4-Substituted 1-(2-methylphenyl)thieno[2,3-c]-1,5-naphthyridines as possible reversible inhibitors of gastric H+,K+-ATPase

European Journal of Medicinal Chemistry

Volumn 31, Issue 5, 1996, Pages 411-416

  Bjork P ^a   Hornfeldt A B ^a   Gronowitz, S ^a   Edvardsson, U ^b  

^a LUND UNIVERSITY   (Sweden)

^b ASTRAZENECA R AND D   (Sweden)

Author keywords

Chlorination; Gastric H+,K+ ATPase cross coupling; Heterocycle; Oxidation

Indexed keywords

1 (2 METHYLPHENYL) 4 (1 METHYL 4 PIPERAZINYL)THIENO[2,3 C][1,5]NAPHTHYRIDINE; 3 BUTYRYL 8 METHOXY 4 (2 METHYLANILINO)QUINOLINE; ADENOSINE TRIPHOSPHATASE (POTASSIUM); ANTIULCER AGENT; NAPHTHYRIDINE DERIVATIVE; THIENO[2,3 C][1,5]NAPHTHYRIDONE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; ENZYME INHIBITION; MEMBRANE VESICLE; NONHUMAN; RABBIT; REACTION ANALYSIS; STOMACH ACID SECRETION; STOMACH GLAND; SWINE;

EID: 0029890340     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/0223-5234(96)89168-9     Document Type: Article

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