메뉴 건너뛰기




Volumn 21, Issue 3, 1996, Pages 339-345

Metrifonate and dichlorvos: Effects of a single oral administration on cholinesterase activity in rat brain and blood

Author keywords

Alzheimer's disease; blood; cholinesterase inhibition; dichlorvos; in vivo; metrifonate; oral administration; rat, brain

Indexed keywords

CHOLINESTERASE; CHOLINESTERASE INHIBITOR; DICHLORVOS; METRIFONATE;

EID: 0029863987     PISSN: 03643190     EISSN: None     Source Type: Journal    
DOI: 10.1007/BF02531650     Document Type: Article
Times cited : (43)

References (40)
  • 1
    • 0022506213 scopus 로고
    • Rates of senile dementia, Alzheimer's type, in the Baltimore Longitudinal Study
    • Sayetta, R. B. 1986. Rates of senile dementia, Alzheimer's type, in the Baltimore Longitudinal Study. J. Chronic Dis. 4:271-286.
    • (1986) J. Chronic Dis. , vol.4 , pp. 271-286
    • Sayetta, R.B.1
  • 2
    • 0025072966 scopus 로고
    • The politics of Alzheimer's disease: A case study in apocalyptic demography
    • Robertson, A. 1990. The politics of Alzheimer's disease: a case study in apocalyptic demography. Int. J. Health Serv. 20:429-442.
    • (1990) Int. J. Health Serv. , vol.20 , pp. 429-442
    • Robertson, A.1
  • 3
    • 0011162190 scopus 로고
    • Selective loss of central cholinergic neurons in Alzheimer's disease
    • Davies, P., and Maloney, A. 1976. Selective loss of central cholinergic neurons in Alzheimer's disease. Lancet 2:1403.
    • (1976) Lancet , vol.2 , pp. 1403
    • Davies, P.1    Maloney, A.2
  • 4
    • 0020072221 scopus 로고
    • Alzheimer's disease and senile dementia: Loss of neurons in the basal forebrain
    • Whitehouse P. J., Price, D. L., Struble, R. G., Clark, A. W. Coyle J. T., and Delong, M. R. 1982. Alzheimer's disease and senile dementia: loss of neurons in the basal forebrain. Science 215: 1237-1239.
    • (1982) Science , vol.215 , pp. 1237-1239
    • Whitehouse, P.J.1    Price, D.L.2    Struble, R.G.3    Clark, A.W.4    Coyle, J.T.5    Delong, M.R.6
  • 5
    • 0018078940 scopus 로고
    • Correlation of cholinergic abnormalities with senile plaques and mental test scores in senile dementia
    • Perry, E. K., Tomlinson, E., Blessed, G., Bergmann, K., Gibson, P. H., and Perry, R. H. 1978. Correlation of cholinergic abnormalities with senile plaques and mental test scores in senile dementia. Br. J. Med. 42:1457-1459.
    • (1978) Br. J. Med. , vol.42 , pp. 1457-1459
    • Perry, E.K.1    Tomlinson, E.2    Blessed, G.3    Bergmann, K.4    Gibson, P.H.5    Perry, R.H.6
  • 6
    • 84886617908 scopus 로고
    • Pre- and postsynaptic neurochemical alterations in Alzheimer's disease
    • Reisine, T., Yamamura, H. I., Bird, E. D., Spokes, E., and Enna, S. J. 1978. Pre- and postsynaptic neurochemical alterations in Alzheimer's disease. Brain Res. 159:477-481.
    • (1978) Brain Res. , vol.159 , pp. 477-481
    • Reisine, T.1    Yamamura, H.I.2    Bird, E.D.3    Spokes, E.4    Enna, S.J.5
  • 7
    • 0024314648 scopus 로고
    • A brain regional analysis of morphologic and cholinergic abnormalities in Alzheimer's disease
    • Zubenko, G. S., Moossey, J., Martinez, A. J., Rao, G. R., Kopp, U., and Hanin, I. 1989. A brain regional analysis of morphologic and cholinergic abnormalities in Alzheimer's disease. Arch. Neurol. 46:634-638.
    • (1989) Arch. Neurol. , vol.46 , pp. 634-638
    • Zubenko, G.S.1    Moossey, J.2    Martinez, A.J.3    Rao, G.R.4    Kopp, U.5    Hanin, I.6
  • 8
    • 0021962590 scopus 로고
    • Loss of M2 muscarinic receptors in the cerebral cortex in Alzheimer's disease and experimental cholinergic denervation
    • Mash, D. C., Flynn, D. D., and Potter, L. T. 1985. Loss of M2 muscarinic receptors in the cerebral cortex in Alzheimer's disease and experimental cholinergic denervation. Science 228:1115-1117.
    • (1985) Science , vol.228 , pp. 1115-1117
    • Mash, D.C.1    Flynn, D.D.2    Potter, L.T.3
  • 9
    • 0023818217 scopus 로고
    • Reductions in 3H-nicotinic acetylcholine binding in Alzheimer's disease and Parkinson's disease - An autoradiographic study
    • Whitehouse, P. J., Martino, A. M., Wagster, M. V., Price, D. L., Mayeux, R., Atack, J. R., and Kellar, K. J. 1988. Reductions in 3H-nicotinic acetylcholine binding in Alzheimer's disease and Parkinson's disease - an autoradiographic study. Neurology 38: 720-723.
    • (1988) Neurology , vol.38 , pp. 720-723
    • Whitehouse, P.J.1    Martino, A.M.2    Wagster, M.V.3    Price, D.L.4    Mayeux, R.5    Atack, J.R.6    Kellar, K.J.7
  • 10
    • 0024810785 scopus 로고
    • The cholinergic receptor system of the human brain. Neurochemical and pharmacological aspects in aging and Alzheimer's disease
    • Nordberg, A. (ed.), Elsevier, Amsterdam
    • Giacobini, E., DeSarno, P., Clark, B., and McIlhany, M. 1989. The cholinergic receptor system of the human brain. Neurochemical and pharmacological aspects in aging and Alzheimer's disease. Pages 335-343, in Nordberg, A. (ed.), Progress in Brain Research, Elsevier, Amsterdam.
    • (1989) Progress in Brain Research , pp. 335-343
    • Giacobini, E.1    DeSarno, P.2    Clark, B.3    McIlhany, M.4
  • 11
    • 0019223566 scopus 로고
    • Acetylcholine and choline levels in post-mortem human brain tissue: Preliminary observations in Alzheimer's disease
    • Richter, J. A., Perry, E. K., and Tomlinson, B. E. 1980. Acetylcholine and choline levels in post-mortem human brain tissue: preliminary observations in Alzheimer's disease. Life Sci. 26: 1683-1689.
    • (1980) Life Sci. , vol.26 , pp. 1683-1689
    • Richter, J.A.1    Perry, E.K.2    Tomlinson, B.E.3
  • 13
    • 0024465639 scopus 로고
    • Clinical pharmacology of tetrahydroaminoacridine: A possible therapeutic agent for Alzheimer's disease
    • Kumar, V., and Becker, R. E. 1989. Clinical pharmacology of tetrahydroaminoacridine: a possible therapeutic agent for Alzheimer's disease. Int. J. Clin. Pharmacol. Ther. Toxicol. 27:478-485.
    • (1989) Int. J. Clin. Pharmacol. Ther. Toxicol. , vol.27 , pp. 478-485
    • Kumar, V.1    Becker, R.E.2
  • 14
    • 33746140058 scopus 로고
    • Clinical pharmacology of aminoacridines in Alzheimer's disease
    • Schneider, L. S. 1993. Clinical pharmacology of aminoacridines in Alzheimer's disease. Neurology 43:64-79.
    • (1993) Neurology , vol.43 , pp. 64-79
    • Schneider, L.S.1
  • 15
    • 0022230177 scopus 로고
    • Efficacy of oral physostigmine in primary degenerative dementia. a double blind study of response to different dose levels
    • Suha, A., Beller, S. A., Overall, J. E., and Swann, A. C. 1985. Efficacy of oral physostigmine in primary degenerative dementia. A double blind study of response to different dose levels. Psychopharmacology 87:147-151.
    • (1985) Psychopharmacology , vol.87 , pp. 147-151
    • Suha, A.1    Beller, S.A.2    Overall, J.E.3    Swann, A.C.4
  • 16
    • 0023920818 scopus 로고
    • Potential pharmacotherapy of Alzheimer's disease. A comparison of various forms of physostigmine administration
    • Becker, R. E., Giacobini, E., Elble, R., Mcllhany, M., and Sherman, K. 1988. Potential pharmacotherapy of Alzheimer's disease. A comparison of various forms of physostigmine administration. Acta Neurol. Scand. Suppl. 116:19-32.
    • (1988) Acta Neurol. Scand. Suppl. , vol.116 , pp. 19-32
    • Becker, R.E.1    Giacobini, E.2    Elble, R.3    Mcllhany, M.4    Sherman, K.5
  • 17
    • 0023899578 scopus 로고
    • Mechanisms of cholinesterase inhibition in senile dementia of the Alzheimer type: Clinical, pharmacological, and therapeutic aspects
    • Becker, R. E., and Giacobini, E., 1988. Mechanisms of cholinesterase inhibition in senile dementia of the Alzheimer type: clinical, pharmacological, and therapeutic aspects. Drug Dev. Res. 12: 163-195.
    • (1988) Drug Dev. Res. , vol.12 , pp. 163-195
    • Becker, R.E.1    Giacobini, E.2
  • 18
    • 0002654491 scopus 로고
    • The second generation of cholinesterase inhibitors: Pharmacological aspects
    • Becker, R. and Giacobini, E. (eds.), Birkhauser, Boston
    • Giacobini, E., 1991. The second generation of cholinesterase inhibitors: pharmacological aspects. Pages 247-262, in Becker, R. and Giacobini, E. (eds.), Cholinergic Basis for Alzheimer Therapy, Birkhauser, Boston.
    • (1991) Cholinergic Basis for Alzheimer Therapy , pp. 247-262
    • Giacobini, E.1
  • 19
    • 34447114183 scopus 로고
    • The cholinergic approach in ATD: Focus on international multicentre drug study
    • Spiegel, R., Enz, A., Meier, D., and Emre, M. 1994. The cholinergic approach in ATD: Focus on international multicentre drug study. Neuropsychopharmacology 10:7355.
    • (1994) Neuropsychopharmacology , vol.10 , pp. 7355
    • Spiegel, R.1    Enz, A.2    Meier, D.3    Emre, M.4
  • 21
    • 0002775701 scopus 로고
    • Pharmacodynamics of oral E2020 and tacrine in humans: Novel approaches
    • Becker, R. and Giacobini, E. (eds.), Birkhauser, Boston
    • Sherman, K. A. 1991. Pharmacodynamics of oral E2020 and tacrine in humans: novel approaches. Pages 321-329, in Becker, R. and Giacobini, E. (eds.), Cholinergic Basis for Alzheimer Therapy, Birkhauser, Boston.
    • (1991) Cholinergic Basis for Alzheimer Therapy , pp. 321-329
    • Sherman, K.A.1
  • 22
    • 0018163960 scopus 로고
    • Metrifonate: Summary' of toxicological and pharmacological information available
    • Holmstedt, B., Nordgren, I., Sandoz, M., and Sundwall, A. 1978. Metrifonate: Summary' of toxicological and pharmacological information available. Arch. Toxicol. 41:3-29.
    • (1978) Arch. Toxicol. , vol.41 , pp. 3-29
    • Holmstedt, B.1    Nordgren, I.2    Sandoz, M.3    Sundwall, A.4
  • 23
    • 0016852324 scopus 로고
    • Mechanism of inhibition in vitro of mammalian acetylcholinesterase and cholinesterase in solutions of 0,0-dimethyl 2,2,2-trichloro-1-hydroxyethyl phosphonate (Trichlorfon)
    • Reiner, E., Krauthacker, B., Simeon, V., and Skrinjaric-Spoljar, M, 1975. Mechanism of inhibition in vitro of mammalian acetylcholinesterase and cholinesterase in solutions of 0,0-dimethyl 2,2,2-trichloro-1-hydroxyethyl phosphonate (Trichlorfon). Biochem. Pharmacol. 24:717-722.
    • (1975) Biochem. Pharmacol. , vol.24 , pp. 717-722
    • Reiner, E.1    Krauthacker, B.2    Simeon, V.3    Skrinjaric-Spoljar, M.4
  • 28
    • 0029610697 scopus 로고
    • Effects of metrifonate and tacrine in the spatial Morris maze task and modified Irwin test: Evaluation of the efficacy/safety profile in rats
    • in press
    • Blokland, A., Hinz, V., and Schmidt, B. 1995. Effects of metrifonate and tacrine in the spatial Morris maze task and modified Irwin test: Evaluation of the efficacy/safety profile in rats. Drug Dev. Res.: in press.
    • (1995) Drug Dev. Res.
    • Blokland, A.1    Hinz, V.2    Schmidt, B.3
  • 29
    • 0025563812 scopus 로고
    • Effect of acute and chronic cholinesterase inhibition on biogenic amines in rat brain
    • Soininen, H. S., Unni, I., and Shillcutt, S. 1990. Effect of acute and chronic cholinesterase inhibition on biogenic amines in rat brain. Neurochem. Res. 15:1185-1190.
    • (1990) Neurochem. Res. , vol.15 , pp. 1185-1190
    • Soininen, H.S.1    Unni, I.2    Shillcutt, S.3
  • 30
    • 0024589925 scopus 로고
    • Physostigmine, tacrine and metrifonate: The effect of multiple doses on acetylcholine metabolism in rat brain
    • Hallak, M., and Giacobini, E. 1989. Physostigmine, tacrine and metrifonate: the effect of multiple doses on acetylcholine metabolism in rat brain. Neuropharmacol. 28:199-206.
    • (1989) Neuropharmacol. , vol.28 , pp. 199-206
    • Hallak, M.1    Giacobini, E.2
  • 31
    • 0019836429 scopus 로고
    • Metrifonate in schistosomiasis-therapy and prophylaxis
    • Jewsbury, J. M. 1981. Metrifonate in schistosomiasis-therapy and prophylaxis. Acta Pharmacol. Toxicol. 49:123-130.
    • (1981) Acta Pharmacol. Toxicol. , vol.49 , pp. 123-130
    • Jewsbury, J.M.1
  • 32
    • 34447114347 scopus 로고
    • Metrifonate induces cholinesterase inhibition exclusively via slow release of dichlorvos
    • Hinz, V. C., Grewig, S., and Schmidt, B. H. 1995. Metrifonate induces cholinesterase inhibition exclusively via slow release of dichlorvos. Naunyn Schmiedeberg's Arch. Pharmacol. 351(S): R135.
    • (1995) Naunyn Schmiedeberg's Arch. Pharmacol. , vol.351 , Issue.S
    • Hinz, V.C.1    Grewig, S.2    Schmidt, B.H.3
  • 33
    • 0018731624 scopus 로고
    • Mode of action of anticholinesterases
    • Main, A. R. 1979. Mode of action of anticholinesterases. Pharmacol. Ther. 6:579-628.
    • (1979) Pharmacol. Ther. , vol.6 , pp. 579-628
    • Main, A.R.1
  • 34
    • 0016758710 scopus 로고
    • Dichlorvos and the cholinergic system: Effects on cholinesterase and acetylcholinesterase and choline contents of rat tissue
    • Modak, A. T., Stavinoha, W. B., and Weintraub, S. T. 1975. Dichlorvos and the cholinergic system: effects on cholinesterase and acetylcholinesterase and choline contents of rat tissue. Arch. Int. Pharmacodyn. 217:293-301.
    • (1975) Arch. Int. Pharmacodyn. , vol.217 , pp. 293-301
    • Modak, A.T.1    Stavinoha, W.B.2    Weintraub, S.T.3
  • 35
    • 0018650313 scopus 로고
    • Regeneration of cholinesterase activities in humans and rats after inhibition of 0,0-dimethyl 2,2-dichlorovinyl phosphate
    • Reiner, E., and Pleština, R. 1979. Regeneration of cholinesterase activities in humans and rats after inhibition of 0,0-dimethyl 2,2-dichlorovinyl phosphate. Toxicol. Appl. Pharmacol. 49:451-454.
    • (1979) Toxicol. Appl. Pharmacol. , vol.49 , pp. 451-454
    • Reiner, E.1    Pleština, R.2
  • 36
    • 0019767954 scopus 로고
    • Factors modifying the toxicity of organophosphorous compounds including dichlorvos
    • Sterri, S. H. 1981. Factors modifying the toxicity of organophosphorous compounds including dichlorvos. Acta Pharmacol. Toxicol. 49:67-71.
    • (1981) Acta Pharmacol. Toxicol. , vol.49 , pp. 67-71
    • Sterri, S.H.1
  • 37
    • 0016634851 scopus 로고
    • The distribution of dichlorvos in the tissues of mammals after its inhalation or intravenous administration
    • Blair, D., Hoadley, E. C., and Hutson, D. H. 1975. The distribution of dichlorvos in the tissues of mammals after its inhalation or intravenous administration. Toxicol. Appl. Pharmacol. 31:243-253.
    • (1975) Toxicol. Appl. Pharmacol. , vol.31 , pp. 243-253
    • Blair, D.1    Hoadley, E.C.2    Hutson, D.H.3
  • 38
    • 0023226136 scopus 로고
    • A comparison of the effects of two inhibitors on brain cholinesterase
    • Hallak, M., and Giacobini, E. 1987. A comparison of the effects of two inhibitors on brain cholinesterase. Neuropharmacology 26: 521-530.
    • (1987) Neuropharmacology , vol.26 , pp. 521-530
    • Hallak, M.1    Giacobini, E.2
  • 39
    • 0011355206 scopus 로고
    • Studies on the toxicity and mechanism of action of dipterex
    • DuBois, K. P., and Cotter, G. J. 1955. Studies on the toxicity and mechanism of action of dipterex. Arch. Industr. Health 11:53-60.
    • (1955) Arch. Industr. Health , vol.11 , pp. 53-60
    • DuBois, K.P.1    Cotter, G.J.2
  • 40
    • 2642665034 scopus 로고
    • Mode of action of insecticides. Metabolism and selectivity of 0,0-dimethyl 2,2,2-trichloro1-hydroxyethyl phosphonate and its acetyl and vinyl derivatives
    • Arthur, B. W., and Casida, J. E. 1957. Mode of action of insecticides. Metabolism and selectivity of 0,0-dimethyl 2,2,2-trichloro1-hydroxyethyl phosphonate and its acetyl and vinyl derivatives. J. Agric. Food Chem. 5:186-192.
    • (1957) J. Agric. Food Chem. , vol.5 , pp. 186-192
    • Arthur, B.W.1    Casida, J.E.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.