Necessity of dual blockade of endothelin ETA and ETB receptor subtypes for antagonism of endothelin-1-induced contraction in human bronchi

British Journal of Pharmacology

Volumn 117, Issue 6, 1996, Pages 995-999

  Fukuroda, Takahiro ^a   Ozaki, Satoshi ^a   Ihara, Masaki ^a   Ishikawa, Kiyofumi ^a   Yano, Mitsuo ^a   Miyauchi, Takashi ^b   Ishikawa, Shigemi ^b   Onizuka, Masataka ^b   Goto, Katsutoshi ^b   Nishikibe, Masaru ^a  

^a BANYU PHARMACEUTICAL CO LTD   (Japan)

^b UNIVERSITY OF TSUKUBA   (Japan)

Author keywords

BQ 123; BQ 788; BQ 928; Bronchi (human); Endothelin 1; ETA receptors; ETB receptors; Sarafotoxin S6c

Indexed keywords

CYCLO(DEXTRO TRYPTOPHYL DEXTRO ASPARTYLPROLYL DEXTRO VALYLLEUCYL); ENDOTHELIN 1; ENDOTHELIN A RECEPTOR; ENDOTHELIN B RECEPTOR; N (2,6 DIMETHYLPIPERIDINOCARBONYL) 4 METHYLLEUCYL DEXTRO (1 METHOXYCARBONYLTRYPTOPHANYL) DEXTRO NORLEUCINE; RECEPTOR SUBTYPE; SARAFOTOXIN S6C;

ADULT; AGED; ARTICLE; BRONCHOSPASM; BRONCHUS MUSCLE; CLINICAL ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; FEMALE; HUMAN; HUMAN TISSUE; MALE; MEMBRANE BINDING; OBSTRUCTIVE AIRWAY DISEASE; PRIORITY JOURNAL; RECEPTOR BLOCKING;

ADULT; AGED; AGED, 80 AND OVER; BRONCHI; BRONCHOCONSTRICTION; ENDOTHELINS; FEMALE; HUMANS; MALE; MIDDLE AGED; OLIGOPEPTIDES; PEPTIDES, CYCLIC; PIPERIDINES; RECEPTOR, ENDOTHELIN A; RECEPTOR, ENDOTHELIN B; RECEPTORS, ENDOTHELIN;

EID: 0029866739     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1476-5381.1996.tb16688.x     Document Type: Article

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