메뉴 건너뛰기




Volumn 212, Issue 1, 1996, Pages 84-93

Efficacy of the class III antiarrhythmic agent azimilide in rodent models of ventricular arrhythmia

Author keywords

[No Author keywords available]

Indexed keywords

1 [2 (6 METHYL 2 PYRIDYL)ETHYL] 4 (4 METHYLSULFONYLAMINOBENZOYL)PIPERIDINE; ANTIARRHYTHMIC AGENT; AZIMILIDE; DOFETILIDE; OUABAIN; SEMATILIDE;

EID: 0029878868     PISSN: 00379727     EISSN: None     Source Type: Journal    
DOI: 10.3181/00379727-212-43995     Document Type: Article
Times cited : (23)

References (44)
  • 1
    • 0345578344 scopus 로고
    • In vitro electrophysiology of NE-10064, a novel and highly selective class III antiarrhythmic agent
    • Tatla DS, David BC, Malloy KJ, Moorehead TJ. In vitro electrophysiology of NE-10064, a novel and highly selective class III antiarrhythmic agent. FASEB J 7:A107-615, 1993.
    • (1993) FASEB J , vol.7
    • Tatla, D.S.1    David, B.C.2    Malloy, K.J.3    Moorehead, T.J.4
  • 4
    • 3042994764 scopus 로고
    • Effects of clofilium and NE-10064 on IKs, the slow component of the cardiac delayed rectifier
    • Smith MA, Conder ML, Atwal KS, McCullough JR. Effects of clofilium and NE-10064 on IKs, the slow component of the cardiac delayed rectifier. Biophys J 66:A209-Tu-Pos402, 1994.
    • (1994) Biophys J , vol.66
    • Smith, M.A.1    Conder, M.L.2    Atwal, K.S.3    McCullough, J.R.4
  • 5
    • 0000514610 scopus 로고
    • Characterization of azimilide effects on ion currents of the repolarization phase
    • Zhang Z, Boutjdir M, Brooks RR, Chen L, El-Sherif N. Characterization of azimilide effects on ion currents of the repolarization phase. Biophys J 68:A111-M-Pos485, 1995.
    • (1995) Biophys J , vol.68
    • Zhang, Z.1    Boutjdir, M.2    Brooks, R.R.3    Chen, L.4    El-Sherif, N.5
  • 6
    • 0029163243 scopus 로고
    • Use-dependent effects of the class III antiarrhythmic agent NE-10064 (azimilide) on cardiac repolarization: Block of delayed rectifier potassium and L-type calcium currents
    • Fermini B, Jurkiewicz NK, Jow B, Guinosso PJJ, Baskin EP, Lynch JJJ, Salata JJ. Use-dependent effects of the class III antiarrhythmic agent NE-10064 (azimilide) on cardiac repolarization: Block of delayed rectifier potassium and L-type calcium currents. J Cardiovasc Pharmacol 26:259-271, 1995.
    • (1995) J Cardiovasc Pharmacol , vol.26 , pp. 259-271
    • Fermini, B.1    Jurkiewicz, N.K.2    Jow, B.3    Guinosso, P.J.J.4    Baskin, E.P.5    Lynch, J.J.J.6    Salata, J.J.7
  • 8
    • 0038453740 scopus 로고
    • Pharmacologic identification of IKs in canine ventricular myocytes: Effects of NE-10064 (azimilide)
    • Gintant GA. Pharmacologic identification of IKs in canine ventricular myocytes: Effects of NE-10064 (azimilide). Circulation 90:1-146-0781, 1994.
    • (1994) Circulation , vol.90
    • Gintant, G.A.1
  • 9
    • 0028208260 scopus 로고
    • Comparison of the cardiac electrophysiologic effects of NE-10064 with sotalol and E-4031 and their modification by simulated ischaemia
    • Mcintosh MA, Tanira M, Pacini D, Kane KA. Comparison of the cardiac electrophysiologic effects of NE-10064 with sotalol and E-4031 and their modification by simulated ischaemia. J Cardiovasc Pharmacol 23:653-657, 1994.
    • (1994) J Cardiovasc Pharmacol , vol.23 , pp. 653-657
    • Mcintosh, M.A.1    Tanira, M.2    Pacini, D.3    Kane, K.A.4
  • 10
    • 0027381889 scopus 로고
    • Protection against programmed electrical stimulation-induced ventricular tachycardia and sudden cardiac death by NE-10064, a class III antiarrhythmic drug
    • Black SC, Butterfield JL, Lucchesi BR. Protection against programmed electrical stimulation-induced ventricular tachycardia and sudden cardiac death by NE-10064, a class III antiarrhythmic drug. J Cardiovasc Pharmacol 22:810-818, 1993.
    • (1993) J Cardiovasc Pharmacol , vol.22 , pp. 810-818
    • Black, S.C.1    Butterfield, J.L.2    Lucchesi, B.R.3
  • 11
    • 0024339647 scopus 로고
    • Broad sensitivity of rodent arrhythmia models to class I, II, III, and IV antiarrhythmic agents
    • Brooks RR, Miller KE, Carpenter JF, Jones SM. Broad sensitivity of rodent arrhythmia models to class I, II, III, and IV antiarrhythmic agents. Proc Soc Exp Biol Med 191:201-208, 1989.
    • (1989) Proc Soc Exp Biol Med , vol.191 , pp. 201-208
    • Brooks, R.R.1    Miller, K.E.2    Carpenter, J.F.3    Jones, S.M.4
  • 12
    • 3042920501 scopus 로고
    • Efficacy of a novel class III antiarrhythmic agent NE-10064 against ischemia/reperfusion arrhythmias in rats
    • Brooks RR, Carpenter JF, Maynard AE, Decker GE. Efficacy of a novel class III antiarrhythmic agent NE-10064 against ischemia/reperfusion arrhythmias in rats. FASEB J 7:A97-557, 1993.
    • (1993) FASEB J , vol.7
    • Brooks, R.R.1    Carpenter, J.F.2    Maynard, A.E.3    Decker, G.E.4
  • 13
    • 0344310195 scopus 로고
    • The class III antiarrhythmic NE-10064 suppresses ouabain-induced arrhythmias in guinea pigs
    • Miller KE, Decker GE, Brittain D, Carpenter JF, Brooks RR. The class III antiarrhythmic NE-10064 suppresses ouabain-induced arrhythmias in guinea pigs. Can J Physiol Pharmacol 72(Suppl 1):82-01.1.20, 1994.
    • (1994) Can J Physiol Pharmacol , vol.72 , Issue.1 SUPPL.
    • Miller, K.E.1    Decker, G.E.2    Brittain, D.3    Carpenter, J.F.4    Brooks, R.R.5
  • 14
    • 0014266599 scopus 로고
    • Antiarrhythmic activity of some isoquinoline derivatives determined by a rapid screening procedure in the mouse
    • Lawson JW. Antiarrhythmic activity of some isoquinoline derivatives determined by a rapid screening procedure in the mouse. J Pharmacol Exp Ther 160:22-31, 1968.
    • (1968) J Pharmacol Exp Ther , vol.160 , pp. 22-31
    • Lawson, J.W.1
  • 15
    • 0021690255 scopus 로고
    • Ischemia and reperfusion-induced arrhythmias in the rat. Effects of xanthine oxidase inhibition with allopurinol
    • Manning AS, Coltart DJ, Hearse DJ. Ischemia and reperfusion-induced arrhythmias in the rat. Effects of xanthine oxidase inhibition with allopurinol. Circ Res 55:545-548, 1984.
    • (1984) Circ Res , vol.55 , pp. 545-548
    • Manning, A.S.1    Coltart, D.J.2    Hearse, D.J.3
  • 16
    • 0020655627 scopus 로고
    • Reperfusion-induced cardiac arrhythmias in the anesthetized rat and their susceptibility to drugs
    • Kane KA, Paratt JR, Williams EM. Reperfusion-induced cardiac arrhythmias in the anesthetized rat and their susceptibility to drugs. Br J Pharmacol 78:122P, 1984.
    • (1984) Br J Pharmacol , vol.78
    • Kane, K.A.1    Paratt, J.R.2    Williams, E.M.3
  • 17
    • 84961058932 scopus 로고
    • Simple techniques for the surgical occlusion of coronary vessels in the rat
    • Selye H, Bajusz E, Grasso S, Mendell P. Simple techniques for the surgical occlusion of coronary vessels in the rat. Angiol 11:398-407, 1960.
    • (1960) Angiol , vol.11 , pp. 398-407
    • Selye, H.1    Bajusz, E.2    Grasso, S.3    Mendell, P.4
  • 18
    • 85047679058 scopus 로고
    • The Lambeth Conventions: Guidelines for the study of arrhythmias in ischaemia, infarction, and reperfusion
    • Walker MJA, Curtis MJ, Hearse DJ, et al. The Lambeth Conventions: Guidelines for the study of arrhythmias in ischaemia, infarction, and reperfusion. Cardiovasc Res 22:447-455, 1988.
    • (1988) Cardiovasc Res , vol.22 , pp. 447-455
    • Walker, M.J.A.1    Curtis, M.J.2    Hearse, D.J.3
  • 19
    • 0018173865 scopus 로고
    • Ventricular arrhythmias associated with coronary artery occlusion and reperfusion in the isolated perfused rat heart: A model for assessment of antifibrillatory action of antiarrhythmic agents
    • Lubbe WF, Daries PS, Opie LH. Ventricular arrhythmias associated with coronary artery occlusion and reperfusion in the isolated perfused rat heart: A model for assessment of antifibrillatory action of antiarrhythmic agents. Cardiovasc Res 12:212-220, 1978.
    • (1978) Cardiovasc Res , vol.12 , pp. 212-220
    • Lubbe, W.F.1    Daries, P.S.2    Opie, L.H.3
  • 20
    • 0021046531 scopus 로고
    • Responses to ligation of a coronary artery in conscious rats and the actions of antiarrhythmics
    • Johnston KM, MacLeod BA, Walker MJA. Responses to ligation of a coronary artery in conscious rats and the actions of antiarrhythmics. Can J Physiol Pharmacol 61:1340-1353, 1983.
    • (1983) Can J Physiol Pharmacol , vol.61 , pp. 1340-1353
    • Johnston, K.M.1    MacLeod, B.A.2    Walker, M.J.A.3
  • 21
    • 0023624425 scopus 로고
    • Effects of nicainoprol on reperfusion arrhythmia in the isolated working rat heart and on ischemia and reperfusion arrhythmia and myocardial infarct size in the anesthetized rat
    • Martorana PA, Linz W, Göbel H, Petry P, Schölkens BA. Effects of nicainoprol on reperfusion arrhythmia in the isolated working rat heart and on ischemia and reperfusion arrhythmia and myocardial infarct size in the anesthetized rat. Eur J Pharmacol 143:391-401, 1987.
    • (1987) Eur J Pharmacol , vol.143 , pp. 391-401
    • Martorana, P.A.1    Linz, W.2    Göbel, H.3    Petry, P.4    Schölkens, B.A.5
  • 22
    • 0020428775 scopus 로고
    • Ouabain-induced tachyarrhythmias and cell damage in isolated perfused guinea-pig hearts: I. Protection by propranolol
    • Tanz RD, Russell NJ, Banerian SP, Sharp VH. Ouabain-induced tachyarrhythmias and cell damage in isolated perfused guinea-pig hearts: I. Protection by propranolol. J Mol Cell Cardiol 14:655-671, 1982.
    • (1982) J Mol Cell Cardiol , vol.14 , pp. 655-671
    • Tanz, R.D.1    Russell, N.J.2    Banerian, S.P.3    Sharp, V.H.4
  • 23
    • 0017161183 scopus 로고
    • Cardiac Na,K-ATPase activity during positive inotropic and toxic actions of ouabain
    • Rhee HM, Dutta S, Marks BH. Cardiac Na,K-ATPase activity during positive inotropic and toxic actions of ouabain. Eur J Pharmacol 37:141-153, 1976.
    • (1976) Eur J Pharmacol , vol.37 , pp. 141-153
    • Rhee, H.M.1    Dutta, S.2    Marks, B.H.3
  • 24
    • 3042923195 scopus 로고
    • The effects of pronethalol, dichloroisoprenaline and disopyramide on the toxicity to the heart of ouabain and anaesthetics
    • Sekiya A, Vaughan Williams EM. The effects of pronethalol, dichloroisoprenaline and disopyramide on the toxicity to the heart of ouabain and anaesthetics. Br J Anaesth 21:462-472, 1963.
    • (1963) Br J Anaesth , vol.21 , pp. 462-472
    • Sekiya, A.1    Vaughan Williams, E.M.2
  • 25
    • 0028001747 scopus 로고
    • Release of adenine nucleotide metabolites by toxic concentrations of cardiac glycosides
    • Bernauer W. Release of adenine nucleotide metabolites by toxic concentrations of cardiac glycosides. Basic Res Cardiol 89:308-321, 1994.
    • (1994) Basic Res Cardiol , vol.89 , pp. 308-321
    • Bernauer, W.1
  • 26
    • 0029045235 scopus 로고
    • Digoxin-induced ventricular arrhythmias in the guinea pig heart in vivo: Evidence for a role of endogenous catecholamines in the genesis of delayed afterdepolarizations and triggered activity
    • Xu J, Hurt CM, Pelleg A. Digoxin-induced ventricular arrhythmias in the guinea pig heart in vivo: Evidence for a role of endogenous catecholamines in the genesis of delayed afterdepolarizations and triggered activity. Heart Vessels 10:119-127, 1995.
    • (1995) Heart Vessels , vol.10 , pp. 119-127
    • Xu, J.1    Hurt, C.M.2    Pelleg, A.3
  • 27
    • 0026463632 scopus 로고
    • Effects of cyclooxygenase and lipoxygenase inhibitors on digoxin-induced arrhythmias and haemodynamics in guinea-pigs
    • Kanzik I, Çakici I, Ersoy S, Ark M, Abacioglu N, Zengil H. Effects of cyclooxygenase and lipoxygenase inhibitors on digoxin-induced arrhythmias and haemodynamics in guinea-pigs. Pharmacol Res 26:305-316, 1992.
    • (1992) Pharmacol Res , vol.26 , pp. 305-316
    • Kanzik, I.1    Çakici, I.2    Ersoy, S.3    Ark, M.4    Abacioglu, N.5    Zengil, H.6
  • 28
    • 0002108525 scopus 로고
    • NE-10064 exhibits class III antiarrhythmic effects after intravenous or oral administration in conscious dogs
    • Brandt MA, Maynard AE. NE-10064 exhibits class III antiarrhythmic effects after intravenous or oral administration in conscious dogs. FASEB J 8:A7-38, 1994.
    • (1994) FASEB J , vol.8
    • Brandt, M.A.1    Maynard, A.E.2
  • 29
    • 0014502322 scopus 로고
    • A critical evaluation of three methods for the study of adrenergic beta-blocking and anti-arrhythmic agents
    • Vargaftig B, Coignet JL. A critical evaluation of three methods for the study of adrenergic beta-blocking and anti-arrhythmic agents. Eur J Pharmacol 6:49-55, 1969.
    • (1969) Eur J Pharmacol , vol.6 , pp. 49-55
    • Vargaftig, B.1    Coignet, J.L.2
  • 30
    • 0019861030 scopus 로고
    • Prevention of chloroform-induced ventricular tachycardia in mice as an index of antiarrhythmic activity
    • Block AJ. Prevention of chloroform-induced ventricular tachycardia in mice as an index of antiarrhythmic activity. Life Sci 28:2623-2629, 1981.
    • (1981) Life Sci , vol.28 , pp. 2623-2629
    • Block, A.J.1
  • 31
    • 0000827357 scopus 로고
    • Binding profile of NE-10064, a novel class III antiarrhythmic agent, to rat brain receptors
    • Pong SF, Kinney CM, Moorehead TJ. Binding profile of NE-10064, a novel class III antiarrhythmic agent, to rat brain receptors. FASEB J 7:A474-2748, 1993.
    • (1993) FASEB J , vol.7
    • Pong, S.F.1    Kinney, C.M.2    Moorehead, T.J.3
  • 32
    • 3042952316 scopus 로고
    • β-Adrenergic effects of the class III antiarrhythmic agent NE-10064 in the isolated perfused guinea pig heart
    • Miller KE, Carpenter JF, Brooks RR. β-Adrenergic effects of the class III antiarrhythmic agent NE-10064 in the isolated perfused guinea pig heart. FASEB J 7:A108-620, 1993.
    • (1993) FASEB J , vol.7
    • Miller, K.E.1    Carpenter, J.F.2    Brooks, R.R.3
  • 33
    • 0021132403 scopus 로고
    • Methods for the detection and assessment of antiarrhythmic activity
    • Winslow E. Methods for the detection and assessment of antiarrhythmic activity. Pharmacol Ther 24:401-433, 1984.
    • (1984) Pharmacol Ther , vol.24 , pp. 401-433
    • Winslow, E.1
  • 34
    • 0025740845 scopus 로고
    • + currents in isolated adult rat ventricular myocytes
    • + currents in isolated adult rat ventricular myocytes. J Gen Physiol 97:973-1011, 1991.
    • (1991) J Gen Physiol , vol.97 , pp. 973-1011
    • Apkon, M.1    Nerbonne, J.M.2
  • 35
    • 0027225392 scopus 로고
    • Ionic currents and action potentials in rabbit, rat, and guinea pig ventricular myocytes
    • Varro A, Lathrop DA, Hester SB, Nanasi PP, Papp JG. Ionic currents and action potentials in rabbit, rat, and guinea pig ventricular myocytes. Basic Res Cardiol 88:93-102, 1993.
    • (1993) Basic Res Cardiol , vol.88 , pp. 93-102
    • Varro, A.1    Lathrop, D.A.2    Hester, S.B.3    Nanasi, P.P.4    Papp, J.G.5
  • 36
    • 0025864092 scopus 로고
    • Pretranslational mechanisms determine the type of potassium channels expressed in the rat skeletal and cardiac muscles
    • Matsubara H, Liman ER, Hess P, Koren G. Pretranslational mechanisms determine the type of potassium channels expressed in the rat skeletal and cardiac muscles. J Biol Chem 266:13324-13328, 1991.
    • (1991) J Biol Chem , vol.266 , pp. 13324-13328
    • Matsubara, H.1    Liman, E.R.2    Hess, P.3    Koren, G.4
  • 37
    • 0028003753 scopus 로고
    • + channel gene expression in ventricle of rat heart
    • + channel gene expression in ventricle of rat heart. Circ Res 75:1006-1013, 1994.
    • (1994) Circ Res , vol.75 , pp. 1006-1013
    • Takimoto, K.1    Levitan, E.S.2
  • 38
    • 0028018183 scopus 로고
    • Time course of postnatal changes in rat heart action potential and in transient outward current is different
    • Wahler GM, Dollinger SJ, Smith JM, Flemal KL. Time course of postnatal changes in rat heart action potential and in transient outward current is different. Am J Physiol 267:H1157-H1166, 1994.
    • (1994) Am J Physiol , vol.267
    • Wahler, G.M.1    Dollinger, S.J.2    Smith, J.M.3    Flemal, K.L.4
  • 39
    • 0027192173 scopus 로고
    • Actions and interactions of E-4031 and tedisamil on reperfusion-induced arrhythmias and QT interval in rat in vivo
    • Bril A, Landais L, Gout B. Actions and interactions of E-4031 and tedisamil on reperfusion-induced arrhythmias and QT interval in rat in vivo. Cardiovasc Drugs Ther 7:233-240, 1993.
    • (1993) Cardiovasc Drugs Ther , vol.7 , pp. 233-240
    • Bril, A.1    Landais, L.2    Gout, B.3
  • 40
    • 0027132962 scopus 로고
    • Inwardly rectifying potassium current in rat fetal and neonatal ventricular cardiomyocytes
    • Masuda H, Sperelakis N. Inwardly rectifying potassium current in rat fetal and neonatal ventricular cardiomyocytes. Am J Physiol 265:H1107-H1111, 1993.
    • (1993) Am J Physiol , vol.265
    • Masuda, H.1    Sperelakis, N.2
  • 41
    • 0027339835 scopus 로고
    • Selective IK blockade as an antiarrhythmic mechanism: Effects of UK66.914 on ischaemia and reperfusion arrhythmias in rat and rabbit hearts
    • Rees SA, Curtis MJ. Selective IK blockade as an antiarrhythmic mechanism: Effects of UK66.914 on ischaemia and reperfusion arrhythmias in rat and rabbit hearts. Br J Pharmacol 108:139-145, 1993.
    • (1993) Br J Pharmacol , vol.108 , pp. 139-145
    • Rees, S.A.1    Curtis, M.J.2
  • 43
    • 0020606072 scopus 로고
    • Mechanism of cardiac glycoside-induced toxicity: Physiology, biochemistry, and electron microscopy
    • Tanz RD, Russell NJ. Mechanism of cardiac glycoside-induced toxicity: Physiology, biochemistry, and electron microscopy. Fed Proc 42:2470-2474, 1983.
    • (1983) Fed Proc , vol.42 , pp. 2470-2474
    • Tanz, R.D.1    Russell, N.J.2
  • 44
    • 0016681721 scopus 로고
    • Effect of beta receptor blockade on the initiation and perpetuation of ouabain-induced ventricular tachyarrhythmia
    • Apantaku FO, Baumgarten CM, Ten Eick RE. Effect of beta receptor blockade on the initiation and perpetuation of ouabain-induced ventricular tachyarrhythmia. J Pharmacol Exp Ther 193:327-335, 1975.
    • (1975) J Pharmacol Exp Ther , vol.193 , pp. 327-335
    • Apantaku, F.O.1    Baumgarten, C.M.2    Ten Eick, R.E.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.