Halogenated analogs of the antimalarial bialamicol

Synthesis

Volumn , Issue 5, 1996, Pages 591-593

  Schlosser, Manfred ^a   Michel, Dominique ^a   Croft, Simon L ^b  

^a UNIVERSITY OF LAUSANNE   (Switzerland)

^b LONDON SCHOOL OF HYGIENE AND TROPICAL MEDICINE   (United Kingdom)

Author keywords

2 fluoroallyl moieties; C3F building block; Claisen rearrangement; Mannich reaction; tropical diseases

Indexed keywords

ANTIMALARIAL AGENT; BIALAMICOL DERIVATIVE; BIPHENYL DERIVATIVE; UNCLASSIFIED DRUG;

ANTIPROTOZOAL ACTIVITY; ARTICLE; DRUG SYNTHESIS; HUMAN; LEISHMANIA DONOVANI; REACTION ANALYSIS; TRYPANOSOMA BRUCEI; TRYPANOSOMA CRUZI;

EID: 0029882607     PISSN: 00397881     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-1996-4262     Document Type: Article

References (9)

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3. Hung, J.; Werbel, L. M. Eur. J. Med. Chem. 1983, 18, 61.
4. Schlosser, M. Tetrahedron 1978, 34, 3.
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6. For details see: Michel, D. Ph. D. Thesis, Ecole Polytechnique Fédérale, Lausanne, 1995.
7. Nagakura, I.; Savary, D. N. H.; Schlosser, M. Helv. Chim. Acta 1980, 63, 1257.
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