Crystal receptor models in medicinal chemistry: Application to the generation of highly potent potassium channel openers

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 7, 1996, Pages 913-918

  Russell, Keith ^a  

^a ASTRAZENECA   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

CROMAKALIM; POTASSIUM CHANNEL; POTASSIUM CHANNEL STIMULATING AGENT;

ARTICLE; COMPUTER SIMULATION; DRUG DESIGN; MOLECULAR MODEL; STRUCTURE ACTIVITY RELATION;

EID: 0029864830     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0960-894X(96)00143-6     Document Type: Article

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12. 50 of 0.6 μM in this assay.
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