Naturally occurring clavines: Antagonism/partial agonism at 5-HT(2A) receptors and antagonism at α1-adrenoceptors in blood vessels

Planta Medica

Volumn 62, Issue 5, 1996, Pages 387-392

  Pertz, H ^a  

^a FREIE UNIVERSITÄT BERLIN   (Germany)

Author keywords

1 adrenoceptors; 5 HT(2A) receptors; antagonism; naturally occurring clavines; partial agonism

Indexed keywords

AGROCLAVINE; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; CLAVINE DERIVATIVE; COCAINE; COSTACLAVINE; DIHYDROLYSERGOL; ELYMOCLAVINE; FESTUCLAVINE; KETANSERIN; LYSERGENE; LYSERGOL; PARTIAL AGONIST; PHENYLEPHRINE; PRAZOSIN; PROPRANOLOL; PYROCLAVINE; SEROTONIN; SEROTONIN 2A AGONIST; SEROTONIN 2A ANTAGONIST; SEROTONIN 2A RECEPTOR; SEROTONIN AGONIST; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BLOOD VESSEL; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG ANTAGONISM; MALE; NONHUMAN; RAT; RECEPTOR AFFINITY; RECEPTOR BINDING; SMOOTH MUSCLE CONTRACTILITY; STRUCTURE ACTIVITY RELATION; TAIL ARTERY; THORACIC AORTA;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMALS; AORTA; ARTERIES; ERGOLINES; MUSCLE CONTRACTION; MUSCLE, SMOOTH, VASCULAR; RATS; RECEPTOR, SEROTONIN, 5-HT2A; RECEPTORS, ADRENERGIC, ALPHA-1; RECEPTORS, SEROTONIN; SEROTONIN; SEROTONIN ANTAGONISTS; STRUCTURE-ACTIVITY RELATIONSHIP;

ANIMALIA;

EID: 0029850871     PISSN: 00320943     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-2006-957922     Document Type: Article

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