Partial β2-agonists and their impartial assessment

Chest

Volumn 110, Issue 5, 1996, Pages 1131-1132

  Dickey, B F ^a   Clark, R C ^a   Barber, R ^a  

^a MICHAEL E DEBAKEY VETERANS AFFAIRS MEDICAL CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BETA 2 ADRENERGIC RECEPTOR; BETA 2 ADRENERGIC RECEPTOR STIMULATING AGENT; BRONCHODILATING AGENT; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE DIPHOSPHATE; GUANOSINE TRIPHOSPHATE;

ASTHMA; BRONCHODILATATION; DRUG EFFICACY; EDITORIAL; HUMAN; INHALATIONAL DRUG ADMINISTRATION; PRIORITY JOURNAL; RECEPTOR DOWN REGULATION;

EID: 0029848001     PISSN: 00123692     EISSN: None     Source Type: Journal    
DOI: 10.1378/chest.110.5.1131     Document Type: Editorial

References (14)

1. Barrett TE Strom BL. Inhaled beta-adrenergic receptor agonists in asthma: more harm than good? Am J Respir Crit Care Med 151 1995 574 577
2. Kenakin T. Pharmacological analysis of drug-receptor interaction 1993 Raven Press New York
3. Whaley BS Yean Y Birnbaumer L Differential expression of the P-adrenergic receptor modifies agonist stimulation of adenylyl cyclase: a quantitative evaluation Mol Pharmacol 45 1994 481 489
4. 2-adrenergic receptor stimulation of adenylyl cyclase by salmeterol: evidence for quasi-irreversible binding to an exosite Mol Pharmacol 49 1996 182 189
5. Kalra S Swystun VA Bhagat R Inhaled corticosteroids do not prevent the development of tolerance to the bronchoprotective effect of salmeterol Chest 109 1996 953 956
6. Bremner P Siebers R Crane J Partial vs full β-receptor agonism: a clinical study of inhaled albuterol and fenoterol Chest 109 1996 957 962
7. Sears MR. Long-acting β-agonists, tachyphylaxis, and corticosteroids [editorial] Chest 109 1996 862 864
8. 2-adrenergic receptor Science 264 1994 582 586
9. Schutz W Freissmuth M. Reverse intrinsic activity of antagonists on G protein-coupled receptors Trends Pharmacol Sci 13 1992 376 380
10. Barnes PJ. Molecular mechanisms of steroid action in asthma J Allergy Clin Immunol 97 1996 159 168
11. Pearlman DS Chervinsky P LaForce C A comparison of salmeterol with albuterol in the treatment of mild-to-moderate asthma N Engl J Med 327 1992 1420 1425
12. D'Alonzo GE Nathan RA Henochowicz S Salmeterol xinafoate as maintenance therapy compared with albuterol in patients with asthma JAMA 271 1994 1412 1416
13. 2 adrenoceptor agonist/antagonist activity of formoterol and salmeterol Thorax 51 1996 54 58
14. Newhouse MT Chapman KR McCallum AL Cardiovascular safety of high doses of inhaled fenoterol and albuterol in acute severe asthma Chest 110 1996 595 603