Studies on inhibition of μ and δ opioid receptor binding by dithiothreitol and N-ethylmaleimide: His223 is critical for μopioid receptor binding and inactivation by N-ethylmaleimide

Journal of Biological Chemistry

Volumn 271, Issue 10, 1996, Pages 5505-5512

  Shahrestanifar, Mandana ^a   Wang, William W ^a   Howells, Richard D ^a,b  

^a UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY   (United States)

^b RUTGERS NEW JERSEY MEDICAL SCHOOL   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DELTA OPIATE RECEPTOR; DITHIOTHREITOL; ENKEPHALIN[2 DEXTRO ALANINE 4 METHYLPHENYLALANINE 5 GLYCINE]; ETORPHINE; LEUCINE ENKEPHALIN[2 DEXTRO SERINE 6 THREONINE]; MORPHINE; MU OPIATE RECEPTOR; N ETHYLMALEIMIDE; NALOXONE; OPIATE AGONIST; SODIUM CHLORIDE;

AMINO ACID SUBSTITUTION; ARTICLE; BINDING KINETICS; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; HUMAN; HUMAN CELL; KIDNEY CELL; PRIORITY JOURNAL;

AMINO ACID SEQUENCE; ANALGESICS; BASE SEQUENCE; BINDING SITES; CELL LINE; CELL MEMBRANE; DITHIOTHREITOL; DNA PRIMERS; ENKEPHALIN, ALA(2)-MEPHE(4)-GLY(5)-; ENKEPHALIN, LEUCINE; ENKEPHALINS; ETHYLMALEIMIDE; HISTIDINE; HUMANS; KIDNEY; KINETICS; LIGANDS; MODELS, STRUCTURAL; MOLECULAR SEQUENCE DATA; MUTAGENESIS, SITE-DIRECTED; POINT MUTATION; POLYMERASE CHAIN REACTION; PROTEIN STRUCTURE, SECONDARY; RECEPTORS, OPIOID, DELTA; RECEPTORS, OPIOID, MU; RECOMBINANT FUSION PROTEINS; SERINE; TRANSFECTION;

EID: 0029863220     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.271.10.5505     Document Type: Article

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