Conformationally restrained β-blocking oxime ethers. 3. Synthesis and β-adrenergic antagonistic activity of diastereomeric anti and syn 2-(5′-(3′-methyl)isoxazolidinyl)-N-alkylethanolamines

European Journal of Medicinal Chemistry

Volumn 31, Issue 2, 1996, Pages 159-163

  Breschi, M C ^a   Macchia, M ^a   Manera, C ^a   Micali, E ^a   Nardini, C ^a   Nencetti, S ^a   Rossello, A ^a   Scatizzi, R ^a  

^a UNIVERSITY OF PISA   (Italy)

Author keywords

2 (5 isoxazolidinyl)ethanolamine; Adrenergic drug; blocking agent

Indexed keywords

BETA 1 ADRENERGIC RECEPTOR; BETA 2 ADRENERGIC RECEPTOR; BETA ADRENERGIC RECEPTOR BLOCKING AGENT; DICHLORISOPRENALINE; ETHANOLAMINE DERIVATIVE; ISOPRENALINE; ISOXAZOLIDINE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; GUINEA PIG; HEART ATRIUM; MALE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; STEREOCHEMISTRY; STRUCTURE ACTIVITY RELATION; TRACHEA;

EID: 0029874896     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/0223-5234(96)80449-1     Document Type: Article

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