human colon cancer cell line both in vivo and in vitro. Aust. N.Z. J. Surg. 1996 (in press).
    • (1996) Aust. N.Z. J. Surg.
    • Romani, R.1    Howes, L.G.2    Morris, D.L.3
  • 16
    • 0017259817 scopus 로고
    • Establishment of a human carcinoembryonic antigen-producing colon adenocarcinoma cell line
    • Drewinko B, Ramsdahl MM, Yang LY, Ahearn MJ, Trujillo LM. Establishment of a human carcinoembryonic antigen-producing colon adenocarcinoma cell line. Cancer Res. 1976; 36: 467-75.
    • (1976) Cancer Res. , vol.36 , pp. 467-475
    • Drewinko, B.1    Ramsdahl, M.M.2    Yang, L.Y.3    Ahearn, M.J.4    Trujillo, L.M.5
  • 17
    • 3643113361 scopus 로고
    • Potent new family of gastrin receptor antagonists (GRAs) produces in vitro and in vivo inhibition of human colorectal cancer (CRC) cell lines
    • A2369
    • Romani R, Howes LG, Morris DL. Potent new family of gastrin receptor antagonists (GRAs) produces in vitro and in vivo inhibition of human colorectal cancer (CRC) cell lines. Proc. Am. Assoc. Cancer Res. 1994; 35: 397 (A2369).
    • (1994) Proc. Am. Assoc. Cancer Res. , vol.35 , pp. 397
    • Romani, R.1    Howes, L.G.2    Morris, D.L.3
  • 18
    • 0028351718 scopus 로고
    • Effects of gastrin on 3′,5′-cyclic adenosine monophosphate, intracellular calcium, and phosphatidylinositol hydrolysis in human colon cancer cells
    • Ishizuka J, Townsend CM Jr, Bold RJ, Martinez J, Rodriguez M, Thompson JC. Effects of gastrin on 3′,5′-cyclic adenosine monophosphate, intracellular calcium, and phosphatidylinositol hydrolysis in human colon cancer cells. Cancer Res. 1994; 54: 2129-35.
    • (1994) Cancer Res. , vol.54 , pp. 2129-2135
    • Ishizuka, J.1    Townsend Jr., C.M.2    Bold, R.J.3    Martinez, J.4    Rodriguez, M.5    Thompson, J.C.6
  • 19
    • 0026053051 scopus 로고
    • In vitro influence of gastrin, oestradiol and gonadotropin-releasing hormone on HCT-15 and LoVo human colorectal neoplastic cell proliferation
    • Kiss R, Salom I, Pauwels O et al. In vitro influence of gastrin, oestradiol and gonadotropin-releasing hormone on HCT-15 and LoVo human colorectal neoplastic cell proliferation. Eur. J. Cancer 1991; 27: 1268-74.
    • (1991) Eur. J. Cancer , vol.27 , pp. 1268-1274
    • Kiss, R.1    Salom, I.2    Pauwels, O.3
  • 20
    • 0343531708 scopus 로고
    • Gastrin trophic effects on transplanted colon cancer cells
    • Walsh JH (ed.). Raven Press, New York
    • Townsend CM, Ishizuka J, Thompson JC. Gastrin trophic effects on transplanted colon cancer cells. In: Walsh JH (ed.). Gastrin. Raven Press, New York. 1993; 407-17.
    • (1993) Gastrin , pp. 407-417
    • Townsend, C.M.1    Ishizuka, J.2    Thompson, J.C.3
  • 23
    • 0023264943 scopus 로고
    • Inhibition of pentagastrin stimulated up-regulation of gastrin receptors and growth of mouse colon tumor in vivo by proglumide, a gastrin receptor antagonist
    • Singh P, Le S, Beauchamp P, Townsend CM, Thompson JC. Inhibition of pentagastrin stimulated up-regulation of gastrin receptors and growth of mouse colon tumor in vivo by proglumide, a gastrin receptor antagonist. Cancer Res. 1987; 47: 5000-4.
    • (1987) Cancer Res. , vol.47 , pp. 5000-5004
    • Singh, P.1    Le, S.2    Beauchamp, P.3    Townsend, C.M.4    Thompson, J.C.5
  • 24
    • 0025073147 scopus 로고
    • Alpha-methyl trytophanylphenylalanines and their arylethylamine 'dipeptoid' analogues of the tetrapeptide cholecystokinin (30-33)
    • Horwell DC, Birchmore B, Boden PR et al. Alpha-methyl trytophanylphenylalanines and their arylethylamine 'dipeptoid' analogues of the tetrapeptide cholecystokinin (30-33). Eur. J. Med. Chem. 1990; 25: 53-60.
    • (1990) Eur. J. Med. Chem. , vol.25 , pp. 53-60
    • Horwell, D.C.1    Birchmore, B.2    Boden, P.R.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.