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Volumn 6, Issue 2, 1996, Pages 148-156

Permeation enhancement of methionine enkephalin by combinations of enzyme inhibitors and enhancers

Author keywords

Enzyme inhibitor; Methionine enkephalin; Penetration enhancer; Permeation; Transmucosal delivery

Indexed keywords

ENZYME INHIBITOR; FUSIDIC ACID DERIVATIVE; METENKEPHALIN; UNCLASSIFIED DRUG;

EID: 0029884147     PISSN: 11571489     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (1)

References (30)
  • 1
    • 0024310984 scopus 로고
    • Modification of morphine withdrawal in rats by alterations of the endogenous opioid system : Effects of actinonin and GEMSA
    • DZOLJIC D AND DZOLJIC M.R. - Modification of morphine withdrawal in rats by alterations of the endogenous opioid system : effects of actinonin and GEMSA. - Drug Dev. Res., 18, 255-261, 1989.
    • (1989) Drug Dev. Res. , vol.18 , pp. 255-261
    • Dzoljic, D.1    Dzoljic, M.R.2
  • 2
    • 0022297929 scopus 로고
    • Hydrolysis of leucine enkephalin in the nasal cavity of the rat : A possible factor in the low bioavailability of nasally administered peptides
    • HUSSAIN A., FARAJ J., ARAMAKI Y. and TRUELOVE J.E. - Hydrolysis of leucine enkephalin in the nasal cavity of the rat : a possible factor in the low bioavailability of nasally administered peptides. - Biochem. Biophys. Res. Commun., 133, 923-928, 1985.
    • (1985) Biochem. Biophys. Res. Commun. , vol.133 , pp. 923-928
    • Hussain, A.1    Faraj, J.2    Aramaki, Y.3    Truelove, J.E.4
  • 3
    • 0022460440 scopus 로고
    • Enkephalin hydrolysis in homogenates of various absorptive mucosas of the albino rabbit : Similarities in rats and involvement of aminopeptidases
    • DODDA-KASHI S. and LEE V.H.L. - Enkephalin hydrolysis in homogenates of various absorptive mucosas of the albino rabbit : similarities in rats and involvement of aminopeptidases. - Life Sci., 38, 2019-2028, 1986.
    • (1986) Life Sci. , vol.38 , pp. 2019-2028
    • Dodda-Kashi, S.1    Lee, V.H.L.2
  • 4
    • 0022495940 scopus 로고
    • Hydrolysis of enkephalins in homogenates of anterior segment tissues of the albino rabbit eyes
    • DODDA-KASHI S. and LEE V.H.L. - Hydrolysis of enkephalins in homogenates of anterior segment tissues of the albino rabbit eyes. - Invest. Ophthalmol. Vis. Sci., 27, 1300-1303, 1986.
    • (1986) Invest. Ophthalmol. Vis. Sci. , vol.27 , pp. 1300-1303
    • Dodda-Kashi, S.1    Lee, V.H.L.2
  • 5
    • 0023723477 scopus 로고
    • Buccal drug absorption. I. Comparative levels of esterase and peptidase activities in rat and hamster buccal and intestinal homogenates
    • GARREN K.W. and REPTA A.J. - Buccal drug absorption. I. Comparative levels of esterase and peptidase activities in rat and hamster buccal and intestinal homogenates. - Int. J. Pharm., 48, 189-194, 1988.
    • (1988) Int. J. Pharm. , vol.48 , pp. 189-194
    • Garren, K.W.1    Repta, A.J.2
  • 6
    • 0025224856 scopus 로고
    • Transdermal delivery of bioactive peptides : The effect of n-decylmethyl sulfoxide, pH, and inhibitors on enkephalin metabolism and transport
    • CHOI H K., FLYNN G.L. and AMIDON G.L. - Transdermal delivery of bioactive peptides : the effect of n-decylmethyl sulfoxide, pH, and inhibitors on enkephalin metabolism and transport. - Pharm. Res., 7, 1099-1106, 1990.
    • (1990) Pharm. Res. , vol.7 , pp. 1099-1106
    • Choi, H.K.1    Flynn, G.L.2    Amidon, G.L.3
  • 7
    • 0027156176 scopus 로고
    • Transmucosal delivery of methionine enkephalin. I. Solution stability and kinetics of degradation in various rabbit mucosa extracts
    • CHUN I.K and CHIEN Y.W. - Transmucosal delivery of methionine enkephalin. I. Solution stability and kinetics of degradation in various rabbit mucosa extracts. - J. Pharm. Sci., 82, 373-378, 1993.
    • (1993) J. Pharm. Sci. , vol.82 , pp. 373-378
    • Chun, I.K.1    Chien, Y.W.2
  • 8
    • 0021832039 scopus 로고
    • Aminopeptidase activity in albino rabbit extraocular tissues relative to the small intestine
    • STRATFORD R.E. Jr. and LEE V.H.L. - Aminopeptidase activity in albino rabbit extraocular tissues relative to the small intestine. - J. Pharm. Sci., 74, 731-734, 1985.
    • (1985) J. Pharm. Sci. , vol.74 , pp. 731-734
    • Stratford Jr., R.E.1    Lee, V.H.L.2
  • 9
    • 0022592643 scopus 로고
    • Aminopeptidase activity in homogenates of various absorptive mucosae in the albino rabbit : Implication in peptide delivery
    • STRATFORD R E. Jr. and LEE V.HL. - Aminopeptidase activity in homogenates of various absorptive mucosae in the albino rabbit : implication in peptide delivery. - Int. J. Pharm., 30, 73-82, 1986.
    • (1986) Int. J. Pharm. , vol.30 , pp. 73-82
    • Stratford Jr., R.E.1    Lee, V.H.L.2
  • 11
    • 0024539596 scopus 로고
    • The use of α-aminoboronic acid derivatives to stabilize peptide drugs during their intranasal absorption
    • HUSSAIN M.A., SHENVI A.B., ROWE S.M. and SHEFTER E. - The use of α-aminoboronic acid derivatives to stabilize peptide drugs during their intranasal absorption. - Pharm. Res., 6, 186-189, 1989.
    • (1989) Pharm. Res. , vol.6 , pp. 186-189
    • Hussain, M.A.1    Shenvi, A.B.2    Rowe, S.M.3    Shefter, E.4
  • 14
    • 0024208342 scopus 로고
    • Systemic absorption of ocularly administered enkephalinamide and inulin in the albino rabbit : Extent, pathways, and vehicle effects
    • STRATFORD R.E. Jr., CARSON L.W., DODDA-KASHI S. and LEE V.H.L. - Systemic absorption of ocularly administered enkephalinamide and inulin in the albino rabbit : extent, pathways, and vehicle effects. - J. Pharm. Sci., 77. 838-842, 1988.
    • (1988) J. Pharm. Sci. , vol.77 , pp. 838-842
    • Stratford Jr., R.E.1    Carson, L.W.2    Dodda-Kashi, S.3    Lee, V.H.L.4
  • 15
    • 0020546435 scopus 로고
    • Studies on the transport of enkephalin-like oligopeptides in rat intestinal mucosa
    • KERCHNER G.A. and GEARY L.E. - Studies on the transport of enkephalin-like oligopeptides in rat intestinal mucosa. - J. Pharmacol. Exp. Ther., 226, 33-38, 1983.
    • (1983) J. Pharmacol. Exp. Ther. , vol.226 , pp. 33-38
    • Kerchner, G.A.1    Geary, L.E.2
  • 16
    • 0029030420 scopus 로고
    • Stabilization of methionine enkephalin in various rabbit mucosal extracts by enzyme inhibitors
    • CHUN I.K. and CHIEN Y.W. - Stabilization of methionine enkephalin in various rabbit mucosal extracts by enzyme inhibitors. - Int. J. Pharm., 121, 217-231, 1995.
    • (1995) Int. J. Pharm. , vol.121 , pp. 217-231
    • Chun, I.K.1    Chien, Y.W.2
  • 18
    • 0023241884 scopus 로고
    • Simple spectrophotometric determination of urinary albumin by dye-binding with use of bromphenol blue
    • SCHOSINSKY K.H., VARGAS M., EQUIVEL A.L. and CHAVARRIA M.A. - Simple spectrophotometric determination of urinary albumin by dye-binding with use of bromphenol blue. - Clin. Chem., 33, 223-226, 1987.
    • (1987) Clin. Chem. , vol.33 , pp. 223-226
    • Schosinsky, K.H.1    Vargas, M.2    Equivel, A.L.3    Chavarria, M.A.4
  • 19
    • 0024207642 scopus 로고
    • Quantification of albumin in cerebrospinal fluid
    • BONATE P.L. - Quantification of albumin in cerebrospinal fluid. - Anal. Biochem., 175, 300-304, 1988.
    • (1988) Anal. Biochem. , vol.175 , pp. 300-304
    • Bonate, P.L.1
  • 20
    • 0025253424 scopus 로고
    • Characterization of the barrier properties of mucosal membranes
    • CORBO D.C., LIU J.C. and CHIEN Y.W - Characterization of the barrier properties of mucosal membranes. - J. Pharm Sci, 79, 202-206, 1990.
    • (1990) J. Pharm Sci , vol.79 , pp. 202-206
    • Corbo, D.C.1    Liu, J.C.2    Chien, Y.W.3
  • 21
    • 0019426552 scopus 로고
    • Mechanisms for the enhancement of the nasal absorption of insulin by surfactants
    • HIRAI S., YOSHIKI T. and MIMA H. - Mechanisms for the enhancement of the nasal absorption of insulin by surfactants. - Int J. Pharm., 9, 173-184, 1981.
    • (1981) Int J. Pharm. , vol.9 , pp. 173-184
    • Hirai, S.1    Yoshiki, T.2    Mima, H.3
  • 24
    • 0024316885 scopus 로고
    • Absorption enhancement of intranasally administered insulin by sodium taurodihydrofusidate (STDHF) in rabbits and rats
    • DEURLOO M.J.M., HERMENS W.A.J.J., ROMEYN S.G., VERHOEF J.C. and MERKUS F.W.H.M. - Absorption enhancement of intranasally administered insulin by sodium taurodihydrofusidate (STDHF) in rabbits and rats. - Pharm. Res., 6, 853-856, 1989.
    • (1989) Pharm. Res. , vol.6 , pp. 853-856
    • Deurloo, M.J.M.1    Hermens, W.A.J.J.2    Romeyn, S.G.3    Verhoef, J.C.4    Merkus, F.W.H.M.5
  • 25
    • 0025007507 scopus 로고
    • The effects of permeation enhancers on the surface morphology of the rat nasal mucosa : A scanning electron microscopy study
    • ENNIS R.D., BORDEN L. and LEE W.A. - The effects of permeation enhancers on the surface morphology of the rat nasal mucosa : a scanning electron microscopy study. - Pharm. Res., 7, 468-475, 1990.
    • (1990) Pharm. Res. , vol.7 , pp. 468-475
    • Ennis, R.D.1    Borden, L.2    Lee, W.A.3
  • 26
    • 0025313194 scopus 로고
    • Effects of absorption enhancers on human nasal tissue ciliary movement in vitro
    • HERMENS W.A.J.J., HOOYMANS P.M., VERHOEF J C. and MERKUS F.W.H.M. - Effects of absorption enhancers on human nasal tissue ciliary movement in vitro. - Pharm. Res., 7, 144-146, 1990.
    • (1990) Pharm. Res. , vol.7 , pp. 144-146
    • Hermens, W.A.J.J.1    Hooymans, P.M.2    Verhoef, J.C.3    Merkus, F.W.H.M.4
  • 27
    • 0025312082 scopus 로고
    • Recovery of rat nasal mucosa from the effects of aminopeptidase inhibitors
    • HUSSAIN M.A., KOLVAL C.A., SHENVI A.B. and AUNGST B.J. - Recovery of rat nasal mucosa from the effects of aminopeptidase inhibitors. - J Pharm. Sci., 79, 398-400, 1990.
    • (1990) J Pharm. Sci. , vol.79 , pp. 398-400
    • Hussain, M.A.1    Kolval, C.A.2    Shenvi, A.B.3    Aungst, B.J.4
  • 28
    • 0025377458 scopus 로고
    • Absorption enhancement of rectally infused insulin by sodium tauro-24,25-dihydrofusidate (STDHF) in rats
    • HOOGDALEM V.EJ., HEULINGER-FEIJEN C.D., VERHOEF J.C., BOER A.G. and BREIMER D.D. - Absorption enhancement of rectally infused insulin by sodium tauro-24,25-dihydrofusidate (STDHF) in rats. - Pharm. Res., 7, 180-183, 1990.
    • (1990) Pharm. Res. , vol.7 , pp. 180-183
    • Hoogdalem, V.E.J.1    Heulinger-Feijen, C.D.2    Verhoef, J.C.3    Boer, A.G.4    Breimer, D.D.5
  • 29
    • 0019790314 scopus 로고
    • Biological inactivation of enkephalins and the role of enkephalin-dipeptidyl-carboxylpeptidase (« enkephalinase ») as neuropeptidase
    • SCHWARTZ J.C., MALFROY B. and BAUME S.D.L. - Biological inactivation of enkephalins and the role of enkephalin-dipeptidyl-carboxylpeptidase (« enkephalinase ») as neuropeptidase. -Life Sci., 29, 1715-1740, 1988.
    • (1988) Life Sci. , vol.29 , pp. 1715-1740
    • Schwartz, J.C.1    Malfroy, B.2    Baume, S.D.L.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.