Endothelins and endothelin receptor antagonists: Binding to plasma proteins

Life Sciences

Volumn 58, Issue 21, 1996, Pages 1839-1847

  Wu Wong, Jinshyun R ^a   Chiou, William J ^a   Hoffman, Daniel J ^a   Winn, Martin ^a   Von Geldern, Thomas W ^a   Opgenorth, Terry J ^a  

^a ABBOTT LABORATORIES   (United States)

Author keywords

A 127722; endothelin; endothelin receptor; L 749329; PD 156707; Ro 47 0203

Indexed keywords

2 (4 CARBOXY 2 PROPYLPHENOXY) N (4 ISOPROPYLBENZENESULFONYL) 2 (3,4 METHYLENEDIOXYPHENYL)ACETAMIDE; 4 (4 METHOXYPHENYL) 2 (3,4 METHYLENEDIOXYPHENYL) 4 OXO 3 (3,4,5 TRIMETHOXYBENZYL) 2 BUTENOIC ACID; A 127772; BOSENTAN; ENDOTHELIN; ENDOTHELIN 1; ENDOTHELIN 3; ENDOTHELIN A RECEPTOR; ENDOTHELIN B RECEPTOR; ENDOTHELIN RECEPTOR; ENDOTHELIN RECEPTOR ANTAGONIST; HUMAN SERUM ALBUMIN; IODINE 125; L 749329; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BINDING COMPETITION; CELL MEMBRANE; CEREBELLUM; CHO CELL; CONTROLLED STUDY; DRUG POTENCY; HUMAN; HYPOPHYSIS CELL; LIGAND BINDING; NONHUMAN; PATHOPHYSIOLOGY; PLASMA; PLASMA PROTEIN BINDING; RAT; RECEPTOR BINDING; SWINE;

ANIMALIA; SUS SCROFA;

EID: 0029886638     PISSN: 00243205     EISSN: None     Source Type: Journal    
DOI: 10.1016/0024-3205(96)00168-3     Document Type: Article

References (17)

1. M. YANAGISAWA, H. KURIHARA, S. KIMURA, Y. TOMOBE, Y. KOBAYASHI, M. MITSUI, Y. YAZAKI, K. GOTO, and T. MASAKI, Nature (London) 332 411-415 (1988).
2. A. INOUE, M. YANAGISAWA, S. KIMURA, Y. KASUYA, T. MIYAUCHI, K. GOTO and T. MASAKI, Proc. Natl. Acad. Sci. USA 86 2863-2867 (1989).
3. M. SOKOLOVSKY, J. Neurochem. 59 809-821 (1992).
4. M. KOZUKA, T. ITO, S. HIROSE, K. M. LODHI and H. HAGIWARA, J. Biol. Chem. 266 16892-16896 (1991).
5. K. WADA, H. TABUCHI, R. OHBA, M. SATOH, Y. TACHIBANA, N. AKIYAMA, O. HIRAOKA, A. ASAKURA, C. MIYAMOTO and Y. FURUICHI, Biochem, Biophys. Res. Commun. 167 251-257 (1990).
6. H. ARAI, S. HORI, I. ARIMORI, H. OHKUBO and S. NAKANISHI, Nature (London) 348 730-732 (1990).
7. T. SAKURAI, M. YANAGISAWA, Y. TAKUWA, H. MIYAZAKI, S. KIMURA, K. GOTO and T. MASAKI, Nature (London) 348 732-735 (1990).
8. H. Y. LIN, E. H. KAJI, G. K. WINKEL, H. E. IVES and H. F. LODISH, Proc. Natl. Acad. Sci. USA 88 3185-3189 (1991).
9. T. J. OPGENORTH, Advances in Pharmacology 33 1-65 (1995).
10. E. E. REYNOLDS, J. A. KEISER, S. J. HALEEN, D. M. WALKER, B. OLSZEWSKI, R. L. SCHROEDER, D. G. TAYLOR, OK HWANG, K. M. WELCH, M. A. FLYNN, D. M. THOMPSON, J. J. EDMUNDS, K. A. BERRYMAN, M. PLUMMER, X.-M. CHENG, W. C. PATT and A. M. DOHERTY, J. Pharm. Exp. Ther. 273 1410-1417 (1995).
11. T. F. WALSH, Annual Reports in Medicinal Chemistry, 91-100, Academic Press, (1995).
12. M. CLOZEL, V. BREU, G. A. GRAY, B. KALINA, B.-M. LÖFFLER, K. BURRI, J.-M. CASSAL, G. HIRTH, M. MÜLLER, W. NEIDHART and H. RAMUZ, J. Pharm. Exp. Ther. 264 1040-1046 (1993).
13. T. J. OPGENORTH, A. L. ADLER, S. CALZADILLA, W. J. CHIOU, B. D. DAYTON, D. B. DIXON, L. J. GEHRKE, L. HERNANDEZ, S. R. MAGNUSON, K. MARSH, E. I. NOVOSAD, T. W. VON GELDERN, J. L. WESSALE, M. WINN, and J. R. WU-WONG, J. Pharm. Exp. Ther. in press (1995).
14. J. R. WU-WONG, W. CHIOU, K. E. NAUGLES, and T. J. OPGENORTH, Biochim. Biophys. Acta 1224 288-294 (1994).
15. J. R. WU-WONG, W. CHIOU, Z.-J. HUANG, M. J. VIDAL, and T. J. OPGENORTH, Am. J. Physiol. 267 C1185-C1195 (1994).
16. J. R. WU-WONG, W. CHIOU and T. J. OPGENORTH, Mol. Pharmacol. 44 422-429 (1993).
17. W. F. BOWERS, S. FULTON, and J. THOMPSON, Clincal Pharmacokinetics 9 49-60 (1984).