Synthesis and activity of pseudotripeptide inhibitors of HIV-1 protease containing D(-)-O-(benzyl)-tartaric acid

Arzneimittel-Forschung/Drug Research

Volumn 46, Issue 11, 1996, Pages 1099-1101

  Marastoni, Mauro ^a   Fantin, Giancarlo ^a   Bortolotti, Fabrizio ^a   Tomatis, Roberto ^a,b  

^a UNIVERSITY OF FERRARA   (Italy)

^b Dipto di Scienze Farmaceutiche   (Italy)

Author keywords

(S,S) O (benzyl)tartaric acid monomethyl esters; HIV 1 protease inhibitor, transition state mimic; pseudopeptides

Indexed keywords

ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; N ACETYLPEPSTATIN; PEPTIDE DERIVATIVE; PROTEINASE INHIBITOR; PSEUDOPEPTIDE; TARTARIC ACID DERIVATIVE; VIRUS ENZYME;

ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME PURIFICATION; HUMAN IMMUNODEFICIENCY VIRUS 1; SPECTROPHOTOMETRY;

AMINO ACIDS; CHEMISTRY, PHYSICAL; HIV PROTEASE INHIBITORS; HIV-1; MAGNETIC RESONANCE SPECTROSCOPY; OLIGOPEPTIDES; STRUCTURE-ACTIVITY RELATIONSHIP; TARTRATES;

EID: 0029850452     PISSN: 00044172     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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