A short radiosynthesis of 6-[C3H3]-dorzolamide at very high specific activity and optical purity

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 38, Issue 11, 1996, Pages 963-970

  Eng, W S ^a   Burns, H D ^a   Ponticello, G S ^a   Selnick, H G ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

dorzolamide; methyl iodide; methylation; MK 507; tritium

Indexed keywords

ALKYLATION; METHYLATION; SULFUR COMPOUNDS;

DIASTEREOMERIC; DORZOLAMIDE; HIGH SPECIFIC ACTIVITIES; METHYL IODIDE; MK-507; OPTICAL PURITY; PROTECTING GROUP; RADIOSYNTHESIS; REGIO-SELECTIVE; SULPHONAMIDES;

TRITIUM;

DORZOLAMIDE; TRITIUM;

ARTICLE; DRUG PURIFICATION; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; ISOTOPE LABELING; REACTION ANALYSIS;

TRITIUM;

EID: 0029851407     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199611)38:11<963::AID-JLCR913>3.0.CO;2-W     Document Type: Article

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